Sfoglia per Rivista
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity.
1998 Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M.
Molecular structure and stereoelectronic properties of herbicide sulphonylureas
2002 Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C.
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action.
2010 Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A.
New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles
2014 Cosimo G., Fortuna; Roberto, Berardozzi; Carmela, Bonaccorso; Gianluigi, Caltabiano; Lorenzo Di, Bari; Goracci, Laura; Annalisa, Guarcello; Andrea, Pace; Antonio Palumbo, Piccionello; Gennaro, Pescitelli; Paola, Pierro; Elena, Lonati; Alessandra, Bulbarelli; Clementina E. A., Cocuzza; Giuseppe, Musumarra; Rosario, Musumeci
New substituted 9-alkylpurines as adenosine receptor ligands
1998 Camaioni, Emidio; Costanzi, S; Vittori, S; Volpini, R; Klotz, Kn; Cristalli, G.
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
2010 Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation
2006 Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Fringuelli, Renata
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors.
2008 Monforte, Am; Rao, A; Logoteta, P; Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, A.
Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists
2012 Marinozzi, Maura; Carotti, Andrea; E., Sansone; Macchiarulo, Antonio; Rosatelli, Emiliano; Sardella, Roccaldo; Natalini, Benedetto; G., Rizzo; L., Adorini; D., Passeri; F., De Franco; M., Pruzanski; Pellicciari, Roberto
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase
2012 Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta
Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction
2003 Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor
2010 DE LUCA, L; Ferro, S; Gitto, R; Barreca, MARIA LETIZIA; Agnello, S; Christ, F; Debyser, Z; Chimirri, A.
Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones
1999 Cecchetti, Violetta; Tabarrini, Oriana; Sabatini, Stefano; Miao, H.; Filipponi, Enrica; Fravolini, Arnaldo
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position
2009 Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta
Synthesis and Antibacterial Evaluation of [1,3]Benzothiazino[3,2-a]quinoline and [3,1]Benzothiazino[1,2-a]quinoline-6-carboxylic Acid Derivatives
1997 Cecchetti, Violetta; Cruciani, Gabriele; Filipponi, E.; Fravolini, Arnaldo; Tabarrini, Oriana; Xin, T.
Synthesis and biological evaluation of (2S)- and (2R)-2-(3'-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands.
2006 Filosa, R.; Marinozzi, Maura; Costantino, Gabriele; Brunsgaard Hemit, M.; Thomsen, C.; Pellicciari, Roberto
Synthesis and Biological Evaluation of 2-(3’-(1H-tetrazol-5-yl)bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 Receptor
2001 Costantino, Gabriele; Marinozzi, Maura; Camaioni, Emidio; Pellicciari, Roberto; Maltoni, K.; Prezeau, L.; Pin, J.
Synthesis and characterization of carnitine nitro-derivatives.
2008 Piermatti, Oriana; Fringuelli, Francesco; Pochini, L.; Indiveri, C.; Palmerini, Carlo Alberto
Synthesis and preliminary pharmacological evaluation of the four stereoisomers of (2S)-2-(2'-phosphono-3'-phenylcyclopropyl)glycine, the first class of 3'-substituted trans-2-(2'-phosphonocyclopropyl)glycines
2007 Marinozzi, Maura; M., Serpi; L., Amori; M., GAVILAN DIAZ; G., Costantino; U., Meyer; P. J., Flor; F., Gasparini; R., Heckendorn; R., Kuhn; G., Giorgi; M., BRUNSGAARD HERMIT; C., Thomsen; R., Pellicciari
Synthesis and Prelyminary Pharmacological Evaluation of the Four Stereoisomers of (2S)-2-(2’-Phosphono-3’-phenylcyclopropyl)glycine, the First Stereolibrary of trans 3’- Substituted -2-(2’-Phosphonocyclopropyl) glycine
2007 Marinozzi, Maura; M., Serpi; L., Amori; M. G., Diaz; Costantino, Gabriele; U., Mayer; P. J., Flor; F., Gasparini; R., Heckendorn; R., Kuhn; G., Giorgi; M. B., Hermit; C., Thomsen; Pellicciari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity. | 1998 | Sissi, C.; Andreolli, M.; Cecchetti, Violetta; Fravolini, Arnaldo; Gatto, B.; Palumbo, M. | |
Molecular structure and stereoelectronic properties of herbicide sulphonylureas | 2002 | Galeazzi, R.; Marucchini, C.; Orena, M.; Zadra, and C. | |
