Sfoglia per Autore
Binding Mode of 6ECDCA, a Potent Bile Acid Agonist of the Farnesoid X Receptor (FXR)
2003 Costantino, Gabriele; Macchiarulo, Antonio; Entrena Guadix, A.; Camaioni, Emidio; Pellicciari, Roberto
Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction
2003 Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto
Towards New Neuroprotective Agents: Design and Synthesis of Thieno[2,3-c]-isoquinolinon-5-one as a Potent PARP-1 Inhibitor.
2003 Pellicciari, Roberto; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Moroni, F.; Natalini, Benedetto
Novel Isoquinoline-Derived Inhibitors of Poly(ADP-Ribose) Polymerase-1: Pharmacological Characterization and Neuroprotective Effects in an in Vitro Model of Cerebral Ischemia
2003 Chiarugi, A; Meli, E; Calvani, M; Picca, R; Baronti, R; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Pellegrini Giampietro, De; Pellicciari, Roberto; Moroni, F.
Studies on the interaction between PARP’s catalytic site and inhibitors. Design and synthesis of new class of inhibitor derivatives
2004 Camaioni, Emidio; A., Leone; Costantino, Gabriele; D., Bellocchi; Macchiarulo, Antonio; Pellicciari, Roberto
Design, synthesis and S.A.R. of bile acid analogs as novel and selective FXR ligands
2004 Sadeghpour, B. M.; Gioiello, Antimo; Costantino, G.; Camaioni, Emidio; Rizzo, G.; Renga, B.; Fiorucci, Stefano; Pellicciari, Roberto
Life or Death Decisions. The case of Poly(ADP-Ribose)Polymerase (PARP) as therapeutic target for brain ischemia
2004 Pellicciari, Roberto; Camaioni, Emidio; Costantino, G.
Stereoselective Synthesis and Preliminary Evaluation of (+)- and (-)-3-methyl-5-carboxy-thien-2-yl-glycine (3-MATIDA): Identification of (+)-3-MATIDA as a Novel mGluR1 Competitive Antagonist
2004 Costantino, Gabriele; Marinozzi, Maura; Camaioni, Emidio; Natalini, Benedetto; Sarichelou, I.; Micheli, F.; Cavanni, P.; Faedo, S.; Noe, C.; Moroni, F.; Pellicciari, Roberto
Bile Acid Derivatives as Ligands of the Farnesoid X Receptor. Synthesis, Evaluation, and Structure Activity Relationship of a Series of Body and Side Chain Modified Analogs of Chenodeoxycholic Acid
2004 Pellicciari, Roberto; Costantino, Gabriele; Camaioni, Emidio; Sadeghpour, B. M.; Entrena Guadix, A.; Willson, T.; Fiorucci, Stefano; Clerici, C.; Gioiello, Antimo
Novel PARP Inhibitors: Synthesis and Molecular Modeling Studies
2005 Pellicciari, Roberto; Camaioni, Emidio; Moroni, F.; Chiarugi, A.; Costantino, Gabriele
Poly(ADP-ribose) Polymerase Inhibitors and Protection of Ischemia-Induced Brain Damage: Time Course and Dose-Response Studies in Rats with Middle Cerebral Artery Occlusion
2006 F., Moroni; A., Cozzi; A., Chiarugi; Camaioni, Emidio; Pellicciari, Roberto; D. E., Pellegrini Giampietro
Isocratic hydrophobicity index, phi0: a tool for studying the hydrophobic/hydrophilic balance of bile salts
2006 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; S., Natalini; Pellicciari, Roberto
RP-18-BASE-DEACTIVATED, una nuova fase stazionaria per l’analisi cromatografica degli acidi biliari
2006 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; S., Natalini; Pellicciari, Roberto
Design, Molecular Modeling Studies, Synthesis and Preliminary Evaluation of Novel PARP-1 Inhibitors on the Road of Antiischemic Agents
2006 Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; D., Bellocchi; A., Chiarugi; F., Moroni; A., Wood; Pellicciari, Roberto
3alpha-6alpha-Dihydroxy-7alpha-fluoro-5beta-cholanoate (UPF-680), physicochemical and physiological properties of a new fluorinated bile acid that prevents 17alpha-ethynyl-estradiol-induced cholestasis in rats..
