Sfoglia per Autore
Prediction ability of regression models. Part 1. Standard deviation of prediction errors (SDEP)
1992 Cruciani, Gabriele; Baroni, Massimo; Clementi, Sergio; Costantino, Gabriele; D., Riganelli; B., Skagerberg
Prediction ability of regression models. Part 2. Selection of the best predictive PLS model
1992 Baroni, Massimo; Clementi, Sergio; Cruciani, Gabriele; Costantino, Gabriele; D., Riganelli; E., Oberrauch
HETEROCYCLIC MODULATORS OF THE NMDA RECEPTOR
1993 Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; A., Garzon; R., Luneia; M. R., Mahmoud; Marinozzi, Maura; M., Roberti; G. C., Rosato; S. A., Shiba
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi
Conformational requirements for interaction of L-glutamate with the metabotropic EAA receptor
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto
Series design
1993 Clementi, Sergio; Cruciani, Gabriele; Baroni, Massimo; Costantino, Gabriele
Autocorrelation as a tool for a congruent description of molecu¬les in 3D-QSAR studies
1993 Clementi, Sergio; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Costantino, Gabriele; Baroni, Massimo; S., Wold
Generating Optimal Linear PLS Estimations (GOLPE): An Advanced Chemometric Tool for Handling 3D-QSAR Problems
1993 Baroni, Massimo; Costantino, Gabriele; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Clementi, Sergio
GOLPE: An Advanced Chemometric Tool for 3D-QSAR Problems
1993 Baroni, Massimo; Costantino, Gabriele; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Clementi, Sergio
MODULATION OF THE KYNURENINE PATHWAY IN SEARCH FOR NEW NEUROPROTECTIVE AGENTS - SYNTHESIS AND PRELIMINARY EVALUATION OF (M-NITROBENZOYL)ALANINE, A POTENT INHIBITOR OF KYNURENINE-3-HYDROXYLASE
1994 Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; M. R., Mahmoud; L., Mattoli; B. M., Sadeghpour; F., Moroni; A., Chiarugi; R., Carpenedo
SYNTHESIS AND BIOLOGICAL EVALUATION OF 6-CARBOXY-3,4-METHANOPROLINES, NEW RIGID GLUTAMATE ANALOGS
1995 Marinozzi, Maura; Natalini, Benedetto; M. H., Ni; Costantino, Gabriele; Pellicciari, Roberto; C., Thomsen
Disjoint Principal Properties of Organic Substituents
1995 H., van de Waterbeemd; Costantino, Gabriele; Clementi, Sergio; Cruciani, Gabriele; Valigi, Roberta
The Pseudoactive Site as a Tool for Indirect Drug Design. Application to Inhibitors of Kynurenine-3-hydroxylase
1995 Costantino, Gabriele; Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto
1-AMINOINDAN-1,5-DICARBOXYLIC ACID - A NOVEL ANTAGONIST AT PHOSPHOLIPASE C-LINKED METABOTROPIC GLUTAMATE RECEPTORS
1995 Pellicciari, Roberto; R., Luneia; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; P., Jakobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen
S-(+)-2-(3'carboxy-bicyclo[1.1.1]pentyl)glycine, a structurally new group I metabotropic glutamate receptor antagonist
1996 Pellicciari, Roberto; Raimondo, M. R.; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Thomsen, C.
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-Phenylcarboxycyclopropylglycine (PCCG-4): a Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors
1996 Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; P., Tijskens; C., Thomsen; Pellicciari, Roberto
Synthesis of 6,6-dicarboxy-3,4-methano-L-proline, a new constrained glutamate analog endowed with neuroprotective properties
1996 Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Pellicciari, Roberto; V., Bruno; F., Nicoletti
Kynurenine-3-hydroxylase and its selective inhibitors. Molecular modeling studies.
