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Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole. 2005 Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto
Ester derivatives of annulated tetrahydroazocines: a new class of selective acetylcholinesterase inhibitors 2006 Carotti, Andrea; M., de Candia; M., Catto; T. N., Borisova; A. V., Varlamov; E., Mendez Alvarez; R., Soto Otero; L. G., Voskressensky; C., Altomare
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands 2014 Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana
Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3a,7a-dihydroxy-6a-ethyl-24-nor-5b-cholan-23-amine 2011 Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; P., Filipponi; G., Costantino; G., Rizzo; L., Adorini; Pellicciari, Roberto
Fragment based drug design and diversity-oriented synthesis of carboxylic acid isosteres 2020 Ferri, M.; Alunno, M.; Greco, F. A.; Mammoli, A.; Saluti, G.; Carotti, A.; Sardella, R.; Macchiarulo, A.; Camaioni, E.; Liscio, P.
GRIND/ALMOND investigations on CysLT(1) receptor antagonists of the quinolinyl(bridged)aryl type 2004 Benedetti, Paolo; Mannhold, R.; Cruciani, Gabriele; Ottaviani, G.
High Affinity Central Benzodiazepine Receptor Ligands. Part 3: Insights into the Pharmacophore and Pattern Recognition Study of Intrinsic Activities of Pyrazolo[4,3-c]quinolin-3-ones 2003 Carotti, Andrea; C., Altomare; L., Savini; L., Chiasserini; C., Pellerano; M. P., Mascia; E., Maciocco; F., Busonero; M., Mameli; G., Biggio; E., Sanna
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1 2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin. 2008 Stancanelli, R; Crupi, V; DE LUCA, L; Ficarra, P; Ficarra, R; Gitto, R; Guardo, M; Iraci, Nunzio; Majolino, D; Tommasini, S; Venuti, V.
Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei. 2013 Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O.
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity. 1998 Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M.
Molecular structure and stereoelectronic properties of herbicide sulphonylureas 2002 Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C.
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action. 2010 Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A.
New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles 2014 Cosimo G., Fortuna; Roberto, Berardozzi; Carmela, Bonaccorso; Gianluigi, Caltabiano; Lorenzo Di, Bari; Goracci, Laura; Annalisa, Guarcello; Andrea, Pace; Antonio Palumbo, Piccionello; Gennaro, Pescitelli; Paola, Pierro; Elena, Lonati; Alessandra, Bulbarelli; Clementina E. A., Cocuzza; Giuseppe, Musumarra; Rosario, Musumeci
New substituted 9-alkylpurines as adenosine receptor ligands 1998 Camaioni, Emidio; Costanzi, S; Vittori, S; Volpini, R; Klotz, Kn; Cristalli, G.
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. 2010 Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation 2006 Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Fringuelli, Renata
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors. 2008 Monforte, Am; Rao, A; Logoteta, P; Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, A.
Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists 2012 Marinozzi, Maura; Carotti, Andrea; E., Sansone; Macchiarulo, Antonio; Rosatelli, Emiliano; Sardella, Roccaldo; Natalini, Benedetto; G., Rizzo; L., Adorini; D., Passeri; F., De Franco; M., Pruzanski; Pellicciari, Roberto
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase 2012 Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta
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