New chloro,fluorobenzylindole derivatives as integrase strand-transfer inhibitors (INSTIs) and their mode of action. | 2010 | Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; DE GRAZIA, S; Christ, F; Debyser, Z; Chimirri, A. | |
New potent antibacterials against Gram-positive multiresistant pathogens: Effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles | 2014 | Cosimo G., Fortuna; Roberto, Berardozzi; Carmela, Bonaccorso; Gianluigi, Caltabiano; Lorenzo Di, Bari; Goracci, Laura; Annalisa, Guarcello; Andrea, Pace; Antonio Palumbo, Piccionello; Gennaro, Pescitelli; Paola, Pierro; Elena, Lonati; Alessandra, Bulbarelli; Clementina E. A., Cocuzza; Giuseppe, Musumarra; Rosario, Musumeci | |
New substituted 9-alkylpurines as adenosine receptor ligands | 1998 | Camaioni, Emidio; Costanzi, S; Vittori, S; Volpini, R; Klotz, Kn; Cristalli, G. | |
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. | 2010 | Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A. | |
Novel ketoconazole analogues based on the replacement of 2,4-dichlorophenyl group with 1,4-benzothiazine moiety: design, synthesis, and microbiological evaluation | 2006 | Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Fringuelli, Renata | |
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside reverse transcriptase inhibitors. | 2008 | Monforte, Am; Rao, A; Logoteta, P; Ferro, S; DE LUCA, L; Barreca, MARIA LETIZIA; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, A. | |
Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonists | 2012 | Marinozzi, Maura; Carotti, Andrea; E., Sansone; Macchiarulo, Antonio; Rosatelli, Emiliano; Sardella, Roccaldo; Natalini, Benedetto; G., Rizzo; L., Adorini; D., Passeri; F., De Franco; M., Pruzanski; Pellicciari, Roberto | |
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase | 2012 | Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta | |
Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction | 2003 | Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto | |
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor | 2010 | DE LUCA, L; Ferro, S; Gitto, R; Barreca, MARIA LETIZIA; Agnello, S; Christ, F; Debyser, Z; Chimirri, A. | |
Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones | 1999 | Cecchetti, Violetta; Tabarrini, Oriana; Sabatini, Stefano; Miao, H.; Filipponi, Enrica; Fravolini, Arnaldo | |
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position | 2009 | Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta | |
Synthesis and Antibacterial Evaluation of [1,3]Benzothiazino[3,2-a]quinoline and [3,1]Benzothiazino[1,2-a]quinoline-6-carboxylic Acid Derivatives | 1997 | Cecchetti, Violetta; Cruciani, Gabriele; Filipponi, E.; Fravolini, Arnaldo; Tabarrini, Oriana; Xin, T. | |
Synthesis and biological evaluation of (2S)- and (2R)-2-(3'-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands. | 2006 | Filosa, R.; Marinozzi, Maura; Costantino, Gabriele; Brunsgaard Hemit, M.; Thomsen, C.; Pellicciari, Roberto | |
Synthesis and Biological Evaluation of 2-(3’-(1H-tetrazol-5-yl)bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 Receptor | 2001 | Costantino, Gabriele; Marinozzi, Maura; Camaioni, Emidio; Pellicciari, Roberto; Maltoni, K.; Prezeau, L.; Pin, J. | |
Synthesis and characterization of carnitine nitro-derivatives. | 2008 | Piermatti, Oriana; Fringuelli, Francesco; Pochini, L.; Indiveri, C.; Palmerini, Carlo Alberto | |
Synthesis and preliminary pharmacological evaluation of the four stereoisomers of (2S)-2-(2'-phosphono-3'-phenylcyclopropyl)glycine, the first class of 3'-substituted trans-2-(2'-phosphonocyclopropyl)glycines | 2007 | Marinozzi, Maura; M., Serpi; L., Amori; M., GAVILAN DIAZ; G., Costantino; U., Meyer; P. J., Flor; F., Gasparini; R., Heckendorn; R., Kuhn; G., Giorgi; M., BRUNSGAARD HERMIT; C., Thomsen; R., Pellicciari | |
Synthesis and Prelyminary Pharmacological Evaluation of the Four Stereoisomers of (2S)-2-(2’-Phosphono-3’-phenylcyclopropyl)glycine, the First Stereolibrary of trans 3’- Substituted -2-(2’-Phosphonocyclopropyl) glycine | 2007 | Marinozzi, Maura; M., Serpi; L., Amori; M. G., Diaz; Costantino, Gabriele; U., Mayer; P. J., Flor; F., Gasparini; R., Heckendorn; R., Kuhn; G., Giorgi; M. B., Hermit; C., Thomsen; Pellicciari, Roberto |
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