Sfoglia per Autore
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
2010 Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Response of a simian immunodeficiency virus (SIVmac251) to raltegravir: a basis for a new treatment for simian AIDS and an animal model for studying lentiviral persistence during antiretroviral therapy.
2010 Lewis, M. G.; Norelli, S.; Collins, M.; Barreca, M. L.; Iraci, Nunzio; Chirullo, B.; Yalley Ogunro, J.; Greenhouse, J.; Titti, F.; Garaci, E.; Savarino, A.; Barreca, MARIA LETIZIA
Designed Multiple Ligands (DLMs) as innovative anti-HIV agents
2010 Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Sabatini, Stefano; Daelemans, D.; Pannecouque, C.; Cecchetti, Violetta; Tabarrini, Oriana
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development
2011 Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Cecchetti, Violetta
RE-EVOLUTION OF THE 2-PHENYL-4-HYDROXYQUINOLINES: OPTIMIZATION OF A POTENT NEW CLASS OF S. AUREUS NorA EFFLUX PUMP INHIBITORS
2012 S., Serritella; Gosetto, Francesca; Iraci, Nunzio; Sancineto, Luca; Sabatini, Stefano; Cecchetti, Violetta
Structural optimization of the 2-Phenyl-4-hydroxyquinoline Class of S. aureus NorA Efflux Pump Inhibitors
2012 Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; A. M., Schito; G. W., Kaatz; Cecchetti, Violetta
Targeting the HIV Tat-mediated transcriptional machinery: P-TEFb complex inhibitors
2012 Tabarrini, Oriana; Sancineto, Luca; Iraci, Nunzio; Massari, Serena; V., Attanasio; Sabatini, Stefano; Manfroni, Giuseppe; A., Marcello; Cecchetti, Violetta
New chemotypes to fight HCV infection: discovery of selective inhibitors of HCV replication with pyrazolobenzothiazine scaffold
2012 Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Iraci, Nunzio; Cannalire, R.; Tabarrini, Oriana; Cecchetti, Violetta
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase
2012 Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta
A highly intensified ART regimen induces long-term viral suppression and restriction of the viral reservoir in a simian AIDS model.
2012 Shytaj, Il; Norelli, S; Chirullo, B; Della Corte, A; Collins, M; Yalley Ogunro, J; Greenhouse, J; Iraci, Nunzio; Acosta, Ep; Barreca, MARIA LETIZIA; Lewis, Mg; Savarino, A.
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors
2012 Sabatini, Stefano; Gosetto, F; Serritella, S; Manfroni, Giuseppe; Tabarrini, Oriana; Iraci, Nunzio; Brincat, Jp; Carosati, Emanuele; Villarini, Milena; Kaatz, Gw; Cecchetti, Violetta
Prion protein ligands as therapeutic agents for neurodegenerative disorders
2013 Biasini, Emiliano; Harris, David A.; Beeler, Aaron; Fluharty, Brian R.; Barreca, MARIA LETIZIA; Iraci, Nunzio; Ingham, Oscar
TARGETING CDKs TO INHIBIT THE HIV-1 TAT-MEDIATED TRANSCRIPTION
2013 Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Targeting CDKs to inhibit the HIV-1 TAT-mediated transcription
2013 Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance
2013 Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta
Structure-Based Discovery of Pyrazolobenzothiazine Derivatives As Inhibitors of Hepatitis C Virus Replication
2013 Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Pieter, Leyssen; Johan, Winquist; Neerja Kaushik, Basu; Jan, Paeshuyse; Ramalingam, Krishnan; Iraci, Nunzio; Sabatini, Stefano; Tabarrini, Oriana; Amartya, Basu; U., Helena Danielson; Johan, Neyts; Cecchetti, Violetta
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana
From Small to Powerful: The Fragments Universe and its "Chem-Appeal"
2013 Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Tabarrini, Oriana
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel 1,3-dihydro-benzimidazol-2-ones and their analogues as potent non-nucleoside HIV-1 reverse transcriptase inhibitors. | 2010 | Monforte, A. M.; Logoteta, P.; De Luca, L.; Iraci, Nunzio; Ferro, S.; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A. | |
