Sfoglia per Autore
Predictive models for hERG potassium channel blockers
2005 Cianchetta, Giovanni; Li, Y.; Kang, J.; Rampe, D.; Fravolini, Arnaldo; Cruciani, Gabriele; Vaz, R. J.
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation.
2005 Stevens, M.; Balzarini, J.; Tabarrini, Oriana; Andrei, G.; Snoeck, R.; Cecchetti, Violetta; Fravolini, Arnaldo; De Clercq, E.; Pannecouque, C.
A pharmacophore hypothesis for P-glycoprotein substrate recognition using GRIND-based 3D-QSAR.
2005 Cianchetta, Giovanni; Singleton, R. W.; Zhang, M.; Wildgoose, M.; Giesing, D.; Fravolini, Arnaldo; Cruciani, Gabriele; Vaz, R. J.
2-phenylquinolones as HIV-1 Tat/TAR interaction inhibitors
2006 Manfroni, Giuseppe; Tabarrini, Oriana; Sabatini, Stefano; Gatto, B.; Giaretta, G.; Palumbo, M.; Parolin, C.; Fravolini, Arnaldo; Cecchetti, V.
Synthesis and Activity of New Modified 1,4-Benzothiazine Derivatives as Inhibitors of the NorA Efflux Pump of Staphylococcus aureus
2006 Sabatini, Stefano; Giuliani, F.; Fusi, C.; Cecchetti, Violetta; Rossolini, G. M.; Fravolini, Arnaldo
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition. Abstr. P62
2006 Gatto, B; Giaretta, G; Palumbo, M; Richter, S; Parolin, C; Palu, G; Tabarrini, Oriana; Fravolini, Arnaldo; Cecchetti, Violetta
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition
2006 Gatto, B.; Giaretta, G.; Palumbo, M.; Richter, S.; Parolin, C.; Palù, G.; Tabarrini, Oriana; Fravolini, Arnaldo; Cecchetti, Violetta
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents
2006 Tabarrini, Oriana; Manfroni, Giuseppe; Fravolini, Arnaldo; Cecchetti, Violetta; Sabatini, Stefano; De Clercq, E.; Rozenski, J.; Canard, B.; Dutartre, H.; Paeshuyse, J.; Neyts, J.
Derivati 2-fenilchinolonici come inibitori della pompa di efflusso NorA dello Staphylococcus aureus ciprofloxacin resistente
2007 Sabatini, Stefano; Pieroni, Marco; Manfroni, Giuseppe; Giuliani, F.; Rossolini, G. M.; Fravolini, Arnaldo
Novel In Vivo Model for the Study of Human Immunodeficiency Virus Type 1 Transcription Inhibitors: Evaluation of New 6-Desfluoroquinolone Derivatives
2007 Stevens, M.; Pollicita, M.; Pannecouque, C.; Verbeken, E.; Tabarrini, Oriana; Cecchetti, Violetta; Acquaro, S.; Perno, C. F.; Fravolini, Arnaldo; De Clercq, E.; Schols, D.; Balzarini, J.
Structure-activity relationship study on anti-HIV 6-desfluoroquinolones.
2008 Tabarrini, Oriana; Massari, Serena; Daelemans, D.; Stevens, M.; Manfroni, Giuseppe; Sabatini, Stefano; Balzarini, J.; Cecchetti, Violetta; Pannecouque, C.; Fravolini, Arnaldo
From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump.
2008 Sabatini, Stefano; Kaatz, G. W.; Rossolini, G. M.; Brandini, David; Fravolini, Arnaldo
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump
2009 Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta; Fravolini, Arnaldo
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump
2009 Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta; Fravolini, Arnaldo
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor.
2009 Manfroni, Giuseppe; Paeshuyse, J; Massari, Serena; Gatto, B; Zanoli, S; Maga, G; Tabarrini, Oriana; Cecchetti, Violetta; Fravolini, Arnaldo; Neyts, J.
Syhtesis and Biological Evaluation of 2-Phenylquinolones Targeted at Tat/TAR Recognition
2009 Manfroni, Giuseppe; Gatto, B; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta; Giaretta, G; Parolin, C; DEL VECCHIO, C; Calisti, A; Palumbo, M; Fravolini, Arnaldo
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction.
2009 Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta
From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps.
2010 Pieroni, Marco; M., Dimovska; Brincat, JEAN PIERRE; Sabatini, Stefano; Carosati, Emanuele; Massari, Serena; G. W., Kaatz; Fravolini, Arnaldo
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus.
