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Binding Mode and Structure-Activity Relationships of ITE as an Aryl Hydrocarbon Receptor (AhR) Agonist 2018 Dolciami, Daniela; Gargaro, Marco; Cerra, Bruno; Scalisi, Giulia; Bagnoli, Luana; Servillo, Giuseppe; Della, FAZIA MARIA AGNESE; Puccetti, Paolo; Quintana, Francisco J.; Fallarino, Francesca; Macchiarulo, Antonio
BF3·Et2O-Promoted Decomposition of Cyclic α-Diazo-β-Hydroxy Ketones: Novel Insights into Mechanistic Aspects 2018 Venturoni, Francesco; Cerra, Bruno; Marinozzi, Maura; Camaioni, Emidio; Gioiello, Antimo; Pellicciari, Roberto
Flow Nanoprecipitation of Size-Controlled D-Leucine Nanoparticles as Excipient for Spray-Drying Formulations 2019 Cerra, B.; Mosca, G.; TALI SHANDIZ, Shiva; Ricci, M.; Schoubben, A.; Gioiello, A.
Mesofluidic Flash Nanoprecipitation of D-Leucine Particles as Excipient in Powders for Inhalation 2019 Mosca, G.; Cerra, B.; Gioiello, A.; Ricci, M.; Schoubben, A.
Exploiting Chemical Toolboxes for the Expedited Generation of Tetracyclic Quinolines as a Novel Class of PXR Agonists 2019 Cerra, B.; Carotti, A.; Passeri, D.; Sardella, R.; Moroni, G.; Di Michele, A.; Macchiarulo, A.; Pellicciari, R.; Gioiello, A.
Optimisation by design of experiment of benzimidazol-2-one synthesis under flow conditions 2019 Mostarda, S.; Maz, T. G.; Piccinno, A.; Cerra, B.; Banoglu, E.
Flow nanoprecipitation of size-controlled d-leucine nanoparticles for spray-drying formulations 2019 Cerra, B.; Mosca, G.; Ricci, M.; Schoubben, A.; Gioiello, A.
Identification and quantification of oxo-bile acids in human faeces with liquid chromatography–mass spectrometry: A potent tool for human gut acidic sterolbiome studies 2019 Franco, P.; Porru, E.; Fiori, J.; Gioiello, A.; Cerra, B.; Roda, G.; Caliceti, C.; Simoni, P.; Roda, A.
Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor 2020 Bartolini, D.; De Franco, F.; Torquato, P.; Marinelli, R.; Cerra, B.; Ronchetti, R.; Schon, A.; Fallarino, F.; De Luca, A.; Bellezza, G.; Ferri, I.; Sidoni, A.; Walton, W. G.; Pellock, S. J.; Redinbo, M. R.; Mani, S.; Pellicciari, R.; Gioiello, A.; Galli, F.
A streamlined synthesis of the neurosteroid 3β-methoxypregnenolone assisted by a statistical experimental design and automation 2020 Mancino, Valentina; Croci, Federico; Lozza, ANNA MARIA; Cerra, Bruno; Gioiello, Antimo
Enantioselective HPLC analysis to assist the chemical exploration of chiral imidazolines 2020 Cerra, B.; Macchiarulo, A.; Carotti, A.; Camaioni, E.; Varfaj, I.; Sardella, R.; Gioiello, A.
Integrating experimental and computational techniques to study chromatographic enantioresolutions of chiral tetrahydroindazole derivatives 2020 Ianni, Federica; Cerra, Bruno; Shandiz, Shiva Tali; Michele, Alessandro Di; Saluti, Giorgio; Galarini, Roberta; Gioiello, Antimo; Sardella, Roccaldo; Carotti, Andrea
The Medicinal Chemistry in the Era of Machines and Automation: Recent Advances in Continuous Flow Technology 2020 Gioiello, A; Piccinno, A; Lozza, Am; Cerra, B
The Stone Guest: How Does pH Affect Binding Properties of PD-1/PD-L1 Inhibitors? 2021 Riccio, A.; Coletti, A.; Dolciami, D.; Mammoli, A.; Cerra, B.; Moretti, S.; Gioiello, A.; Ferlin, S.; Puxeddu, E.; Macchiarulo, A.
Future medicinal chemists experience flow chemistry: optimization by experimental design of the limiting synthetic step to the antifungal drug econazole nitrate 2021 Cerra, B.; Gioiello, A.
Integrated Systems for Continuous Synthesis and Biological Screenings 2022 Gioiello, Antimo; Moroni, Giada; Cerra, Bruno
Development of 3α, 7α-dihydroxy-6α-ethyl-24-nor-5β-cholan-23-sulfate sodium salt (INT-767): Process optimization, synthesis and characterization of metabolites 2022 Cerra, Bruno; Venturoni, Francesco; Souma, Maria; Ceccarelli, Giada; Maria Lozza, Anna; Passeri, Daniela; De Franco, Francesca; R Baxendale, Ian; Pellicciari, Roberto; Macchiarulo, Antonio; Gioiello, Antimo
Combining molecular modeling approaches to establish the chromatographic enantiomer elution order in the absence of pure enantiomeric standards: A study case with two tetracyclic quinolines 2022 Ianni, F; Cerra, B; Moroni, G; Varfaj, I; Di Michele, A; Gioiello, A; Carotti, A; Sardella, R
Continuous Flow Synthesis of the PARP-1/2 Inhibitor HYDAMTIQ: Synthetic Strategy, Optimization, and Green Metrics Evaluation 2023 Filipponi, Paolo; Cerra, Bruno; Piccinno, Alessandro; Camaioni, Emidio; Gioiello, Antimo
Multi-Gram Scale Synthesis and Characterization of Mometasone Furoate EP Impurity C 2023 Ronchetti, Riccardo; Pannone, Luigi Alfonso; Cerra, Bruno; Camaioni, Emidio; Lopopolo, Gianfranco; Attolino, Emanuele; Gioiello, Antimo
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