Sfoglia per Autore
Modeling of Amino-Terminal Domains of Group I Metabotropic Glutamate Receptors: Structural Motifs Affecting Ligand Selectivity
1999 Costantino, G.; Pellicciari, Roberto; Macchiarulo, Antonio
Pharmacophore Models of Group I and Group II Metabotropic Glutamate Receptors Agonists. Analysis of Conformational, Steric and Topological Parameters Affecting Potency and Selectivity
1999 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Metabotropic Glutamate Receptors: A Structural View Point
2000 Pellicciari, Roberto; Costantino, Gabriele; Macchiarulo, Antonio
New potent and selective mGluR1 competitive antagonists: pharmacological characterization and their exploitation in molecular modeling of receptor blocking
2001 Costantino, Gabriele; Camaioni, Emidio; Macchiarulo, Antonio; D., Pellegrini Giampietro; F., Moroni; Pellicciari, Roberto
Exploring the Molecular Dasis of the Selectivity in Metabotropic Glutamate Receptors (mGluRs)
2001 Macchiarulo, Antonio; R., Sbaglia; S., Aiello; M., Meniconi; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Pellicciari, Roberto
Metabotropic Glutamate Receptors: Targets for Therapy of Cerebral Ischemia
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Design, Synthesis and Preliminay Evaluation of Novel 3’-Substituted Carboxycyclopropylglycines as Antagonists at Group 2 Metabotropic Glutamate Receptors
2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Amori, L.; Flor, P.; Gasparini, F.; Kuhn, R.; Urwyler, S.
Metabotropic glutamate receptors: structure and new subtype-selective ligands
2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Camaioni, Emidio; Natalini, Benedetto
Conformational analysis of carboxyphenylglycine (CPG) Derivatives: insight into bioactive and bioselective conformations of group-I mGluRs antagonists.
2001 Macchiarulo, Antonio; Entrena Guadix, A.; Costantino, G.
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
QSAR and Molecular Modeling Studies of Baclofen Analogues as GABAB Agonists. Insights into the Role of the Aromatic Moiety in GABAB Binding Activation
2001 Costantino, G.; Pellicciari, Roberto; Macchiarulo, Antonio; Entrena Guadix, A.
Modeling of Poly(ADP-ribose)polymerase (PARP) Inhibitors. Docking of Ligands and QSAR
2001 Costantino, G.; Macchiarulo, Antonio; Camaioni, Emidio; Pellicciari, Roberto
Homology Modeling of AMPA Receptors: Route to the identification of noncompetitive antagonists binding site
2002 Barreca, MARIA LETIZIA; Chimirri, A.; Costantino, Gabriele; De Luca, L.; Gitto, R.; Macchiarulo, Antonio; Pellicciari, R.
Molecular determinats for metabotropic glutamate receptor activation and blockade. Molecular dynamics and electrostatic potential analysis studies
2002 Costantino, Gabriele; M., Belenekin; Macchiarulo, Antonio; Camaioni, Emidio; Pellicciari, Roberto
Spiro[2.2]pentane as a dyssymetric scaffold for conformationally constrained analogues of glutamic acid: diastereodivergent synthesis of 1-aminospiro[2.2]pentyl-1,4-dicarboxylic acids
2002 Marinozzi, Maura; Camaioni, Emidio; Costantino, Gabriele; G., Giorgi; Macchiarulo, Antonio; Pellicciari, Roberto
Molecular dynamics simulation of the ligand binding domain of mGluR1 in response to agonist and antagonist binding.
2002 Costantino, Gabriele; Macchiarulo, Antonio; Belenikin, M.; Pellicciari, R.
Glucocorticoid-induced leucine zipper inhibits the Raf-extracellular signal-regulated kinase pathway by binding to Raf-1
2002 Ayroldi, Emira Maria; Zollo, Ornella; Macchiarulo, Antonio; DI MARCO, Barbara; Marchetti, Maria Cristina; Riccardi, Carlo
1,4 Benzothiazine and 1,4 benzoxazine imidazole derivatives with antifungal activity: a docking study
2002 Macchiarulo, Antonio; Costantino, Gabriele; Fringuelli, D.; Vecchiarelli, Anna; Schiaffella, Fausto; Fringuelli, Renata
Spiro[2.2]pentane as a Dissymmetric Scaffold for Conformationally Constrained Analogues of Glutamic Acid: Focus on Racemic 1-Aminospiro[2.2]pentyl-1,4-dicarboxylic Acids
2002 Pellicciari, Roberto; Marinozzi, Maura; Camaioni, Emidio; Costantino, Gabriele; Nunez, M.; Gasparini, F.; Giorgi, G.; Macchiarulo, Antonio; Subramanian, N.
Glucocorticoid Induced Leucine Zipper (GILZ) inhibits the RAF-ERK pathway by binding to RAF-1
2002 Ayroldi, Emira Maria; Zollo, Ornella; Macchiarulo, Antonio; DI MARCO, Barbara; Marchetti, C; Riccardi, Carlo
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