Sfoglia per Autore
Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design
2022 Palomba, Tommaso; Tassone, Giusy; Vacca, Carmine; Bartalucci, Matteo; Valeri, Aurora; Pozzi, Cecilia; Cross, Simon; Siragusa, Lydia; Desantis, Jenny
Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization
2022 Mercorelli, Beatrice; Desantis, Jenny; Celegato, Marta; Bazzacco, Alessandro; Siragusa, Lydia; Benedetti, Paolo; Eleuteri, Michela; Croci, Federico; Cruciani, Gabriele; Goracci, Laura; Loregian, Arianna
CROMATIC: Cross-Relationship Map of Cavities from Coronaviruses
2022 Siragusa, Lydia; Menna, Gabriele; Buratta, Fabrizio; Baroni, Massimo; Desantis, Jenny; Cruciani, Gabriele; Goracci, Laura
Proteolysis targeting chimeras in antiviral research
2022 Desantis, Jenny; Goracci, Laura
PROTACs bearing piperazine-containing linkers: what effect on their protonation state?
2022 Desantis, Jenny; Mammoli, Andrea; Eleuteri, Michela; Coletti, Alice; Croci, Federico; Macchiarulo, Antonio; Goracci, Laura
An overview on small molecules acting as broad-spectrum agents for yellow fever infection
2022 Desantis, J.; Felicetti, T.; Cannalire, R.
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications
2023 Castellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura
MassChemSite for In-Depth Forced Degradation Analysis of PARP Inhibitors Olaparib, Rucaparib, and Niraparib
2023 Bonciarelli, Stefano; Desantis, Jenny; Cerquiglini, Simone; Goracci, Laura
Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity
2024 Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura
Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis
2024 Eleuteri, Michela; Desantis, Jenny; Cruciani, Gabriele; Germani, Raimondo; Goracci, Laura
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design | 2022 | Palomba, Tommaso; Tassone, Giusy; Vacca, Carmine; Bartalucci, Matteo; Valeri, Aurora; Pozzi, Cecilia; Cross, Simon; Siragusa, Lydia; Desantis, Jenny | |
| Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization | 2022 | Mercorelli, Beatrice; Desantis, Jenny; Celegato, Marta; Bazzacco, Alessandro; Siragusa, Lydia; Benedetti, Paolo; Eleuteri, Michela; Croci, Federico; Cruciani, Gabriele; Goracci, Laura; Loregian, Arianna | |
| CROMATIC: Cross-Relationship Map of Cavities from Coronaviruses | 2022 | Siragusa, Lydia; Menna, Gabriele; Buratta, Fabrizio; Baroni, Massimo; Desantis, Jenny; Cruciani, Gabriele; Goracci, Laura | |
| Proteolysis targeting chimeras in antiviral research | 2022 | Desantis, Jenny; Goracci, Laura | |
| PROTACs bearing piperazine-containing linkers: what effect on their protonation state? | 2022 | Desantis, Jenny; Mammoli, Andrea; Eleuteri, Michela; Coletti, Alice; Croci, Federico; Macchiarulo, Antonio; Goracci, Laura | |
| An overview on small molecules acting as broad-spectrum agents for yellow fever infection | 2022 | Desantis, J.; Felicetti, T.; Cannalire, R. | |
| VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications | 2023 | Castellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura | |
| MassChemSite for In-Depth Forced Degradation Analysis of PARP Inhibitors Olaparib, Rucaparib, and Niraparib | 2023 | Bonciarelli, Stefano; Desantis, Jenny; Cerquiglini, Simone; Goracci, Laura | |
| Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity | 2024 | Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura | |
| Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis | 2024 | Eleuteri, Michela; Desantis, Jenny; Cruciani, Gabriele; Germani, Raimondo; Goracci, Laura |
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