Sfoglia per Autore
HIV-1 infection is associated with changes in nuclear receptor transcriptome, pro-inflammatory and lipid profile of monocytes
2012 Renga, Barbara; Francisci, Daniela; D'Amore, Claudio; Schiaroli, Elisabetta; Carino, A.; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana
The bile acid sensor FXR is required for immune-regulatory activities of TLR-9 in intestinal inflammation
2013 Renga, Barbara; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Carino, A; Bruno, A; Francisci, Daniela; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
FXR mediates a chromatin looping in the GR promoter thus promoting the resolution of colitis in rodents.
2013 Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Mencarelli, Andrea; Carino, A; Sepe, V; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
Solomonsterol A, a marine pregnane-X-receptor agonist, attenuates inflammation and immune dysfunction in a mouse model of arthritis.
2013 Mencarelli, Andrea; D'Amore, Claudio; Renga, Barbara; Cipriani, Sabrina; Carino, A; Sepe, V; Perissutti, E; D'Auria, Mv; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
Exploitation of cholane scaffold for the discovery of potent and selective farnesoid X receptor (FXR) and G-protein coupled bile acid receptor 1 (GP-BAR1) ligands
2014 Festa, C; Renga, Barbara; D'Amore, Claudio; Sepe, V; Finamore, C; De Marino, S; Carino, A.; Cipriani, Sabrina; Monti, Mc; Zampella, A; Fiorucci, Stefano; Carino, Adriana
The HIV Matrix Protein p17 promotes the Activation of human hepatic stellate cells through interactions with CXCR2 and Syndecan-2
2014 Renga, Barbara; Francisci, Daniela; Schiaroli, Elisabetta; Carino, A; Cipriani, Sabrina; D'Amore, Claudio; Sidoni, Angelo; DEL SORDO, Rachele; Ferri, Ivana; Lucattelli, M; Lunghi, B; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana
Structural insights into Estrogen Related Receptor-β modulation: 4-methylenesterols from Theonella swinhoei sponge as the first example of marine natural antagonists.
2014 Di Micco, S; Renga, Barbara; Carino, A; D'Auria, Mv; Zampella, A; Riccio, R; Fiorucci, Stefano; Bifulco, G.; Carino, Adriana
Impaired Itching Perception in Murine Models of Cholestasis Is Supported by Dysregulation of GPBAR1 Signaling
2015 Cipriani, Sabrina; Renga, Barbara; D'Amore, Claudio; Simonetti, M; De Tursi, Aa; Carino, Adriana; Monti, Mc; Sepe, V; Zampella, A; Fiorucci, Stefano
Reversal of Endothelial Dysfunction by GPBAR1 Agonism in Portal Hypertension Involves a AKT/FOXOA1 Dependent Regulation of H2S Generation and Endothelin-1
2015 Renga, B.; Cipriani, S.; Carino, A.; Simonetti, M.; Zampella, A.; Fiorucci, S.
Cystathionine gamma-lyase, a H2S-generating enzyme, is a GPBAR1-regulated gene and contributes to vasodilation caused by secondary bile acids
2015 Renga, Barbara; Bucci, M; Cipriani, Sabrina; Carino, Adriana; Monti, Mc; Zampella, A; Gargiulo, A; d'Emmanuele di Villa Bianca, R; Distrutti, E; Fiorucci, Stefano
The HIV matrix protein p17 induces hepatic lipid accumulation via modulation of nuclear receptor transcriptoma
2015 Renga, Barbara; Francisci, Daniela; Carino, Adriana; Marchianò, Silvia; Cipriani, Sabrina; Chiara Monti, Maria; DEL SORDO, Rachele; Schiaroli, Elisabetta; Distrutti, Eleonora; Baldelli, Franco; Fiorucci, Stefano
Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists
2016 Sepe, V; Festa, C; Renga, B; Carino, A; Cipriani, S; Finamore, C; Masullo, D; Del Gaudio, F; Monti, Mc; Fiorucci, Stefano; Zampella, A.; Carino, Adriana
Navigation in bile acid chemical space: Discovery of novel FXR and GPBAR1 ligands
2016 Finamore, C; Festa, C; Renga, B; Sepe, V; Carino, A; Masullo, D; Biagioli, Michele; Marchianò, S; Capolupo, A; Monti, M; Fiorucci, Stefano; Zampella, A.; Carino, Adriana
A Comprehensive Analysis of Small Heterodimer Partner (SHP) Target Genes in Hepatic Stellate Cells and the Discovery of a New Class of SHP Agonists That Reduces Liver Fibrosis
