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Mostrati risultati da 21 a 40 di 48
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Discovery that theonellasterol a marine sponge sterol is a highly selective FXR antagonist that protects against liver injury in cholestasis. 2012 Renga, Barbara; Mencarelli, Andrea; D'Amore, Claudio; Cipriani, Sabrina; D'Auria, Mv; Sepe, V; Chini, Mg; Monti, Mc; Bifulco, G; Zampella, A; Fiorucci, Stefano
Role of Maraviroc in a dyslipidemic murine model of atherosclerosis RTV-induced 2013 Cipriani, Sabrina; Mencarelli, Andrea; Francisci, Daniela; Renga, Barbara; Schiaroli, Elisabetta; D'Amore, Claudio; Fiorucci, Stefano; Baldelli, Franco
A Novel Source of Intestinal Damage: The HIV Protease Inhibitor Ritonavir Worsens Damage Caused by COX Inhibitors 2013 Mencarelli, A; Renga, B; Cipriani, S; D'Amore, C; Francisci, D; Baldelli, F; Distrutti, E; Donini, A; Fiorucci, S
Oxygenated polyketides from Plakinastrella mamillaris as a new chemotype of PXR agonists. 2013 Festa, C; D'Amore, Claudio; Renga, Barbara; Lauro, G; De Marino, S; D'Auria, Mv; Bifulco, G; Zampella, A; Fiorucci, Stefano
Binding mechanism of the farnesoid X receptor marine antagonist suvanine reveals a strategy to forestall drug modulation on nuclear receptors. Design, synthesis, and biological evaluation of novel ligands. 2013 Di Leva, Fs; Festa, C; D'Amore, Claudio; De Marino, S; Renga, Barbara; D'Auria, Mv; Novellino, E; Limongelli, V; Zampella, A; Fiorucci, Stefano
FXR mediates a chromatin looping in the GR promoter thus promoting the resolution of colitis in rodents. 2013 Renga, Barbara; D'Amore, Claudio; Cipriani, Sabrina; Mencarelli, Andrea; Carino, A; Sepe, V; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
Dissociation of intestinal and hepatic activities of FXR and LXRα supports metabolic effects of terminal ileum interposition in rodents. 2013 Mencarelli, Andrea; Renga, Barbara; D'Amore, Claudio; Santorelli, C; Graziosi, L; Bruno, A; Monti, Mc; Distrutti, Eleonora; Cipriani, Sabrina; Donini, Annibale; Fiorucci, Stefano
Efficacy of the CCR5 antagonist maraviroc in reducing early, ritonavir-induced atherogenesis and advanced plaque progression in mice. 2013 Cipriani, Sabrina; Francisci, Daniela; Mencarelli, Andrea; Renga, Barbara; Schiaroli, Elisabetta; D'Amore, Claudio; Baldelli, Franco; Fiorucci, Stefano
CCR5 Antagonism by Maraviroc Reduces the Potential for Gastric Cancer Cell Dissemination. 2013 Mencarelli, Andrea; Graziosi, L; Renga, Barbara; Cipriani, Sabrina; D'Amore, Claudio; Francisci, Daniela; Bruno, A; Baldelli, Franco; Donini, Annibale; Fiorucci, Stefano
New tridecapeptides of the theonellapeptolide family from the Indonesian sponge Theonella swinhoei. 2013 Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O.
Isoswinholide B and swinholide K, potently cytotoxic dimeric macrolides from Theonella swinhoei. 2013 Sinisi, A; Calcinai, B; Cerrano, C; Dien, Ha; Zampella, A; D'Amore, Claudio; Renga, Barbara; Fiorucci, Stefano; Taglialatela Scafati, O.
The CCR5 Antagonist Maraviroc Reduces the Potential for Gastric Cancer Dissemination in Rodent Models of Peritoneal Metastasis 2013 Renga, B; D'Amore, C; Graziosi, L; Mencarelli, A; Bruno, A; Francisci, D; Baldelli, F; Distrutti, E; Donini, A; Fiorucci, S; Cavazzoni, E
The bile acid sensor FXR is required for immune-regulatory activities of TLR-9 in intestinal inflammation 2013 Renga, Barbara; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Carino, A; Bruno, A; Francisci, Daniela; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
Solomonsterol A, a marine pregnane-X-receptor agonist, attenuates inflammation and immune dysfunction in a mouse model of arthritis. 2013 Mencarelli, Andrea; D'Amore, Claudio; Renga, Barbara; Cipriani, Sabrina; Carino, A; Sepe, V; Perissutti, E; D'Auria, Mv; Zampella, A; Distrutti, Eleonora; Fiorucci, Stefano; Carino, Adriana
Epigenetic modulation by methionine deficiency attenuates the potential for gastric cancer cell dissemination. 2013 Graziosi, Luigina; Mencarelli, Andrea; Renga, Barbara; D'Amore, Claudio; Bruno, A; Santorelli, C; Cavazzoni, Emanuel; Cantarella, Francesco; Rosati, E; Donini, Annibale; Fiorucci, Stefano
The HIV Matrix Protein p17 promotes the Activation of human hepatic stellate cells through interactions with CXCR2 and Syndecan-2 2014 Renga, Barbara; Francisci, Daniela; Schiaroli, Elisabetta; Carino, A; Cipriani, Sabrina; D'Amore, Claudio; Sidoni, Angelo; DEL SORDO, Rachele; Ferri, Ivana; Lucattelli, M; Lunghi, B; Baldelli, Franco; Fiorucci, Stefano; Carino, Adriana
Bazedoxifene-scaffold-based mimetics of solomonsterols A and B as novel pregnane X receptor antagonists. 2014 Hodnik, Ž; Peterlin Mašič, L; Tomašić, T; Smodiš, D; D'Amore, Claudio; Fiorucci, Stefano; Kikelj, D.
Exploitation of cholane scaffold for the discovery of potent and selective farnesoid X receptor (FXR) and G-protein coupled bile acid receptor 1 (GP-BAR1) ligands 2014 Festa, C; Renga, Barbara; D'Amore, Claudio; Sepe, V; Finamore, C; De Marino, S; Carino, A.; Cipriani, Sabrina; Monti, Mc; Zampella, A; Fiorucci, Stefano; Carino, Adriana
Design, synthesis, and biological evaluation of potent dual agonists of nuclear and membrane bile acid receptors. 2014 D'Amore, Claudio; Di Leva, Fs; Sepe, V; Renga, Barbara; Del Gaudio, C; D'Auria, Mv; Zampella, A; Fiorucci, Stefano; Limongelli, V.
In vivo administration of ritonavir worsens intestinal damage caused by cyclooxygease inhibitors. 2014 Renga, Barbara; Mencarelli, Andrea; Cipriani, Sabrina; D'Amore, Claudio; Francisci, Daniela; Santucci, L; Baldelli, Franco; Distrutti, Eleonora; Fiorucci, Stefano
Mostrati risultati da 21 a 40 di 48
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