Response of a simian immunodeficiency virus (SIVmac251) to raltegravir: a basis for a new treatment for simian AIDS and an animal model for studying lentiviral persistence during antiretroviral therapy. | 2010 | Lewis, M. G.; Norelli, S.; Collins, M.; Barreca, M. L.; Iraci, Nunzio; Chirullo, B.; Yalley Ogunro, J.; Greenhouse, J.; Titti, F.; Garaci, E.; Savarino, A.; Barreca, MARIA LETIZIA | |
Designed Multiple Ligands (DLMs) as innovative anti-HIV agents | 2010 | Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Sabatini, Stefano; Daelemans, D.; Pannecouque, C.; Cecchetti, Violetta; Tabarrini, Oriana | |
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development | 2011 | Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Cecchetti, Violetta | |
RE-EVOLUTION OF THE 2-PHENYL-4-HYDROXYQUINOLINES: OPTIMIZATION OF A POTENT NEW CLASS OF S. AUREUS NorA EFFLUX PUMP INHIBITORS | 2012 | S., Serritella; Gosetto, Francesca; Iraci, Nunzio; Sancineto, Luca; Sabatini, Stefano; Cecchetti, Violetta | |
Structural optimization of the 2-Phenyl-4-hydroxyquinoline Class of S. aureus NorA Efflux Pump Inhibitors | 2012 | Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; A. M., Schito; G. W., Kaatz; Cecchetti, Violetta | |
Targeting the HIV Tat-mediated transcriptional machinery: P-TEFb complex inhibitors | 2012 | Tabarrini, Oriana; Sancineto, Luca; Iraci, Nunzio; Massari, Serena; V., Attanasio; Sabatini, Stefano; Manfroni, Giuseppe; A., Marcello; Cecchetti, Violetta | |
New chemotypes to fight HCV infection: discovery of selective inhibitors of HCV replication with pyrazolobenzothiazine scaffold | 2012 | Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Iraci, Nunzio; Cannalire, R.; Tabarrini, Oriana; Cecchetti, Violetta | |
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase | 2012 | Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta | |
A highly intensified ART regimen induces long-term viral suppression and restriction of the viral reservoir in a simian AIDS model. | 2012 | Shytaj, Il; Norelli, S; Chirullo, B; Della Corte, A; Collins, M; Yalley Ogunro, J; Greenhouse, J; Iraci, Nunzio; Acosta, Ep; Barreca, MARIA LETIZIA; Lewis, Mg; Savarino, A. | |
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors | 2012 | Sabatini, Stefano; Gosetto, F; Serritella, S; Manfroni, Giuseppe; Tabarrini, Oriana; Iraci, Nunzio; Brincat, Jp; Carosati, Emanuele; Villarini, Milena; Kaatz, Gw; Cecchetti, Violetta | |
Prion protein ligands as therapeutic agents for neurodegenerative disorders | 2013 | Biasini, Emiliano; Harris, David A.; Beeler, Aaron; Fluharty, Brian R.; Barreca, MARIA LETIZIA; Iraci, Nunzio; Ingham, Oscar | |
TARGETING CDKs TO INHIBIT THE HIV-1 TAT-MEDIATED TRANSCRIPTION | 2013 | Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Targeting CDKs to inhibit the HIV-1 TAT-mediated transcription | 2013 | Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance | 2013 | Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta | |
Structure-Based Discovery of Pyrazolobenzothiazine Derivatives As Inhibitors of Hepatitis C Virus Replication | 2013 | Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Pieter, Leyssen; Johan, Winquist; Neerja Kaushik, Basu; Jan, Paeshuyse; Ramalingam, Krishnan; Iraci, Nunzio; Sabatini, Stefano; Tabarrini, Oriana; Amartya, Basu; U., Helena Danielson; Johan, Neyts; Cecchetti, Violetta | |
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana | |
From Small to Powerful: The Fragments Universe and its "Chem-Appeal" | 2013 | Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Tabarrini, Oriana |
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