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Farnesoid X receptor: from structure to potential clinical applications. 2005 Pellicciari, Roberto; Costantino, Gabriele; Fiorucci, Stefano
Novel PARP Inhibitors: Synthesis and Molecular Modeling Studies 2005 Pellicciari, Roberto; Camaioni, Emidio; Moroni, F.; Chiarugi, A.; Costantino, Gabriele
Molecular Dynamics Simulation of the Ligand Binding Domain of Farnesoid X Receptor (FXR). Insights into Helix-12 Stability and Coactivator Peptide Stabilization in Response to Agonist Binding 2005 Costantino, Gabriele; Entrena Guadix, A.; Macchiarulo, Antonio; Gioiello, Antimo; Pellicciari, Roberto
Synthesis and Preliminary Biological Evaluation of (2S,1’R,2’S)- and (2S,1’S,2’R)-2-(2Phosphonocyclopropyl)glycines, Two novel Conformationally Constrained L-AP4 Analogues 2005 Amori, L.; Serpi, M.; Marinozzi, Maura; Costantino, Gabriele; Gavilan Diaz, M.; Brunsgaard Hemit, M.; Thomsen, C.; Pellicciari, Roberto
Design, Synthesis, and Microbiolgical Evaluation of New Candida albicans CYP51 Inhibitors 2005 Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Costantino, Gabriele; Pietrella, Donatella; Fringuelli, Renata
Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole. 2005 Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto
Is antagonism of E/Z-guggulsterone at the farnesoid X receptor mediated by a noncanonical binding site? A molecular modeling study. 2005 Meyer, U; Costantino, Gabriele; Macchiarulo, Antonio; Pellicciari, Roberto
Synthesis and preliminary biological evaluation of (2S, 1'R, 2'S)- and (2S, 1'S,2' R)-2-(2-phosphonocyclopropyl)glycines, two novel conformationally constrained L-AP4 analogues 2006 L., Amori; M., Serpi; Marinozzi, Maura; Costantino, Gabriele; M., GAVILAN DIAZ; M., BRUNSGAARD HERMIT; C., Thomsen; Pellicciari, Roberto
Poly(ADP-ribose)-polymerase-catalyzed hydrolysis of NAD+: QM/MM simulation of the enzyme reaction. ChemMedChem. 2006 May;1(5):533-9. 2006 Bellocchi, D; Costantino, Gabriele; Pellicciari, Roberto; Re, N; Marrone, A; Coletti, C.
Poly(ADP-ribose)-Polimerase-Catalyzed Hydrolysis of NAD+: QM/MM Simulation of the Enzyme Reaction 2006 Bellocchi, D.; Costantino, Gabriele; Pellicciari, Roberto; Re, N.; Marrone, A.; Coletti, C.
Design, Molecular Modeling Studies, Synthesis and Preliminary Evaluation of Novel PARP-1 Inhibitors on the Road of Antiischemic Agents 2006 Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; D., Bellocchi; A., Chiarugi; F., Moroni; A., Wood; Pellicciari, Roberto
Modulators of the kynurenine pathway of triptophan metabolism. Synthesis and preliminary biological evaluation of (S)-4-(ethylsulfonyl)benzoylalanine, the first potent and selective kynurenine aminotransferse II (KAT II) inhibitor 2006 Pellicciari, Roberto; Rizzo, R.; Costantino, Gabriele; Marinozzi, Maura; Amori, L.; Guidetti, P.; Wu, H.; Schwarcz, R.
Pharmacophore model for bile acids recognition by the FPR receptor. 2006 Ferrari, Cristina; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto
Potential Therapeutic Applications of Farnesoid X Receptor (FXR) Modulators 2006 Pellicciari, Roberto; Gioiello, Antimo; Costantino, Gabriele
Synthesis and biological evaluation of (2S)- and (2R)-2-(3'-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands. 2006 Filosa, R.; Marinozzi, Maura; Costantino, Gabriele; Brunsgaard Hemit, M.; Thomsen, C.; Pellicciari, Roberto
Synthesis and Prelyminary Pharmacological Evaluation of the Four Stereoisomers of (2S)-2-(2’-Phosphono-3’-phenylcyclopropyl)glycine, the First Stereolibrary of trans 3’- Substituted -2-(2’-Phosphonocyclopropyl) glycine 2007 Marinozzi, Maura; M., Serpi; L., Amori; M. G., Diaz; Costantino, Gabriele; U., Mayer; P. J., Flor; F., Gasparini; R., Heckendorn; R., Kuhn; G., Giorgi; M. B., Hermit; C., Thomsen; Pellicciari, Roberto
Towards Selective PARP-2 Inhibitors: Design, Synthesis and Preliminary Evaluation of a Series of Isoquinolinone Derivatives 2007 Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; L., Formentini; F., Venturoni; D., Bellocchi; G., Eren; A., Chiarugi; F., Moroni; Pellicciari, Roberto
On the Way to Selective PARP-2 Inhibitors: Design, Synthesis and Preliminary Evaluation of a Series of Isoquinolinone Derivatives 2007 Camaioni, Emidio; P., Sabbatini; L., Formentini; F., Venturoni; Costantino, Gabriele; D., Bellocchi; A., Chiarugi; F., Moroni; Pellicciari, Roberto
On the way to selective PARP-2 inhibitors. Design, synthesis, and preliminary evaluation of a series of isoquinolinone derivatives. 2008 Pellicciari, Roberto; Camaioni, Emidio; Costantino, Gabriele; Formentini, L.; Sabbatini, P.; Venturoni, F.; Eren, G.; Bellocchi, D.; Chiarugi, A.; Moroni, F.
Exploring Ligand Recognition in the Kynurenine Pathway to Advance the Medicinal Chemistry of Kynurenines 2009 Macchiarulo, Antonio; L., Amori; D., Bellocchi; Camaioni, Emidio; Carotti, Andrea; A., Chiarugi; Costantino, Gabriele; Marinozzi, Maura; Nuti, Roberto; . F., Venturoni; R., Schwarcz; F., Moroni; Pellicciari, Roberto
Mostrati risultati da 61 a 80 di 85
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