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First General Approach to Cyclohex-3-ene-1,1-bis(phosphonates) by Diels-Alder Cycloaddition of Tetraethyl Vinylidenebis(phosphonate) to 1,3-Dienes 2003 Ruzziconi, Renzo; Ricci, G; Gioiello, Antimo; Couthon Gourvès, H; Gourvès, J. P.
Design, synthesis and S.A.R. of bile acid analogs as novel and selective FXR ligands 2004 Sadeghpour, B. M.; Gioiello, Antimo; Costantino, G.; Camaioni, Emidio; Rizzo, G.; Renga, B.; Fiorucci, Stefano; Pellicciari, Roberto
Development and identification of new farnesoid X receptor (FXR) modulators as chemical tool for gene functional analysis 2004 Gioiello, Antimo
Bile Acid Derivatives as Ligands of the Farnesoid X Receptor. Synthesis, Evaluation, and Structure Activity Relationship of a Series of Body and Side Chain Modified Analogs of Chenodeoxycholic Acid 2004 Pellicciari, Roberto; Costantino, Gabriele; Camaioni, Emidio; Sadeghpour, B. M.; Entrena Guadix, A.; Willson, T.; Fiorucci, Stefano; Clerici, C.; Gioiello, Antimo
Molecular Dynamics Simulation of the Ligand Binding Domain of Farnesoid X Receptor (FXR). Insights into Helix-12 Stability and Coactivator Peptide Stabilization in Response to Agonist Binding 2005 Costantino, Gabriele; Entrena Guadix, A.; Macchiarulo, Antonio; Gioiello, Antimo; Pellicciari, Roberto
In search for FXR gene selective modulators: synthesis, biological activity and docking studies of 23-N-carbocinnamyloxy-norchenodeoxycholanylamine (UPF838). 2006 Gioiello, Antimo; Costantino, G.; Sadeghpour, B. M.; Rizzo, G.; Parks, D. J.; Entrena Gaudix, A.; Fiorucci, Stefano; Pellicciari, Roberto
Potential Therapeutic Applications of Farnesoid X Receptor (FXR) Modulators 2006 Pellicciari, Roberto; Gioiello, Antimo; Costantino, Gabriele
The Farnesoid X Receptor Promotes Adipocyte Differentiation and Regulates Adipose Cell Function in Vivo 2006 Rizzo, G.; Disante, M.; Mencarelli, Andrea; Renga, Barbara; Gioiello, Antimo; Pellicciari, R.; Fiorucci, Stefano
Back door modulation of the farnesoid X receptor: design, synthesis, and biological evaluation of a series of side chain modified chenodeoxycholic acid derivatives. 2006 Pellicciari, Roberto; Gioiello, Antimo; Costantino, G.; Sadeghpour, B. M.; Rizzo, G.; Meyer, U.; Parks, D.; Entrena Guadix, A.; Fiorucci, Stefano
In search for FXR gene selective modulators: from guggulsterone to side-chain modified bile acid derivatives 2007 Gioiello, Antimo; Costantino, G.; Sadeghpour, B. M.; Entrena Guadix, A.; Meyer, U.; Fiorucci, Stefano; Pellicciari, Roberto
Heterocyclic α-diazo-β-hydroxy ester derivatives and their reaction with boron trifluoride etherate 2007 Sabbatini, P.; Sadeghpour, B. M.; Gioiello, Antimo; Pellicciari, Roberto
Correlation between CMC and chromatographic index: simple and effective evaluation of the hydrophobic/hydrophilic balance of bile acids 2007 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Gioiello, Antimo; Pellicciari, Roberto
Indium triflate catalyzed reaction of diisopropyl diazomethylphophonate with imines as a new approach to cis- and trans-aziridine-2-phosphonates 2007 Pellicciari, Roberto; Amori, L.; Kuznetsova, N.; Zlotsky, S.; Gioiello, Antimo
Nongenomic Actions of Bile Acids. Synthesis and Preliminary Characterization of 23-and 6,23-Alkyl-Sobstituted Bile Acid Derivatives as Selective Modulators for the G-Protein Coupled Receptor TGR5 2007 Pellicciari, Roberto; H., Sato; Gioiello, Antimo; G., Costatino; Macchiarulo, Antonio; B. M., Sadeghpour; G., Giorgi; K., Schoonjans; J., Auwerx
Derived chromatographic indexes as effective tools to study the self-aggregation process of bile acids. 2008 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Gioiello, Antimo; Pellicciari, Roberto
Molecular field analysis and quantitative structure-activity studies (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5 receptor. 2008 Gioiello, Antimo; Macchiarulo, Antonio; Thomas, C.; Massarotti, A.; Nuti, Roberto; Rosatelli, E.; Sabatini, P.; Schoonjans, K.; Auwerx, J.; Pellicciari, Roberto
Diazoesters in the synthesis of heterocyclic compounds of biological interest 2008 Gioiello, Antimo; Pellicciari, Roberto
Novel Potent and Selective Bile Acid Derivatives as TGR5 Agonists: Biological Screening, Structure-Activity Relationships and Molecular Modeling Studies 2008 Sato, H.; Macchiarulo, Antonio; Thomas, C.; Gioiello, Antimo; Une, M.; Hofmann, A.; Saladin, R.; Schoonjans, K.; Pellicciari, Roberto; Auwerx, J.
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5. 2008 Macchiarulo, Antonio; Gioiello, Antimo; Thomas, C.; Massarotti, A.; Nuti, Roberto; Rosatelli, E.; Sabbatini, P.; Schoonjans, K.; Auwerx, J.; Pellicciari, Roberto
Novel body modified bile acid derivatives as TGR5 modulators 2009 Rosatelli, E; Gioiello, Antimo; Macchiarulo, Antonio; Thomas, C; Rizzo, G; Adorini, L; Auwerx, J; Pellicciari, R.
Mostrati risultati da 1 a 20 di 180
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