Sfoglia per Rivista BIOORGANIC
Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K-ATP channel openers
2005 Carosati, Emanuele; Lemoine, H.; Spogli, Roberto; Grittner, D.; Mannhold, R.; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta
Bulky 1,4-benzoxazine derivatives with antifungal activity
2009 Fringuelli, Renata; Giacche', Nicola; Milanese, Lara; Cenci, Elio; Macchiarulo, Antonio; Vecchiarelli, Anna; Costantino, Gabriele; Schiaffella, Fausto
Cyathane diterpenes from Sarcodon cyrneus and evaluation of their activities of neuritegenesis and nerve growth factor production
2007 Marcotullio, Maria Carla; Pagiotti, Rita; Maltese, F.; Oball Mond Mwankie, G. N.; Hoshino, T.; Obara, Y.; Nakahata, N.
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands.
2009 Filosa, R.; Fulco, MARIA CARMELA; Marinozzi, Maura; Giacchè, N.; Macchiarulo, Antonio; Peduto, A.; Massa, A.; De Caprariis, P.; Thomsen, C.; Christoffersen, C.; Pellicciari, Roberto
Design, synthesis and in vitro antitumor activity of new trans 2-[2-(heteroaryl)vinyl]-1,3-dimethylimidazolium iodides
2004 Ballistreri, Francesco P.; Barresi, Vincenza; Benedetti, Paolo; Caltabiano, Gianluigi; Fortuna, COSIMO GIANLUCA; Longo, Maria L.; Musumarra, Giuseppe
Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents.
2009 Monforte, A. M.; Logoteta, P.; Ferro, S.; De Luca, L.; Iraci, Nunzio; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole.
2005 Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto
Ester derivatives of annulated tetrahydroazocines: a new class of selective acetylcholinesterase inhibitors
2006 Carotti, Andrea; M., de Candia; M., Catto; T. N., Borisova; A. V., Varlamov; E., Mendez Alvarez; R., Soto Otero; L. G., Voskressensky; C., Altomare
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands
2014 Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana
Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3a,7a-dihydroxy-6a-ethyl-24-nor-5b-cholan-23-amine
2011 Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; P., Filipponi; G., Costantino; G., Rizzo; L., Adorini; Pellicciari, Roberto
Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres
2020 Ferri, M.; Alunno, M.; Greco, F. A.; Mammoli, A.; Saluti, G.; Carotti, A.; Sardella, R.; Macchiarulo, A.; Camaioni, E.; Liscio, P.
GRIND/ALMOND investigations on CysLT(1) receptor antagonists of the quinolinyl(bridged)aryl type
2004 Benedetti, Paolo; Mannhold, R.; Cruciani, Gabriele; Ottaviani, G.
High Affinity Central Benzodiazepine Receptor Ligands. Part 3: Insights into the Pharmacophore and Pattern Recognition Study of Intrinsic Activities of Pyrazolo[4,3-c]quinolin-3-ones
2003 Carotti, Andrea; C., Altomare; L., Savini; L., Chiasserini; C., Pellerano; M. P., Mascia; E., Maciocco; F., Busonero; M., Mameli; G., Biggio; E., Sanna
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin.
2008 Stancanelli, R; Crupi, V; DE LUCA, L; Ficarra, P; Ficarra, R; Gitto, R; Guardo, M; Iraci, Nunzio; Majolino, D; Tommasini, S; Venuti, V.
Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei.
2013 Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O.
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity.
1998 Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M.
Molecular structure and stereoelectronic properties of herbicide sulphonylureas
2002 Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C.
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action.
2010 Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K-ATP channel openers | 2005 | Carosati, Emanuele; Lemoine, H.; Spogli, Roberto; Grittner, D.; Mannhold, R.; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta | |
| Bulky 1,4-benzoxazine derivatives with antifungal activity | 2009 | Fringuelli, Renata; Giacche', Nicola; Milanese, Lara; Cenci, Elio; Macchiarulo, Antonio; Vecchiarelli, Anna; Costantino, Gabriele; Schiaffella, Fausto | |
| Cyathane diterpenes from Sarcodon cyrneus and evaluation of their activities of neuritegenesis and nerve growth factor production | 2007 | Marcotullio, Maria Carla; Pagiotti, Rita; Maltese, F.; Oball Mond Mwankie, G. N.; Hoshino, T.; Obara, Y.; Nakahata, N. | |
| Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi | |
| Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands. | 2009 | Filosa, R.; Fulco, MARIA CARMELA; Marinozzi, Maura; Giacchè, N.; Macchiarulo, Antonio; Peduto, A.; Massa, A.; De Caprariis, P.; Thomsen, C.; Christoffersen, C.; Pellicciari, Roberto | |
| Design, synthesis and in vitro antitumor activity of new trans 2-[2-(heteroaryl)vinyl]-1,3-dimethylimidazolium iodides | 2004 | Ballistreri, Francesco P.; Barresi, Vincenza; Benedetti, Paolo; Caltabiano, Gianluigi; Fortuna, COSIMO GIANLUCA; Longo, Maria L.; Musumarra, Giuseppe | |
| Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents. | 2009 | Monforte, A. M.; Logoteta, P.; Ferro, S.; De Luca, L.; Iraci, Nunzio; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A. | |
| Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole. | 2005 | Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto | |
| Ester derivatives of annulated tetrahydroazocines: a new class of selective acetylcholinesterase inhibitors | 2006 | Carotti, Andrea; M., de Candia; M., Catto; T. N., Borisova; A. V., Varlamov; E., Mendez Alvarez; R., Soto Otero; L. G., Voskressensky; C., Altomare | |
| Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands | 2014 | Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana | |
| Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3a,7a-dihydroxy-6a-ethyl-24-nor-5b-cholan-23-amine | 2011 | Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; P., Filipponi; G., Costantino; G., Rizzo; L., Adorini; Pellicciari, Roberto | |
| Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres | 2020 | Ferri, M.; Alunno, M.; Greco, F. A.; Mammoli, A.; Saluti, G.; Carotti, A.; Sardella, R.; Macchiarulo, A.; Camaioni, E.; Liscio, P. | |
| GRIND/ALMOND investigations on CysLT(1) receptor antagonists of the quinolinyl(bridged)aryl type | 2004 | Benedetti, Paolo; Mannhold, R.; Cruciani, Gabriele; Ottaviani, G. | |
| High Affinity Central Benzodiazepine Receptor Ligands. Part 3: Insights into the Pharmacophore and Pattern Recognition Study of Intrinsic Activities of Pyrazolo[4,3-c]quinolin-3-ones | 2003 | Carotti, Andrea; C., Altomare; L., Savini; L., Chiasserini; C., Pellerano; M. P., Mascia; E., Maciocco; F., Busonero; M., Mameli; G., Biggio; E., Sanna | |
| Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1 | 2001 | Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio | |
| Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin. | 2008 | Stancanelli, R; Crupi, V; DE LUCA, L; Ficarra, P; Ficarra, R; Gitto, R; Guardo, M; Iraci, Nunzio; Majolino, D; Tommasini, S; Venuti, V. | |
| Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei. | 2013 | Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O. | |
| Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity. | 1998 | Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M. | |
| Molecular structure and stereoelectronic properties of herbicide sulphonylureas | 2002 | Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C. | |
| New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action. | 2010 | Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A. |
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