Sfoglia per Autore
Triazolopyrimidine nuclei: privileged scaffolds for developing antiviral agents with a proper pharmacokinetic profile.
2021 Felicetti, T; Pismataro, Mc; Cecchetti, V; Tabarrini, O; Massari, S
Microbial efflux pump inhibitors: A journey around quinoline and indole derivatives
2021 Cernicchi, G.; Felicetti, T.; Sabatini, S.
Sustainable, three-component, one-pot procedure to obtain active anti-flavivirus agents
2021 Felicetti, T.; Burali, M. S.; Gwee, C. P.; Ki Chan, K. W.; Alonso, S.; Massari, S.; Sabatini, S.; Tabarrini, O.; Barreca, M. L.; Cecchetti, V.; Vasudevan, S. G.; Manfroni, G.
1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors
2021 Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S.
Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation
2021 Pica, M.; Messere, N.; Felicetti, T.; Sabatini, S.; Pietrella, D.; Nocchetti, M.
Synthesis and Characterization of 1,2,4-Triazolo[1,5-a]pyrimidine-2-carboxamide-based Compounds Targeting the PA-PB1 Interface of Influenza A Virus Polymerase.
2021 Massari, S.; Bertagnin, C.; Pismataro, M. C.; Donnadio, A.; Nannetti, G.; Felicetti, T.; Di Bona, S.; Nizi, M. G.; Tensi, L.; Manfroni, G.; Loza, M. I.; Sabatini, S.; Cecchetti, V.; Brea, J.; Goracci, L.; Loregian, A.; Tabarrini, O.
Targeting miRNA dysregulation with small molecules: The case of enoxacin
2021 Felicetti, T.; Manfroni, G.
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
2021 Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano
Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi
2021 Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio
Building up efflux-mediated antimicrobial resistance in Staphylococcus pseudintermedius
2022 Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio
Virucidal Activity of the Pyridobenzothiazolone Derivative HeE1-17Y against Enveloped RNA Viruses
2022 Milan Bonotto, Rafaela; Bonì, Francesco; Milani, Mario; Chaves-Sanjuan, Antonio; Franze, Silvia; Selmin, Francesca; Felicetti, Tommaso; Bolognesi, Martino; Konstantinidou, Soultana; Poggianella, Monica; Márquez, Chantal L; Dattola, Federica; Zoppè, Monica; Manfroni, Giuseppe; Mastrangelo, Eloise; Marcello, Alessandro
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity
2022 Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana
Drug efflux transporters in Staphylococcus pseudintermedius: in silico prediction and characterization of resistance
2022 Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio
New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains
2022 Felicetti, Tommaso; Cedraro, Nicholas; Astolfi, Andrea; Cernicchi, Giada; Mangiaterra, Gianmarco; Vaiasicca, Salvatore; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Biavasco, Francesca; Cecchetti, Violetta; Vignaroli, Carla; Sabatini, Stefano
An overview on small molecules acting as broad-spectrum agents for yellow fever infection
2022 Desantis, J.; Felicetti, T.; Cannalire, R.
EVALUATION OF DRUG EFFLUX ACTIVITY IN ANTIMICROBIAL RESISTANT STAPHYLOCOCCUS PSEUDINTERMEDIUS CLINICAL ISOLATES
2023 Rampacci, Elisa; Felicetti, Tommaso; Birettoni, Francesco; Arcelli, Rolando; Zelli, Riccardo; Sabatini, Stefano; Passamonti, Fabrizio
Functionalized sulfonyl anthranilic acid derivatives inhibit replication of all the four dengue serotypes
2023 Felicetti, Tommaso; Gwee, Chin Piaw; Burali, Maria Sole; Chan, Kitti Wing Ki; Alonso, Sylvie; Pismataro, Maria Chiara; Sabatini, Stefano; Barreca, Maria Letizia; Cecchetti, Violetta; Vasudevan, Subhash G; Manfroni, Giuseppe
Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations
2023 Palazzotti, Deborah; Felicetti, Tommaso; Sabatini, Stefano; Moro, Stefano; Barreca, Maria Letizia; Sturlese, Mattia; Astolfi, Andrea
Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors
2023 Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio
Switching the three-component Biginelli-like reaction conditions for the regioselective synthesis of new 2-amino[1,2,4]triazolo[1,5-a]pyrimidines
2024 Pacetti, Martina; Pismataro, Maria Chiara; Felicetti, Tommaso; Giammarino, Federica; Bonomini, Anna; Tiecco, Matteo; Bertagnin, Chiara; Barreca, Maria Letizia; Germani, Raimondo; Cecchetti, Violetta; Vicenti, Ilaria; Tabarrini, Oriana; Zazzi, Maurizio; Loregian, Arianna; Massari, Serena
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Triazolopyrimidine nuclei: privileged scaffolds for developing antiviral agents with a proper pharmacokinetic profile. | 2021 | Felicetti, T; Pismataro, Mc; Cecchetti, V; Tabarrini, O; Massari, S | |
