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Discovery of sulfated sterols from marine invertebrates as a new class of marine naturalantagonists of farnesoid-X-receptor. 2011 Sepe, V; Bifulco, G; Renga, Barbara; D'Amore, Claudio; Fiorucci, Stefano; Zampella, A.
Total synthesis and pharmacological characterization of solomonsterol A, a potent marine pregnane-X-receptor agonist endowed with anti-inflammatory activity. 2011 Sepe, V; Ummarino, R; D'Auria, Mv; Mencarelli, Andrea; D'Amore, Claudio; Renga, Barbara; Zampella, A; Fiorucci, Stefano
Farnesoid X receptor suppresses constitutive androstane receptoractivity at the multidrug resistance protein-4 promoter. 2011 Renga, Barbara; Migliorati, M; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Distrutti, Eleonora; Fiorucci, Stefano
Leflunomide protects against dyslipidemia development induced by ritonavir in mice 2011 Baldelli, Franco; A., Mencarelli; Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Schiaroli, Elisabetta; L., Bernini; Francisci, Daniela; Fiorucci, Stefano
The nuclear receptor FXR regulates hepatic transport and metabolism of glutamine and glutamate 2011 Renga, Barbara; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Zampella, A; Monti, Mc; Distrutti, Eleonora; Fiorucci, Stefano
Theonellasterols and conicasterols fromTheonella swinhoei. Novel marine natural ligands for human nuclear receptors. 2011 De Marino, S; Ummarino, R; D'Auria, Mv; Chini, Mg; Bifulco, G; Renga, Barbara; D'Amore, Claudio; Fiorucci, Stefano; Debitus, C; Zampella, A.
Probiotics modulate intestinal expression of nuclear receptor and provide counter-regulatory signals to inflammation-driven adipose tissue activation. 2011 Mencarelli, Andrea; Distrutti, Eleonora; Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Palladino, G; Donini, Annibale; Ricci, Patrizia; Fiorucci, Stefano
SHP-dependent and -independent induction of peroxisomeproliferator-activated receptor-γ by the bile acid sensor farnesoid X receptorcounter-regulates the pro-inflammatory phenotype of liver myofibroblasts. 2011 Renga, Barbara; Mencarelli, Andrea; Migliorati, M; Cipriani, Sabrina; D'Amore, Claudio; Distrutti, Eleonora; Fiorucci, Stefano
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity. 2012 De Marino, S; Ummarino, R; D'Auria, Mv; Chini, Mg; Bifulco, G; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, S; Fiorucci, Stefano; Zampella, A.
HIV-1 infection is associated with changes in nuclear receptor transcriptome, pro-inflammatory and lipid profile of monocytes 2012 Renga, Barbara; Francisci, Daniela; D'Amore, Claudio; Schiaroli, Elisabetta; Carino, A.; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana
VSL#3 Resets Insulin Signaling and Protects against NASH and Atherosclerosis in a Model of Genetic Dyslipidemia and Intestinal Inflammation. 2012 Mencarelli, Andrea; Cipriani, Sabrina; Renga, Barbara; Bruno, A; D'Amore, Claudio; Distrutti, Eleonora; Fiorucci, Stefano
Glucocorticoid receptor mediates the gluconeogenic activity of the farnesoid X receptor in the fasting condition 2012 Renga, Barbara; Mencarelli, Andrea; D'Amore, Claudio; Cipriani, Sabrina; Baldelli, Franco; A., Zampella; Distrutti, Eleonora; Fiorucci, Stefano
Ritonavir-induced lipoatrophy and dyslipidaemia is reversed by the anti-inflammatory drug leflunomide in a PPAR-γ-dependent manner. 2012 Mencarelli, Andrea; Francisci, Daniela; Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Basile, F; Schiaroli, Elisabetta; Baldelli, Franco; Fiorucci, Stefano
The HIV Matrix Protein p17 subverts Nuclear Receptors Expression and induces a STAT1-Dependent Proinflammatory Phenotype in Monocytes 2012 Renga, Barbara; Francisci, Daniela; D'Amore, Claudio; Schiaroli, Elisabetta; Mencarelli, Andrea; Cipriani, Sabrina; Baldelli, Franco; Fiorucci, Stefano
Preliminary structure-activity relationship on theonellasterol, a new chemotype of FXR antagonist, from the marine sponge Theonella swinhoei. 2012 Sepe, V; Ummarino, R; D'Auria, Mv; Taglialatela Scafati, O; Marino, Sd; D'Amore, Claudio; Renga, Barbara; Chini, Mg; Bifulco, G; Nakao, Y; Fusetani, N; Fiorucci, Stefano; Zampella, A.
The Bile Acid Receptor TGR5 Maintains Gastrointestinal Homeostasis and Its Activation Rescues From Gastrointestinal Injury Caused by ASA and NSAIDs 2012 Cipriani, Sabrina; Mencarelli, Andrea; Renga, Barbara; D'Amore, Claudio; Distrutti, Eleonora; Fiorucci, Stefano
Discovery that theonellasterol a marine sponge sterol is a highly selective FXR antagonist that protects against liver injury in cholestasis. 2012 Renga, Barbara; Mencarelli, Andrea; D'Amore, Claudio; Cipriani, Sabrina; D'Auria, Mv; Sepe, V; Chini, Mg; Monti, Mc; Bifulco, G; Zampella, A; Fiorucci, Stefano
a Farnesoid-X-Receptor (FXR)-Glucocorticoid Receptor (GR) Cascade Regulates Intestinal Innate Immunity in Response to FXR Activation 2012 Renga, Barbara; Mencarelli, Andrea; D'Amore, Claudio; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano
Conicasterol E, a Small Heterodimer PartnerSparing Farnesoid X Receptor Modulator Endowed with a Pregnane X ReceptorAgonistic Activity, from the Marine Sponge Theonella swinhoei 2012 Sepe, V; Ummarino, R; D'Auria, Mv; Chini, Mg; Bifulco, G; Renga, Barbara; D'Amore, Claudio; Debitus, C; Fiorucci, Stefano; Zampella, A.
Reciprocal Regulation of TLRS and Nuclear Receptors: IRF-7 Dependent Regulation of FXR Mediates Counter-Regulatory Effects of TLR-9 in Colitis 2012 Renga, Barbara; Mencarelli, A; Cipriani, Sabrina; D'Amore, Claudio; Carino, A; Distrutti, E; Fiorucci, Stefano; Carino, Adriana
Mostrati risultati da 1 a 20 di 48
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