Sfoglia per Autore  MACCHIARULO, Antonio

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Titolo Data di pubblicazione Autore(i) File
Pharmacophore Models of Group I and Group II Metabotropic Glutamate Receptors Agonists. Analysis of Conformational, Steric and Topological Parameters Affecting Potency and Selectivity 1999 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Modeling of Amino-Terminal Domains of Group I Metabotropic Glutamate Receptors: Structural Motifs Affecting Ligand Selectivity 1999 Costantino, G.; Pellicciari, Roberto; Macchiarulo, Antonio
Metabotropic Glutamate Receptors: A Structural View Point 2000 Pellicciari, Roberto; Costantino, Gabriele; Macchiarulo, Antonio
Design, Synthesis and Preliminay Evaluation of Novel 3’-Substituted Carboxycyclopropylglycines as Antagonists at Group 2 Metabotropic Glutamate Receptors 2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Amori, L.; Flor, P.; Gasparini, F.; Kuhn, R.; Urwyler, S.
New potent and selective mGluR1 competitive antagonists: pharmacological characterization and their exploitation in molecular modeling of receptor blocking 2001 Costantino, Gabriele; Camaioni, Emidio; Macchiarulo, Antonio; D., Pellegrini Giampietro; F., Moroni; Pellicciari, Roberto
Exploring the Molecular Dasis of the Selectivity in Metabotropic Glutamate Receptors (mGluRs) 2001 Macchiarulo, Antonio; R., Sbaglia; S., Aiello; M., Meniconi; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Pellicciari, Roberto
Metabotropic Glutamate Receptors: Targets for Therapy of Cerebral Ischemia 2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Metabotropic glutamate receptors: structure and new subtype-selective ligands 2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Camaioni, Emidio; Natalini, Benedetto
QSAR and Molecular Modeling Studies of Baclofen Analogues as GABAB Agonists. Insights into the Role of the Aromatic Moiety in GABAB Binding Activation 2001 Costantino, G.; Pellicciari, Roberto; Macchiarulo, Antonio; Entrena Guadix, A.
Conformational analysis of carboxyphenylglycine (CPG) Derivatives: insight into bioactive and bioselective conformations of group-I mGluRs antagonists. 2001 Macchiarulo, Antonio; Entrena Guadix, A.; Costantino, G.
Modeling of Poly(ADP-ribose)polymerase (PARP) Inhibitors. Docking of Ligands and QSAR 2001 Costantino, G.; Macchiarulo, Antonio; Camaioni, Emidio; Pellicciari, Roberto
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1 2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Molecular dynamics simulation of the ligand binding domain of mGluR1 in response to agonist and antagonist binding. 2002 Costantino, Gabriele; Macchiarulo, Antonio; Belenikin, M.; Pellicciari, R.
Molecular determinats for metabotropic glutamate receptor activation and blockade. Molecular dynamics and electrostatic potential analysis studies 2002 Costantino, Gabriele; M., Belenekin; Macchiarulo, Antonio; Camaioni, Emidio; Pellicciari, Roberto
Structure of Metal-Carbenoid Intermediates Derived from the Dirhodium(II)Tetracarboxylate Mediated Decomposition of ?-Diazocarbonyl Compounds. An ab initio and DTF Study 2002 Costantino, G.; Macchiarulo, Antonio; Rovito, R.; Pellicciari, Roberto
Homology Modeling of AMPA Receptors: Route to the identification of noncompetitive antagonists binding site 2002 Barreca, MARIA LETIZIA; Chimirri, A.; Costantino, Gabriele; De Luca, L.; Gitto, R.; Macchiarulo, Antonio; Pellicciari, R.
Spiro[2.2]pentane as a dyssymetric scaffold for conformationally constrained analogues of glutamic acid: diastereodivergent synthesis of 1-aminospiro[2.2]pentyl-1,4-dicarboxylic acids 2002 Marinozzi, Maura; Camaioni, Emidio; Costantino, Gabriele; G., Giorgi; Macchiarulo, Antonio; Pellicciari, Roberto
1,4 Benzothiazine and 1,4 benzoxazine imidazole derivatives with antifungal activity: a docking study 2002 Macchiarulo, Antonio; Costantino, Gabriele; Fringuelli, D.; Vecchiarelli, Anna; Schiaffella, Fausto; Fringuelli, Renata
Glucocorticoid-induced leucine zipper inhibits the Raf-extracellular signal-regulated kinase pathway by binding to Raf-1 2002 Ayroldi, Emira Maria; Zollo, Ornella; Macchiarulo, Antonio; DI MARCO, Barbara; Marchetti, Maria Cristina; Riccardi, Carlo
Glucocorticoid Induced Leucine Zipper (GILZ) inhibits the RAF-ERK pathway by binding to RAF-1 2002 Ayroldi, Emira Maria; Zollo, Ornella; Macchiarulo, Antonio; DI MARCO, Barbara; Marchetti, C; Riccardi, Carlo
Mostrati risultati da 1 a 20 di 251
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