| Microbial efflux pump inhibitors: A journey around quinoline and indole derivatives | 2021 | Cernicchi, G.; Felicetti, T.; Sabatini, S. | |
| Sustainable, three-component, one-pot procedure to obtain active anti-flavivirus agents | 2021 | Felicetti, T.; Burali, M. S.; Gwee, C. P.; Ki Chan, K. W.; Alonso, S.; Massari, S.; Sabatini, S.; Tabarrini, O.; Barreca, M. L.; Cecchetti, V.; Vasudevan, S. G.; Manfroni, G. | |
| 1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors | 2021 | Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S. | |
| Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation | 2021 | Pica, M.; Messere, N.; Felicetti, T.; Sabatini, S.; Pietrella, D.; Nocchetti, M. | |
| Synthesis and Characterization of 1,2,4-Triazolo[1,5-a]pyrimidine-2-carboxamide-based Compounds Targeting the PA-PB1 Interface of Influenza A Virus Polymerase. | 2021 | Massari, S.; Bertagnin, C.; Pismataro, M. C.; Donnadio, A.; Nannetti, G.; Felicetti, T.; Di Bona, S.; Nizi, M. G.; Tensi, L.; Manfroni, G.; Loza, M. I.; Sabatini, S.; Cecchetti, V.; Brea, J.; Goracci, L.; Loregian, A.; Tabarrini, O. | |
| Targeting miRNA dysregulation with small molecules: The case of enoxacin | 2021 | Felicetti, T.; Manfroni, G. | |
| From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | 2021 | Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano | |
| Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi | 2021 | Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio | |
| Building up efflux-mediated antimicrobial resistance in Staphylococcus pseudintermedius | 2022 | Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio | |
| Virucidal Activity of the Pyridobenzothiazolone Derivative HeE1-17Y against Enveloped RNA Viruses | 2022 | Milan Bonotto, Rafaela; Bonì, Francesco; Milani, Mario; Chaves-Sanjuan, Antonio; Franze, Silvia; Selmin, Francesca; Felicetti, Tommaso; Bolognesi, Martino; Konstantinidou, Soultana; Poggianella, Monica; Márquez, Chantal L; Dattola, Federica; Zoppè, Monica; Manfroni, Giuseppe; Mastrangelo, Eloise; Marcello, Alessandro | |
| Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity | 2022 | Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana | |
| Drug efflux transporters in Staphylococcus pseudintermedius: in silico prediction and characterization of resistance | 2022 | Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio | |
| New C-6 functionalized quinoline NorA inhibitors strongly synergize with ciprofloxacin against planktonic and biofilm growing resistant Staphylococcus aureus strains | 2022 | Felicetti, Tommaso; Cedraro, Nicholas; Astolfi, Andrea; Cernicchi, Giada; Mangiaterra, Gianmarco; Vaiasicca, Salvatore; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Biavasco, Francesca; Cecchetti, Violetta; Vignaroli, Carla; Sabatini, Stefano | |
| An overview on small molecules acting as broad-spectrum agents for yellow fever infection | 2022 | Desantis, J.; Felicetti, T.; Cannalire, R. | |
| EVALUATION OF DRUG EFFLUX ACTIVITY IN ANTIMICROBIAL RESISTANT STAPHYLOCOCCUS PSEUDINTERMEDIUS CLINICAL ISOLATES | 2023 | Rampacci, Elisa; Felicetti, Tommaso; Birettoni, Francesco; Arcelli, Rolando; Zelli, Riccardo; Sabatini, Stefano; Passamonti, Fabrizio | |
| Functionalized sulfonyl anthranilic acid derivatives inhibit replication of all the four dengue serotypes | 2023 | Felicetti, Tommaso; Gwee, Chin Piaw; Burali, Maria Sole; Chan, Kitti Wing Ki; Alonso, Sylvie; Pismataro, Maria Chiara; Sabatini, Stefano; Barreca, Maria Letizia; Cecchetti, Violetta; Vasudevan, Subhash G; Manfroni, Giuseppe | |
| Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations | 2023 | Palazzotti, Deborah; Felicetti, Tommaso; Sabatini, Stefano; Moro, Stefano; Barreca, Maria Letizia; Sturlese, Mattia; Astolfi, Andrea | |
| Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors | 2023 | Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio | |
| Switching the three-component Biginelli-like reaction conditions for the regioselective synthesis of new 2-amino[1,2,4]triazolo[1,5-a]pyrimidines | 2024 | Pacetti, Martina; Pismataro, Maria Chiara; Felicetti, Tommaso; Giammarino, Federica; Bonomini, Anna; Tiecco, Matteo; Bertagnin, Chiara; Barreca, Maria Letizia; Germani, Raimondo; Cecchetti, Violetta; Vicenti, Ilaria; Tabarrini, Oriana; Zazzi, Maurizio; Loregian, Arianna; Massari, Serena |
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