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Mostrati risultati da 21 a 40 di 180
Titolo Data di pubblicazione Autore(i) File
A new divergent synthesis of dafachronic acids from bile acids 2009 Sabbatini, P; Gioiello, Antimo; Khamidullina, A; Pellicciari, R.
Discovery of selective TGR5 modulators and their use in unraveling molecular features of bile acid recognition site 2009 Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; Thomas, C.; Rosatelli, E.; Schoonjans, K.; Adorini, L.; Pruzanski, M.; Auwerx, J.
Exploring the reactions of ethyl diazoacetate: new approaches to biologically active compounds 2009 Gioiello, Antimo; Venturoni, F.; Khamidullina, A.; Natalini, Benedetto; Pellicciari, Roberto
Side-chain modified bile acids: chromatographic evaluation of the epimer separation 2009 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto
BF3•Et2O-Induced Decomposition of Ethyl 2-Diazo-3-hydroxy-3,3-diarylpropanoates in Acetonitrile: A Novel Approach to 2,3-Diaryl β-Enamino Ester Derivatives 2009 Gioiello, Antimo; Venturoni, Francesco; Natalini, Benedetto; Pellicciari, Roberto
Side-chain Modified Bile Acids: Chromatographic Separation of 23-Methyl Epimers 2009 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; G., Carbone; M., Dawgul; Pellicciari, Roberto
Derived chromatographic indices as effective tools to study the self-aggregation process of bile acids 2009 Natalini, Benedetto; Sardella, Roccaldo; Camaioni, Emidio; Macchiarulo, Antonio; Gioiello, Antimo; Carbone, G.; Pellicciari, Roberto
New one-pot synthesis of pyrazole-5-carboxylates by 1,3-dipole cycloadditions of ethyl diazoacetate with α-methylene carbonyl compunds 2009 Gioiello, Antimo; A., Khamidullina; M., CARMELA FULCO; F., Venturoni; S., Zlotsky; Pellicciari, Roberto
TGR5-mediated bile acid sensing controls glucose homeostasis. 2009 C., Thomas; Gioiello, Antimo; L., Noriega; A., Strehle; J., Oury; G., Rizzo; Macchiarulo, Antonio; H., Yamamoto; C., Mataki; M., Pruzanski; Pellicciari, Roberto; J., Auwerx; K., Schoonjans
Discovery of 6α-Ethyl-23(S)-methyl-cholic Acid (S-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity 2009 Pellicciari, Roberto; Gioiello, Antimo; Macchiarulo, Antonio; C., Thomas; Rosatelli, Emiliano; Natalini, Benedetto; Sardella, Roccaldo; M., Pruzanski; A., Roda; E., Pastorini; K., Schoonjans; J., Auwerx
Design, synthesis, molecular modeling and biological activity of chenodeoxycholic acid carbamate derivatives as potent and selective FXR agonists 2010 Guerrieri, Elena; Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; Rizzo, Giovanni; Adorini, Luciano; Pellicciari, Roberto
On the route to biologically active heterocycles-containing compounds: Novel explorations with cyclic α-diazo-β-hydroxy ketones 2010 Venturoni, F; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, R.
Chromatographic evaluation of the 25-(R,S)-methyl-bishomo-hyodeoxycholic acid epimers 2010 Natalini, Benedetto; Ianni, F.; Sardella, Roccaldo; Gioiello, Antimo; Sabbatini, P.; Filipponi, P.; Pellicciari, Roberto
On the route of biologically active heterocycles-containing compouds: novel explorations with cyclic alpha-diazo-beta-hydroxy ketones 2010 Venturoni, F.; Gioiello, Antimo; Marinozzi, Maura; Pellicciari, Roberto
High-throughput chromatographic determination of the bile acid critical micellar concentration 2010 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto
Chromatographic hydrophobicity index: a high-throughput tool to estimate the critical micellar concentration of bile acids 2010 Natalini, Benedetto; Sardella, Roccaldo; Gioiello, Antimo; E., Rosatelli; Nuti, Roberto; Camaioni, Emidio; Macchiarulo, Antonio; Pellicciari, Roberto
New potent and selective FXR agonists: design, synthesis and modeling of norcholanylamine derivatives 2010 Gioiello, Antimo; Macchiarulo, Antonio; Guerrieri, E.; Carotti, Andrea; Rizzo, G.; Adorini, L.; Pellicciari, Roberto
Targeting genomic (FXR) and nongenomic (TGR5) bile acids receptor pathways for metabolic disorders: discovery, S.A.R. and molecular modeling of potent and selective bile acids derivatives 2010 Pellicciari, R; Macchiarulo, Antonio; Gioiello, Antimo; Rosatelli, E; Thomas, C; Auwerx, J.
Lewis acid-promoted decomposition of a-diazo-b-hydroxy esters as a wealthy source of useful synthetic intermediates. Novel explorations with isatin 2010 Gioiello, Antimo; Venturoni, F.; Marinozzi, Maura; Pellicciari, Roberto
Thermal and catalytic reactions of ethyl diazopyruvate with [60]fullerene 2010 M., Roberti; Natalini, Benedetto; V., Andrisano; R., Seraglia; Gioiello, Antimo; Pellicciari, Roberto
Mostrati risultati da 21 a 40 di 180
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