Sfoglia per Autore
Dirhodium(II)-tetraacetate-Mediated Decomposition of Ethyldiazo- acetate and Ethyldiazomalonate in the Presence of Fullerene. A New Procedure for the Selective Synthesis of [6-6]-Closed Methanofullerenes
1997 Pellicciari, Roberto; Annibali, D; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto
Metabotropic glutamate receptors: new ligands and molecular modelling studies
1997 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; C., Thomsen; F., Moroni
Modulation of glutamate receptor pathways in the search for new neuroprotective agents
1998 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto
"*-Diazocarbonyl Chemistry - Target Driven Applications"
1998 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Mattoli, L.; Natalini, Benedetto
Asymmetric synthesis of (2R, 1’S, 2’R, 3’S)-2-(2’- Carboxy-3’-phenylcyclopropyl)glicine (PCCG 13), the first selective antagonist of metabotropic glutamate receptors coupled phospholipase D
1998 Marinozzi, Maura; Costantino, Gabriele; D. E., Pellegrini Giampietro; Pellicciari, Roberto
Pharmacophore Models of Group I and Group II Metabotropic Glutamate Receptors Agonists. Analysis of Conformational, Steric and Topological Parameters Affecting Potency and Selectivity
1999 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Evaluation of Hydrophobic/Hydrophilic Balance of Bile Acids by Comparative Molecular Field Analysis (CoMFA)
2000 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; Wolf, C.
Metabotropic Glutamate Receptors: A Structural View Point
2000 Pellicciari, Roberto; Costantino, Gabriele; Macchiarulo, Antonio
Synthesis, Molecular Modeling and Preliminary Biological Evaluation of 1-Amino-3-Phospono-3-Cyclopentene-1-Carboxylic acid and 1-Amino-3-Phosphono-2-Cyclopentene-1-Carboxylic acid, Two Novel Agonists of Metabotropic Glutamate Receptors of Group III
2000 Costantino, Gabriele; Marinozzi, Maura; Pellicciari, Roberto; Amori, L.; Gasparini, F.; Flor, P.; Kuhn, R.; Vranesic, I.
Chromatographic separation and evaluation of the lipophilicity by reversed-phase high-performance liquid chromatography of fullerene-C60 derivatives
2001 Natalini, Benedetto; Marinozzi, Maura; Costantino, Gabriele; Pellicciari, Roberto; Capodiferro, V.; Mattoli, L.
Metabotropic glutamate receptors: structure and new subtype-selective ligands
2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Camaioni, Emidio; Natalini, Benedetto
Design, Synthesis and Preliminay Evaluation of Novel 3’-Substituted Carboxycyclopropylglycines as Antagonists at Group 2 Metabotropic Glutamate Receptors
2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Amori, L.; Flor, P.; Gasparini, F.; Kuhn, R.; Urwyler, S.
Exploring the Molecular Dasis of the Selectivity in Metabotropic Glutamate Receptors (mGluRs)
2001 Macchiarulo, Antonio; R., Sbaglia; S., Aiello; M., Meniconi; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Pellicciari, Roberto
New potent and selective mGluR1 competitive antagonists: pharmacological characterization and their exploitation in molecular modeling of receptor blocking
2001 Costantino, Gabriele; Camaioni, Emidio; Macchiarulo, Antonio; D., Pellegrini Giampietro; F., Moroni; Pellicciari, Roberto
(2R,1’S,2’R,3’S)-2-(2’-Carboxy-3’-phenylcyclopropyl)glycine (PCCG-13), the First Potent and Selective Competitive Antagonist of Phospholipase D-Coupled Metabotropic Glutamate Receptors: Asymmetric Synthesis and Preliminary Biological Properties
2001 Pellicciari, Roberto; Marinozzi, Maura; Costantino, Gabriele; Natalini, Benedetto; Moroni, F.; Pellegrini Giampietro, D.
Synthesis and Preliminary Biological Evaluation of glycineb site (+)- and (-)-3-Oxetanylglycine, Novel non-Proteinogenic Amino Acids
2001 Costantino, Gabriele; Marinozzi, Maura; Pellicciari, Roberto; Teran Moldes, M.
Metabotropic Glutamate Receptors: Targets for Therapy of Cerebral Ischemia
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Synthesis and Biological Evaluation of 2-(3’-(1H-tetrazol-5-yl)bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 Receptor
2001 Costantino, Gabriele; Marinozzi, Maura; Camaioni, Emidio; Pellicciari, Roberto; Maltoni, K.; Prezeau, L.; Pin, J.
Homology Model of the Closed, Functionally Active, Form of the Amino Terminal Domain of mGluR1
2001 Costantino, Gabriele; Pellicciari, Roberto; Macchiarulo, Antonio
Molecular dynamics simulation of the ligand binding domain of mGluR1 in response to agonist and antagonist binding.
2002 Costantino, Gabriele; Macchiarulo, Antonio; Belenikin, M.; Pellicciari, R.
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