Sfoglia per Rivista BIOORGANIC
Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres
2020 Ferri, M.; Alunno, M.; Greco, F. A.; Mammoli, A.; Saluti, G.; Carotti, A.; Sardella, R.; Macchiarulo, A.; Camaioni, E.; Liscio, P.
GRIND/ALMOND investigations on CysLT(1) receptor antagonists of the quinolinyl(bridged)aryl type
2004 Benedetti, Paolo; Mannhold, R.; Cruciani, Gabriele; Ottaviani, G.
High Affinity Central Benzodiazepine Receptor Ligands. Part 3: Insights into the Pharmacophore and Pattern Recognition Study of Intrinsic Activities of Pyrazolo[4,3-c]quinolin-3-ones
2003 Carotti, Andrea; C., Altomare; L., Savini; L., Chiasserini; C., Pellerano; M. P., Mascia; E., Maciocco; F., Busonero; M., Mameli; G., Biggio; E., Sanna
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin.
2008 Stancanelli, R; Crupi, V; DE LUCA, L; Ficarra, P; Ficarra, R; Gitto, R; Guardo, M; Iraci, Nunzio; Majolino, D; Tommasini, S; Venuti, V.
Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei.
2013 Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O.
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity.
1998 Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M.
Molecular structure and stereoelectronic properties of herbicide sulphonylureas
2002 Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C.
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action.
2010 Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A.
New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles
2014 Cosimo G., Fortuna; Roberto, Berardozzi; Carmela, Bonaccorso; Gianluigi, Caltabiano; Lorenzo Di, Bari; Goracci, Laura; Annalisa, Guarcello; Andrea, Pace; Antonio Palumbo, Piccionello; Gennaro, Pescitelli; Paola, Pierro; Elena, Lonati; Alessandra, Bulbarelli; Clementina E. A., Cocuzza; Giuseppe, Musumarra; Rosario, Musumeci
New substituted 9-alkylpurines as adenosine receptor ligands
1998 Camaioni, Emidio; Costanzi, S; Vittori, S; Volpini, R; Klotz, Kn; Cristalli, G.
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
2010 Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation
2006 Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Fringuelli, Renata
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors.
2008 Monforte, Am; Rao, A; Logoteta, P; Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, A.
Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists
2012 Marinozzi, Maura; Carotti, Andrea; E., Sansone; Macchiarulo, Antonio; Rosatelli, Emiliano; Sardella, Roccaldo; Natalini, Benedetto; G., Rizzo; L., Adorini; D., Passeri; F., De Franco; M., Pruzanski; Pellicciari, Roberto
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase
2012 Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta
Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction
2003 Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor
2010 DE LUCA, L; Ferro, S; Gitto, R; Barreca, MARIA LETIZIA; Agnello, S; Christ, F; Debyser, Z; Chimirri, A.
Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones
1999 Cecchetti, Violetta; Tabarrini, Oriana; Sabatini, Stefano; Miao, H.; Filipponi, Enrica; Fravolini, Arnaldo
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position
2009 Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres | 2020 | Ferri, M.; Alunno, M.; Greco, F. A.; Mammoli, A.; Saluti, G.; Carotti, A.; Sardella, R.; Macchiarulo, A.; Camaioni, E.; Liscio, P. | |
| GRIND/ALMOND investigations on CysLT(1) receptor antagonists of the quinolinyl(bridged)aryl type | 2004 | Benedetti, Paolo; Mannhold, R.; Cruciani, Gabriele; Ottaviani, G. | |
| High Affinity Central Benzodiazepine Receptor Ligands. Part 3: Insights into the Pharmacophore and Pattern Recognition Study of Intrinsic Activities of Pyrazolo[4,3-c]quinolin-3-ones | 2003 | Carotti, Andrea; C., Altomare; L., Savini; L., Chiasserini; C., Pellerano; M. P., Mascia; E., Maciocco; F., Busonero; M., Mameli; G., Biggio; E., Sanna | |
| Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1 | 2001 | Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio | |
| Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin. | 2008 | Stancanelli, R; Crupi, V; DE LUCA, L; Ficarra, P; Ficarra, R; Gitto, R; Guardo, M; Iraci, Nunzio; Majolino, D; Tommasini, S; Venuti, V. | |
| Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei. | 2013 | Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O. | |
| Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity. | 1998 | Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M. | |
| Molecular structure and stereoelectronic properties of herbicide sulphonylureas | 2002 | Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C. | |
| New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action. | 2010 | Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A. | |
| New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles | 2014 | Cosimo G., Fortuna; Roberto, Berardozzi; Carmela, Bonaccorso; Gianluigi, Caltabiano; Lorenzo Di, Bari; Goracci, Laura; Annalisa, Guarcello; Andrea, Pace; Antonio Palumbo, Piccionello; Gennaro, Pescitelli; Paola, Pierro; Elena, Lonati; Alessandra, Bulbarelli; Clementina E. A., Cocuzza; Giuseppe, Musumarra; Rosario, Musumeci | |
| New substituted 9-alkylpurines as adenosine receptor ligands | 1998 | Camaioni, Emidio; Costanzi, S; Vittori, S; Volpini, R; Klotz, Kn; Cristalli, G. | |
| Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. | 2010 | Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A. | |
| Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation | 2006 | Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Fringuelli, Renata | |
| Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors. | 2008 | Monforte, Am; Rao, A; Logoteta, P; Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, A. | |
| Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists | 2012 | Marinozzi, Maura; Carotti, Andrea; E., Sansone; Macchiarulo, Antonio; Rosatelli, Emiliano; Sardella, Roccaldo; Natalini, Benedetto; G., Rizzo; L., Adorini; D., Passeri; F., De Franco; M., Pruzanski; Pellicciari, Roberto | |
| Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase | 2012 | Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta | |
| Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction | 2003 | Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto | |
| Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor | 2010 | DE LUCA, L; Ferro, S; Gitto, R; Barreca, MARIA LETIZIA; Agnello, S; Christ, F; Debyser, Z; Chimirri, A. | |
| Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones | 1999 | Cecchetti, Violetta; Tabarrini, Oriana; Sabatini, Stefano; Miao, H.; Filipponi, Enrica; Fravolini, Arnaldo | |
| Studies on Anti-HIV Quinolones: New Insights on the C-6 Position | 2009 | Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta |
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