1996 Costantino, Gabriele; L., Mattoli; F., Moroni; Natalini, Benedetto; Pellicciari, Roberto
Synthesis and pharmacological characterization of all sixteen stereoisomers of 2-(2'-carboxy-3'-phenylcyclopropyl)glycine. Focus on (2S,1'S,2'S,3'R)-2-(2'-carboxy-3'-phenylcyclopropyl)glycine, a novel and selective group II metabotropic glutamate receptors antagonist
1996 Pellicciari, Roberto; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; R., Luneia; G., Giorgi; F., Moroni; C., Thomsen
Synthesis, preliminary evaluation and molecular modeling studies of new, conformationally constrained analogues of the competitive NMDA receptor antagonist 4-(phosphonomethyl)-2-piperidinecarboxylic acid (CGS 19755)
1997 Pellicciari, Roberto; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; D. C., Lankin; J. P., Snyder; J. B., Monahan
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Prediction ability of regression models. Part 1. Standard deviation of prediction errors (SDEP) | 1992 | Cruciani, Gabriele; Baroni, Massimo; Clementi, Sergio; Costantino, Gabriele; D., Riganelli; B., Skagerberg | |
Prediction ability of regression models. Part 2. Selection of the best predictive PLS model | 1992 | Baroni, Massimo; Clementi, Sergio; Cruciani, Gabriele; Costantino, Gabriele; D., Riganelli; E., Oberrauch | |
HETEROCYCLIC MODULATORS OF THE NMDA RECEPTOR | 1993 | Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; A., Garzon; R., Luneia; M. R., Mahmoud; Marinozzi, Maura; M., Roberti; G. C., Rosato; S. A., Shiba | |
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi | |
Conformational requirements for interaction of L-glutamate with the metabotropic EAA receptor | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto | |
Series design | 1993 | Clementi, Sergio; Cruciani, Gabriele; Baroni, Massimo; Costantino, Gabriele | |
Autocorrelation as a tool for a congruent description of molecu¬les in 3D-QSAR studies | 1993 | Clementi, Sergio; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Costantino, Gabriele; Baroni, Massimo; S., Wold | |
Generating Optimal Linear PLS Estimations (GOLPE): An Advanced Chemometric Tool for Handling 3D-QSAR Problems | 1993 | Baroni, Massimo; Costantino, Gabriele; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Clementi, Sergio | |
GOLPE: An Advanced Chemometric Tool for 3D-QSAR Problems | 1993 | Baroni, Massimo; Costantino, Gabriele; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Clementi, Sergio | |
MODULATION OF THE KYNURENINE PATHWAY IN SEARCH FOR NEW NEUROPROTECTIVE AGENTS - SYNTHESIS AND PRELIMINARY EVALUATION OF (M-NITROBENZOYL)ALANINE, A POTENT INHIBITOR OF KYNURENINE-3-HYDROXYLASE | 1994 | Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; M. R., Mahmoud; L., Mattoli; B. M., Sadeghpour; F., Moroni; A., Chiarugi; R., Carpenedo | |
SYNTHESIS AND BIOLOGICAL EVALUATION OF 6-CARBOXY-3,4-METHANOPROLINES, NEW RIGID GLUTAMATE ANALOGS | 1995 | Marinozzi, Maura; Natalini, Benedetto; M. H., Ni; Costantino, Gabriele; Pellicciari, Roberto; C., Thomsen | |
Disjoint Principal Properties of Organic Substituents | 1995 | H., van de Waterbeemd; Costantino, Gabriele; Clementi, Sergio; Cruciani, Gabriele; Valigi, Roberta | |
The Pseudoactive Site as a Tool for Indirect Drug Design. Application to Inhibitors of Kynurenine-3-hydroxylase | 1995 | Costantino, Gabriele; Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto | |
1-AMINOINDAN-1,5-DICARBOXYLIC ACID - A NOVEL ANTAGONIST AT PHOSPHOLIPASE C-LINKED METABOTROPIC GLUTAMATE RECEPTORS | 1995 | Pellicciari, Roberto; R., Luneia; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; P., Jakobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen | |
S-(+)-2-(3'carboxy-bicyclo[1.1.1]pentyl)glycine, a structurally new group I metabotropic glutamate receptor antagonist | 1996 | Pellicciari, Roberto; Raimondo, M. R.; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Thomsen, C. | |
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-Phenylcarboxycyclopropylglycine (PCCG-4): a Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors | 1996 | Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; P., Tijskens; C., Thomsen; Pellicciari, Roberto | |
Synthesis of 6,6-dicarboxy-3,4-methano-L-proline, a new constrained glutamate analog endowed with neuroprotective properties | 1996 | Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Pellicciari, Roberto; V., Bruno; F., Nicoletti | |
Kynurenine-3-hydroxylase and its selective inhibitors. Molecular modeling studies. | 1996 | Costantino, Gabriele; L., Mattoli; F., Moroni; Natalini, Benedetto; Pellicciari, Roberto | |
Synthesis and pharmacological characterization of all sixteen stereoisomers of 2-(2'-carboxy-3'-phenylcyclopropyl)glycine. Focus on (2S,1'S,2'S,3'R)-2-(2'-carboxy-3'-phenylcyclopropyl)glycine, a novel and selective group II metabotropic glutamate receptors antagonist | 1996 | Pellicciari, Roberto; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; R., Luneia; G., Giorgi; F., Moroni; C., Thomsen | |
Synthesis, preliminary evaluation and molecular modeling studies of new, conformationally constrained analogues of the competitive NMDA receptor antagonist 4-(phosphonomethyl)-2-piperidinecarboxylic acid (CGS 19755) | 1997 | Pellicciari, Roberto; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; D. C., Lankin; J. P., Snyder; J. B., Monahan |
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