CERNICCHI, GIADA
CERNICCHI, GIADA
Dipartimento di Scienze Farmaceutiche
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity
2022 Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana
Discovery of 2‐phenylquinazolines as potent Mycobacterium avium efflux pump inhibitors able to synergize with clarithromycin against clinical isolate
2024 Cernicchi, Giada; Rampacci, Elisa; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Cecchetti, Violetta; Felicetti, Tommaso; Di Luca, Mariagrazia; Poma, Noemi Violeta; Tavanti, Arianna; Passamonti, Fabrizio; Rindi, Laura; Sabatini, Stefano
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
2021 Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano
In Vitro and In Vivo Investigations into the Potential of Quinazoline and Quinoline Derivatives as NorA Efflux Pump Inhibitors Against Resistant Staphylococcus aureus Strains
2025 Chandal, Nishtha; Sharma, Nidhi; Cernicchi, Giada; Felicetti, Tommaso; Rondini, Tommaso; Acito, Mattia; Nandanwar, Hemraj; Sabatini, Stefano
Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors
2023 Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio
Microbial efflux pump inhibitors: A journey around quinoline and indole derivatives
2021 Cernicchi, G.; Felicetti, T.; Sabatini, S.
New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains
2022 Felicetti, Tommaso; Cedraro, Nicholas; Astolfi, Andrea; Cernicchi, Giada; Mangiaterra, Gianmarco; Vaiasicca, Salvatore; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Biavasco, Francesca; Cecchetti, Violetta; Vignaroli, Carla; Sabatini, Stefano
NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3‐c][1,2]benzothiazine 5,5‐Dioxide Derivatives
2025 Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity | 2022 | Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana | |
| Discovery of 2‐phenylquinazolines as potent Mycobacterium avium efflux pump inhibitors able to synergize with clarithromycin against clinical isolate | 2024 | Cernicchi, Giada; Rampacci, Elisa; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Cecchetti, Violetta; Felicetti, Tommaso; Di Luca, Mariagrazia; Poma, Noemi Violeta; Tavanti, Arianna; Passamonti, Fabrizio; Rindi, Laura; Sabatini, Stefano | |
| From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | 2021 | Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano | |
| In Vitro and In Vivo Investigations into the Potential of Quinazoline and Quinoline Derivatives as NorA Efflux Pump Inhibitors Against Resistant Staphylococcus aureus Strains | 2025 | Chandal, Nishtha; Sharma, Nidhi; Cernicchi, Giada; Felicetti, Tommaso; Rondini, Tommaso; Acito, Mattia; Nandanwar, Hemraj; Sabatini, Stefano | |
| Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors | 2023 | Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio | |
| Microbial efflux pump inhibitors: A journey around quinoline and indole derivatives | 2021 | Cernicchi, G.; Felicetti, T.; Sabatini, S. | |
| New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains | 2022 | Felicetti, Tommaso; Cedraro, Nicholas; Astolfi, Andrea; Cernicchi, Giada; Mangiaterra, Gianmarco; Vaiasicca, Salvatore; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Biavasco, Francesca; Cecchetti, Violetta; Vignaroli, Carla; Sabatini, Stefano | |
| NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3‐c][1,2]benzothiazine 5,5‐Dioxide Derivatives | 2025 | Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano |