Sfoglia per Autore
A new divergent synthesis of dafachronic acids from bile acids
2009 Sabbatini, P; Gioiello, Antimo; Khamidullina, A; Pellicciari, R.
Discovery of selective TGR5 modulators and their use in unraveling molecular features of bile acid recognition site
2009 Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; Thomas, C.; Rosatelli, E.; Schoonjans, K.; Adorini, L.; Pruzanski, M.; Auwerx, J.
Exploring the reactions of ethyl diazoacetate: new approaches to biologically active compounds
2009 Gioiello, Antimo; Venturoni, F.; Khamidullina, A.; Natalini, Benedetto; Pellicciari, Roberto
Side-chain modified bile acids: chromatographic evaluation of the epimer separation
2009 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto
BF3•Et2O-Induced Decomposition of Ethyl 2-Diazo-3-hydroxy-3,3-diarylpropanoates in Acetonitrile: A Novel Approach to 2,3-Diaryl β-Enamino Ester Derivatives
2009 Gioiello, Antimo; Venturoni, Francesco; Natalini, Benedetto; Pellicciari, Roberto
Side-chain Modified Bile Acids: Chromatographic Separation of 23-Methyl Epimers
2009 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; G., Carbone; M., Dawgul; Pellicciari, Roberto
Derived chromatographic indices as effective tools to study the self-aggregation process of bile acids
2009 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto
New one-pot synthesis of pyrazole-5-carboxylates by 1,3-dipole cycloadditions of ethyl diazoacetate with α-methylene carbonyl compunds
2009 Gioiello, Antimo; A., Khamidullina; M., CARMELA FULCO; F., Venturoni; S., Zlotsky; Pellicciari, Roberto
TGR5-mediated bile acid sensing controls glucose homeostasis.
2009 C., Thomas; Gioiello, Antimo; L., Noriega; A., Strehle; J., Oury; G., Rizzo; Macchiarulo, Antonio; H., Yamamoto; C., Mataki; M., Pruzanski; Pellicciari, Roberto; J., Auwerx; K., Schoonjans
Discovery of 6α-Ethyl-23(S)-methyl-cholic Acid (S-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity
2009 Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; C., Thomas; Rosatelli, Emiliano; Natalini, Benedetto; Sardella, Roccaldo; M., Pruzanski; A., Roda; E., Pastorini; K., Schoonjans; J., Auwerx
Design, synthesis, molecular modeling and biological activity of chenodeoxycholic acid carbamate derivatives as potent and selective FXR agonists
2010 Guerrieri, Elena; Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; Rizzo, Giovanni; Adorini, Luciano; Pellicciari, Roberto
On the route to biologically active heterocycles-containing compounds: Novel explorations with cyclic α-diazo-β-hydroxy ketones
2010 Venturoni, F; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, R.
Chromatographic evaluation of the 25-(R,S)-methyl-bishomo-hyodeoxycholic acid epimers
2010 Natalini, Benedetto; Ianni, F.; Sardella, Roccaldo; Gioiello, Antimo; Sabbatini, P.; Filipponi, P.; Pellicciari, Roberto
On the route of biologically active heterocycles-containing compouds: novel explorations with cyclic alpha-diazo-beta-hydroxy ketones
2010 Venturoni, F.; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, Roberto
High-throughput chromatographic determination of the bile acid critical micellar concentration
2010 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto
Chromatographic hydrophobicity index: a high-throughput tool to estimate the critical micellar concentration of bile acids
2010 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto
New potent and selective FXR agonists: design, synthesis and modeling of norcholanylamine derivatives
2010 Gioiello, Antimo; Macchiarulo, Antonio; Guerrieri, E.; Carotti, Andrea; Rizzo, G.; Adorini, L.; Pellicciari, Roberto
Targeting genomic (FXR) and nongenomic (TGR5) bile acids receptor pathways for metabolic disorders: discovery, S.A.R. and molecular modeling of potent and selective bile acids derivatives
2010 Pellicciari, R; Macchiarulo, Antonio; Gioiello, Antimo; Rosatelli, E; Thomas, C; Auwerx, J.
Lewis acid-promoted decomposition of a-diazo-b-hydroxy esters as a wealthy source of useful synthetic intermediates. Novel explorations with isatin
2010 Gioiello, Antimo; Venturoni, F.; Marinozzi, Maura; Pellicciari, Roberto
Thermal and catalytic reactions of ethyl diazopyruvate with [60]fullerene
2010 M., Roberti; Natalini, Benedetto; V., Andrisano; R., Seraglia; Gioiello, Antimo; Pellicciari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A new divergent synthesis of dafachronic acids from bile acids | 2009 | Sabbatini, P; Gioiello, Antimo; Khamidullina, A; Pellicciari, R. | |
Discovery of selective TGR5 modulators and their use in unraveling molecular features of bile acid recognition site | 2009 | Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; Thomas, C.; Rosatelli, E.; Schoonjans, K.; Adorini, L.; Pruzanski, M.; Auwerx, J. | |
Exploring the reactions of ethyl diazoacetate: new approaches to biologically active compounds | 2009 | Gioiello, Antimo; Venturoni, F.; Khamidullina, A.; Natalini, Benedetto; Pellicciari, Roberto | |
Side-chain modified bile acids: chromatographic evaluation of the epimer separation | 2009 | Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto | |
BF3•Et2O-Induced Decomposition of Ethyl 2-Diazo-3-hydroxy-3,3-diarylpropanoates in Acetonitrile: A Novel Approach to 2,3-Diaryl β-Enamino Ester Derivatives | 2009 | Gioiello, Antimo; Venturoni, Francesco; Natalini, Benedetto; Pellicciari, Roberto | |
Side-chain Modified Bile Acids: Chromatographic Separation of 23-Methyl Epimers | 2009 | Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; G., Carbone; M., Dawgul; Pellicciari, Roberto | |
Derived chromatographic indices as effective tools to study the self-aggregation process of bile acids | 2009 | Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto | |
New one-pot synthesis of pyrazole-5-carboxylates by 1,3-dipole cycloadditions of ethyl diazoacetate with α-methylene carbonyl compunds | 2009 | Gioiello, Antimo; A., Khamidullina; M., CARMELA FULCO; F., Venturoni; S., Zlotsky; Pellicciari, Roberto | |
TGR5-mediated bile acid sensing controls glucose homeostasis. | 2009 | C., Thomas; Gioiello, Antimo; L., Noriega; A., Strehle; J., Oury; G., Rizzo; Macchiarulo, Antonio; H., Yamamoto; C., Mataki; M., Pruzanski; Pellicciari, Roberto; J., Auwerx; K., Schoonjans | |
Discovery of 6α-Ethyl-23(S)-methyl-cholic Acid (S-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity | 2009 | Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; C., Thomas; Rosatelli, Emiliano; Natalini, Benedetto; Sardella, Roccaldo; M., Pruzanski; A., Roda; E., Pastorini; K., Schoonjans; J., Auwerx | |
Design, synthesis, molecular modeling and biological activity of chenodeoxycholic acid carbamate derivatives as potent and selective FXR agonists | 2010 | Guerrieri, Elena; Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; Rizzo, Giovanni; Adorini, Luciano; Pellicciari, Roberto | |
On the route to biologically active heterocycles-containing compounds: Novel explorations with cyclic α-diazo-β-hydroxy ketones | 2010 | Venturoni, F; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, R. | |
Chromatographic evaluation of the 25-(R,S)-methyl-bishomo-hyodeoxycholic acid epimers | 2010 | Natalini, Benedetto; Ianni, F.; Sardella, Roccaldo; Gioiello, Antimo; Sabbatini, P.; Filipponi, P.; Pellicciari, Roberto | |
On the route of biologically active heterocycles-containing compouds: novel explorations with cyclic alpha-diazo-beta-hydroxy ketones | 2010 | Venturoni, F.; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, Roberto | |
High-throughput chromatographic determination of the bile acid critical micellar concentration | 2010 | Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto | |
Chromatographic hydrophobicity index: a high-throughput tool to estimate the critical micellar concentration of bile acids | 2010 | Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto | |
New potent and selective FXR agonists: design, synthesis and modeling of norcholanylamine derivatives | 2010 | Gioiello, Antimo; Macchiarulo, Antonio; Guerrieri, E.; Carotti, Andrea; Rizzo, G.; Adorini, L.; Pellicciari, Roberto | |
Targeting genomic (FXR) and nongenomic (TGR5) bile acids receptor pathways for metabolic disorders: discovery, S.A.R. and molecular modeling of potent and selective bile acids derivatives | 2010 | Pellicciari, R; Macchiarulo, Antonio; Gioiello, Antimo; Rosatelli, E; Thomas, C; Auwerx, J. | |
Lewis acid-promoted decomposition of a-diazo-b-hydroxy esters as a wealthy source of useful synthetic intermediates. Novel explorations with isatin | 2010 | Gioiello, Antimo; Venturoni, F.; Marinozzi, Maura; Pellicciari, Roberto | |
Thermal and catalytic reactions of ethyl diazopyruvate with [60]fullerene | 2010 | M., Roberti; Natalini, Benedetto; V., Andrisano; R., Seraglia; Gioiello, Antimo; Pellicciari, Roberto |
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