2011 Brincat, JEAN PIERRE; Carosati, Emanuele; Sabatini, Stefano; Manfroni, Giuseppe; Fravolini, Arnaldo; Raygada, Jl; Patel, D; Kaatz, Gw; Cruciani, Gabriele
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Predictive models for hERG potassium channel blockers | 2005 | Cianchetta, Giovanni; Li, Y.; Kang, J.; Rampe, D.; Fravolini, Arnaldo; Cruciani, Gabriele; Vaz, R. J. | |
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation. | 2005 | Stevens, M.; Balzarini, J.; Tabarrini, Oriana; Andrei, G.; Snoeck, R.; Cecchetti, Violetta; Fravolini, Arnaldo; De Clercq, E.; Pannecouque, C. | |
A pharmacophore hypothesis for P-glycoprotein substrate recognition using GRIND-based 3D-QSAR. | 2005 | Cianchetta, Giovanni; Singleton, R. W.; Zhang, M.; Wildgoose, M.; Giesing, D.; Fravolini, Arnaldo; Cruciani, Gabriele; Vaz, R. J. | |
2-phenylquinolones as HIV-1 Tat/TAR interaction inhibitors | 2006 | Manfroni, Giuseppe; Tabarrini, Oriana; Sabatini, Stefano; Gatto, B.; Giaretta, G.; Palumbo, M.; Parolin, C.; Fravolini, Arnaldo; Cecchetti, V. | |
Synthesis and Activity of New Modified 1,4-Benzothiazine Derivatives as Inhibitors of the NorA Efflux Pump of Staphylococcus aureus | 2006 | Sabatini, Stefano; Giuliani, F.; Fusi, C.; Cecchetti, Violetta; Rossolini, G. M.; Fravolini, Arnaldo | |
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition. Abstr. P62 | 2006 | Gatto, B; Giaretta, G; Palumbo, M; Richter, S; Parolin, C; Palu, G; Tabarrini, Oriana; Fravolini, Arnaldo; Cecchetti, Violetta | |
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition | 2006 | Gatto, B.; Giaretta, G.; Palumbo, M.; Richter, S.; Parolin, C.; Palù, G.; Tabarrini, Oriana; Fravolini, Arnaldo; Cecchetti, Violetta | |
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents | 2006 | Tabarrini, Oriana; Manfroni, Giuseppe; Fravolini, Arnaldo; Cecchetti, Violetta; Sabatini, Stefano; De Clercq, E.; Rozenski, J.; Canard, B.; Dutartre, H.; Paeshuyse, J.; Neyts, J. | |
Derivati 2-fenilchinolonici come inibitori della pompa di efflusso NorA dello Staphylococcus aureus ciprofloxacin resistente | 2007 | Sabatini, Stefano; Pieroni, Marco; Manfroni, Giuseppe; Giuliani, F.; Rossolini, G. M.; Fravolini, Arnaldo | |
Novel In Vivo Model for the Study of Human Immunodeficiency Virus Type 1 Transcription Inhibitors: Evaluation of New 6-Desfluoroquinolone Derivatives | 2007 | Stevens, M.; Pollicita, M.; Pannecouque, C.; Verbeken, E.; Tabarrini, Oriana; Cecchetti, Violetta; Acquaro, S.; Perno, C. F.; Fravolini, Arnaldo; De Clercq, E.; Schols, D.; Balzarini, J. | |
Structure-activity relationship study on anti-HIV 6-desfluoroquinolones. | 2008 | Tabarrini, Oriana; Massari, Serena; Daelemans, D.; Stevens, M.; Manfroni, Giuseppe; Sabatini, Stefano; Balzarini, J.; Cecchetti, Violetta; Pannecouque, C.; Fravolini, Arnaldo | |
From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump. | 2008 | Sabatini, Stefano; Kaatz, G. W.; Rossolini, G. M.; Brandini, David; Fravolini, Arnaldo | |
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump | 2009 | Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta; Fravolini, Arnaldo | |
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump | 2009 | Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta; Fravolini, Arnaldo | |
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor. | 2009 | Manfroni, Giuseppe; Paeshuyse, J; Massari, Serena; Gatto, B; Zanoli, S; Maga, G; Tabarrini, Oriana; Cecchetti, Violetta; Fravolini, Arnaldo; Neyts, J. | |
Syhtesis and Biological Evaluation of 2-Phenylquinolones Targeted at Tat/TAR Recognition | 2009 | Manfroni, Giuseppe; Gatto, B; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta; Giaretta, G; Parolin, C; DEL VECCHIO, C; Calisti, A; Palumbo, M; Fravolini, Arnaldo | |
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction. | 2009 | Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta | |
From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps. | 2010 | Pieroni, Marco; M., Dimovska; Brincat, JEAN PIERRE; Sabatini, Stefano; Carosati, Emanuele; Massari, Serena; G. W., Kaatz; Fravolini, Arnaldo | |
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus. | 2011 | Brincat, JEAN PIERRE; Carosati, Emanuele; Sabatini, Stefano; Manfroni, Giuseppe; Fravolini, Arnaldo; Raygada, Jl; Patel, D; Kaatz, Gw; Cruciani, Gabriele |
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