2016 Renga, Barbara; Cipriani, Sabrina; Carino, Adriana; Marchianò, Silvia; Zampella, Angela; Distrutti, Eleonora; Fiorucci, Stefano
BAR 501, a Novel GPBAR1 Ligand, Reverses Intestinal and Liver Inflammatory Models Demonstrating That GPBAR1 Is an Essential Modulator of Innate Immunity in Entero-Hepatic Tissues
2016 Cipriani, Sabrina; Renga, Barbara; Simonetti, Michele; Carino, Adriana; Zampella, Angela; Fiorucci, Stefano
The bile acid receptor GPBAR1 (TGR5) is expressed in human gastric cancers and promotes epithelial-mesenchymal transition in gastric cancer cell lines
2016 Carino, Adriana; Graziosi, Luigina; D'Amore, Claudio; Cipriani, Sabrina; Marchiano', Silvia; Marino, Elisabetta; Zampella, Angela; Rende, Mario; Mosci, Paolo; Distrutti, Eleonora; Donini, Annibale; Fiorucci, Stefano
Phallusiasterol C, A New Disulfated Steroid from the Mediterranean Tunicate Phallusia fumigata
2016 Imperatore, C; Senese, M; Aiello, A; Luciano, P; Fiorucci, Stefano; D'Amore, C; Carino, A; Menna, M.; Carino, Adriana
BAR502, a Dual FXR and GPBAR1 Agonist, Reverses Steatosis and Fibrosis in Rodent Model of NASH By Modulating Authophagic Genes
2016 Renga, Barbara; Cipriani, Sabrina; Carino, Adriana; Marchianò, Silvia; Zampella, Angela; Fiorucci, Stefano
Investigation on bile acid receptor regulators. Discovery of cholanoic acid derivatives with dual G-protein coupled bile acid receptor 1 (GPBAR1) antagonistic and farnesoid X receptor (FXR) modulatory activity
2016 Sepe, V; Renga, B; Festa, C; Finamore, C; Masullo, D; Carino, A; Cipriani, S; Distrutti, E; Fiorucci, Stefano; Zampella, A.; Carino, Adriana
New brominated flame retardants and their metabolites as activators of the pregnane X receptor
2016 Gramec Skledar, Darja; Tomašič, Tihomir; Carino, Adriana; Distrutti, Eleonora; Fiorucci, Stefano; Peterlin Mašič, Lucija
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
HIV-1 infection is associated with changes in nuclear receptor transcriptome, pro-inflammatory and lipid profile of monocytes | 2012 | Renga, Barbara; Francisci, Daniela; D'Amore, Claudio; Schiaroli, Elisabetta; Carino, A.; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana | |
The bile acid sensor FXR is required for immune-regulatory activities of TLR-9 in intestinal inflammation | 2013 | Renga, Barbara; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Carino, A; Bruno, A; Francisci, Daniela; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana | |
FXR mediates a chromatin looping in the GR promoter thus promoting the resolution of colitis in rodents. | 2013 | Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Mencarelli, Andrea; Carino, A; Sepe, V; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana | |
Solomonsterol A, a marine pregnane-X-receptor agonist, attenuates inflammation and immune dysfunction in a mouse model of arthritis. | 2013 | Mencarelli, Andrea; D'Amore, Claudio; Renga, Barbara; Cipriani, Sabrina; Carino, A; Sepe, V; Perissutti, E; D'Auria, Mv; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana | |
Exploitation of cholane scaffold for the discovery of potent and selective farnesoid X receptor (FXR) and G-protein coupled bile acid receptor 1 (GP-BAR1) ligands | 2014 | Festa, C; Renga, Barbara; D'Amore, Claudio; Sepe, V; Finamore, C; De Marino, S; Carino, A.; Cipriani, Sabrina; Monti, Mc; Zampella, A; Fiorucci, Stefano; Carino, Adriana | |
The HIV Matrix Protein p17 promotes the Activation of human hepatic stellate cells through interactions with CXCR2 and Syndecan-2 | 2014 | Renga, Barbara; Francisci, Daniela; Schiaroli, Elisabetta; Carino, A; Cipriani, Sabrina; D'Amore, Claudio; Sidoni, Angelo; DEL SORDO, Rachele; Ferri, Ivana; Lucattelli, M; Lunghi, B; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana | |
Structural insights into Estrogen Related Receptor-β modulation: 4-methylenesterols from Theonella swinhoei sponge as the first example of marine natural antagonists. | 2014 | Di Micco, S; Renga, Barbara; Carino, A; D'Auria, Mv; Zampella, A; Riccio, R; Fiorucci, Stefano; Bifulco, G.; Carino, Adriana | |
Impaired Itching Perception in Murine Models of Cholestasis Is Supported by Dysregulation of GPBAR1 Signaling | 2015 | Cipriani, Sabrina; Renga, Barbara; D'Amore, Claudio; Simonetti, M; De Tursi, Aa; Carino, Adriana; Monti, Mc; Sepe, V; Zampella, A; Fiorucci, Stefano | |
Reversal of Endothelial Dysfunction by GPBAR1 Agonism in Portal Hypertension Involves a AKT/FOXOA1 Dependent Regulation of H2S Generation and Endothelin-1 | 2015 | Renga, B.; Cipriani, S.; Carino, A.; Simonetti, M.; Zampella, A.; Fiorucci, S. | |
Cystathionine gamma-lyase, a H2S-generating enzyme, is a GPBAR1-regulated gene and contributes to vasodilation caused by secondary bile acids | 2015 | Renga, Barbara; Bucci, M; Cipriani, Sabrina; Carino, Adriana; Monti, Mc; Zampella, A; Gargiulo, A; d'Emmanuele di Villa Bianca, R; Distrutti, E; Fiorucci, Stefano | |
The HIV matrix protein p17 induces hepatic lipid accumulation via modulation of nuclear receptor transcriptoma | 2015 | Renga, Barbara; Francisci, Daniela; Carino, Adriana; Marchianò, Silvia; Cipriani, Sabrina; Chiara Monti, Maria; DEL SORDO, Rachele; Schiaroli, Elisabetta; Distrutti, Eleonora; Baldelli, Franco; Fiorucci, Stefano | |
Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists | 2016 | Sepe, V; Festa, C; Renga, B; Carino, A; Cipriani, S; Finamore, C; Masullo, D; Del Gaudio, F; Monti, Mc; Fiorucci, Stefano; Zampella, A.; Carino, Adriana | |
Navigation in bile acid chemical space: Discovery of novel FXR and GPBAR1 ligands | 2016 | Finamore, C; Festa, C; Renga, B; Sepe, V; Carino, A; Masullo, D; Biagioli, Michele; Marchianò, S; Capolupo, A; Monti, M; Fiorucci, Stefano; Zampella, A.; Carino, Adriana | |
A Comprehensive Analysis of Small Heterodimer Partner (SHP) Target Genes in Hepatic Stellate Cells and the Discovery of a New Class of SHP Agonists That Reduces Liver Fibrosis | 2016 | Renga, Barbara; Cipriani, Sabrina; Carino, Adriana; Marchianò, Silvia; Zampella, Angela; Distrutti, Eleonora; Fiorucci, Stefano | |
BAR 501, a Novel GPBAR1 Ligand, Reverses Intestinal and Liver Inflammatory Models Demonstrating That GPBAR1 Is an Essential Modulator of Innate Immunity in Entero-Hepatic Tissues | 2016 | Cipriani, Sabrina; Renga, Barbara; Simonetti, Michele; Carino, Adriana; Zampella, Angela; Fiorucci, Stefano | |
The bile acid receptor GPBAR1 (TGR5) is expressed in human gastric cancers and promotes epithelial-mesenchymal transition in gastric cancer cell lines | 2016 | Carino, Adriana; Graziosi, Luigina; D'Amore, Claudio; Cipriani, Sabrina; Marchiano', Silvia; Marino, Elisabetta; Zampella, Angela; Rende, Mario; Mosci, Paolo; Distrutti, Eleonora; Donini, Annibale; Fiorucci, Stefano | |
Phallusiasterol C, A New Disulfated Steroid from the Mediterranean Tunicate Phallusia fumigata | 2016 | Imperatore, C; Senese, M; Aiello, A; Luciano, P; Fiorucci, Stefano; D'Amore, C; Carino, A; Menna, M.; Carino, Adriana | |
BAR502, a Dual FXR and GPBAR1 Agonist, Reverses Steatosis and Fibrosis in Rodent Model of NASH By Modulating Authophagic Genes | 2016 | Renga, Barbara; Cipriani, Sabrina; Carino, Adriana; Marchianò, Silvia; Zampella, Angela; Fiorucci, Stefano | |
Investigation on bile acid receptor regulators. Discovery of cholanoic acid derivatives with dual G-protein coupled bile acid receptor 1 (GPBAR1) antagonistic and farnesoid X receptor (FXR) modulatory activity | 2016 | Sepe, V; Renga, B; Festa, C; Finamore, C; Masullo, D; Carino, A; Cipriani, S; Distrutti, E; Fiorucci, Stefano; Zampella, A.; Carino, Adriana | |
New brominated flame retardants and their metabolites as activators of the pregnane X receptor | 2016 | Gramec Skledar, Darja; Tomašič, Tihomir; Carino, Adriana; Distrutti, Eleonora; Fiorucci, Stefano; Peterlin Mašič, Lucija |
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