2006 Clerici, C; Castellani, D; Asciutti, S; Pellicciari, R; Setchell, Kd; O'Connell, Nc; Sadeghpour, B; Camaioni, Emidio; Fiorucci, Stefano; Renga, Barbara; Nardi, E; Sabatino, G; Clementi, M; Giuliano, V; Baldoni, M; Orlandi, S; Mazzocchi, A; Morelli, A; Morelli, O.
Dominant Factors Affecting the Chromatographic Behaviour of Bile Acids
2006 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Natalini, S.; Pellicciari, Roberto
Inhibition of DPPIV by flavonoids as an alternative strategy for the treatment of type 2 diabetes
2006 Antonyan, A; Lupidi, G; Camaioni, Emidio; Mardanyan, S; Sharoyan, S.
Structural and Conformational Aspects of Molecular Recognition by Indoleamine-2,3-Dioxygenase (IDO), a Novel Target for Cancer Therapy
2007 Macchiarulo, Antonio; Nuti, Roberto; N. E., Campillo; Camaioni, Emidio; Pellicciari, Roberto
Bile acids: property-activity relationship and molecular modelling studies
2007 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto
Towards Selective PARP-2 Inhibitors: Design, Synthesis and Preliminary Evaluation of a Series of Isoquinolinone Derivatives
2007 Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; L., Formentini; F., Venturoni; D., Bellocchi; G., Eren; A., Chiarugi; F., Moroni; Pellicciari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Binding Mode of 6ECDCA, a Potent Bile Acid Agonist of the Farnesoid X Receptor (FXR) | 2003 | Costantino, Gabriele; Macchiarulo, Antonio; Entrena Guadix, A.; Camaioni, Emidio; Pellicciari, Roberto | |
Rat brain guanosine binding site. Biological studies and pseudo-Receptor construction | 2003 | Traversa, U.; Bombi, G.; Camaioni, Emidio; Macchiarulo, Antonio; Costantino, Gabriele; Palmieri, C.; Caciagli, F.; Pellicciari, Roberto | |
Towards New Neuroprotective Agents: Design and Synthesis of Thieno[2,3-c]-isoquinolinon-5-one as a Potent PARP-1 Inhibitor. | 2003 | Pellicciari, Roberto; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Moroni, F.; Natalini, Benedetto | |
Novel Isoquinoline-Derived Inhibitors of Poly(ADP-Ribose) Polymerase-1: Pharmacological Characterization and Neuroprotective Effects in an in Vitro Model of Cerebral Ischemia | 2003 | Chiarugi, A; Meli, E; Calvani, M; Picca, R; Baronti, R; Camaioni, Emidio; Costantino, Gabriele; Marinozzi, Maura; Pellegrini Giampietro, De; Pellicciari, Roberto; Moroni, F. | |
Studies on the interaction between PARP’s catalytic site and inhibitors. Design and synthesis of new class of inhibitor derivatives | 2004 | Camaioni, Emidio; A., Leone; Costantino, Gabriele; D., Bellocchi; Macchiarulo, Antonio; Pellicciari, Roberto | |
Design, synthesis and S.A.R. of bile acid analogs as novel and selective FXR ligands | 2004 | Sadeghpour, B. M.; Gioiello, Antimo; Costantino, G.; Camaioni, Emidio; Rizzo, G.; Renga, B.; Fiorucci, Stefano; Pellicciari, Roberto | |
Life or Death Decisions. The case of Poly(ADP-Ribose)Polymerase (PARP) as therapeutic target for brain ischemia | 2004 | Pellicciari, Roberto; Camaioni, Emidio; Costantino, G. | |
Stereoselective Synthesis and Preliminary Evaluation of (+)- and (-)-3-methyl-5-carboxy-thien-2-yl-glycine (3-MATIDA): Identification of (+)-3-MATIDA as a Novel mGluR1 Competitive Antagonist | 2004 | Costantino, Gabriele; Marinozzi, Maura; Camaioni, Emidio; Natalini, Benedetto; Sarichelou, I.; Micheli, F.; Cavanni, P.; Faedo, S.; Noe, C.; Moroni, F.; Pellicciari, Roberto | |
Bile Acid Derivatives as Ligands of the Farnesoid X Receptor. Synthesis, Evaluation, and Structure Activity Relationship of a Series of Body and Side Chain Modified Analogs of Chenodeoxycholic Acid | 2004 | Pellicciari, Roberto; Costantino, Gabriele; Camaioni, Emidio; Sadeghpour, B. M.; Entrena Guadix, A.; Willson, T.; Fiorucci, Stefano; Clerici, C.; Gioiello, Antimo | |
Novel PARP Inhibitors: Synthesis and Molecular Modeling Studies | 2005 | Pellicciari, Roberto; Camaioni, Emidio; Moroni, F.; Chiarugi, A.; Costantino, Gabriele | |
Poly(ADP-ribose) Polymerase Inhibitors and Protection of Ischemia-Induced Brain Damage: Time Course and Dose-Response Studies in Rats with Middle Cerebral Artery Occlusion | 2006 | F., Moroni; A., Cozzi; A., Chiarugi; Camaioni, Emidio; Pellicciari, Roberto; D. E., Pellegrini Giampietro | |
Isocratic hydrophobicity index, phi0: a tool for studying the hydrophobic/hydrophilic balance of bile salts | 2006 | Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; S., Natalini; Pellicciari, Roberto | |
RP-18-BASE-DEACTIVATED, una nuova fase stazionaria per l’analisi cromatografica degli acidi biliari | 2006 | Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; S., Natalini; Pellicciari, Roberto | |
Design, Molecular Modeling Studies, Synthesis and Preliminary Evaluation of Novel PARP-1 Inhibitors on the Road of Antiischemic Agents | 2006 | Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; D., Bellocchi; A., Chiarugi; F., Moroni; A., Wood; Pellicciari, Roberto | |
3alpha-6alpha-Dihydroxy-7alpha-fluoro-5beta-cholanoate (UPF-680), physicochemical and physiological properties of a new fluorinated bile acid that prevents 17alpha-ethynyl-estradiol-induced cholestasis in rats.. | 2006 | Clerici, C; Castellani, D; Asciutti, S; Pellicciari, R; Setchell, Kd; O'Connell, Nc; Sadeghpour, B; Camaioni, Emidio; Fiorucci, Stefano; Renga, Barbara; Nardi, E; Sabatino, G; Clementi, M; Giuliano, V; Baldoni, M; Orlandi, S; Mazzocchi, A; Morelli, A; Morelli, O. | |
Dominant Factors Affecting the Chromatographic Behaviour of Bile Acids | 2006 | Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Natalini, S.; Pellicciari, Roberto | |
Inhibition of DPPIV by flavonoids as an alternative strategy for the treatment of type 2 diabetes | 2006 | Antonyan, A; Lupidi, G; Camaioni, Emidio; Mardanyan, S; Sharoyan, S. | |
Structural and Conformational Aspects of Molecular Recognition by Indoleamine-2,3-Dioxygenase (IDO), a Novel Target for Cancer Therapy | 2007 | Macchiarulo, Antonio; Nuti, Roberto; N. E., Campillo; Camaioni, Emidio; Pellicciari, Roberto | |
Bile acids: property-activity relationship and molecular modelling studies | 2007 | Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto | |
Towards Selective PARP-2 Inhibitors: Design, Synthesis and Preliminary Evaluation of a Series of Isoquinolinone Derivatives | 2007 | Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; L., Formentini; F., Venturoni; D., Bellocchi; G., Eren; A., Chiarugi; F., Moroni; Pellicciari, Roberto |
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