MANFRONI, GIUSEPPE

MANFRONI, GIUSEPPE  

DIPARTIMENTO DI SCIENZE FARMACEUTICHE  

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1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity 2020 Desantis, J.; Massari, S.; Corona, A.; Astolfi, A.; Sabatini, S.; Manfroni, G.; Palazzotti, D.; Cecchetti, V.; Pannecouque, C.; Tramontano, E.; Tabarrini, O.
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions 2013 Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities 2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction 2018 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
2-phenylquinolones as HIV-1 Tat/TAR interaction inhibitors 2006 Manfroni, Giuseppe; Tabarrini, Oriana; Sabatini, Stefano; Gatto, B.; Giaretta, G.; Palumbo, M.; Parolin, C.; Fravolini, Arnaldo; Cecchetti, V.
6-Aminoquinolones targeting HCV NS5B polymerase. 2012 Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta
6-Desfluoroquinolones as promising HIV transcription inhibitors 2007 Tabarrini, Oriana; Cecchetti, Violetta; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Stevens, M.; Daelemans, D.; Pannecouque, C.
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction 2015 Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana
A cellular screening platform, stably expressing DENV2 NS5, defines a novel anti-DENV mechanism of action of Apigenin based on STAT2 activation 2023 Acchioni, Chiara; Acchioni, Marta; Mancini, Flavia; Amendola, Antonello; Marsili, Giulia; Tirelli, Valentina; Gwee, Chin Piaw; Chan, Kitti Wing-Ki; Sandini, Silvia; Bisbocci, Monica; Mysara, Mohamed; Elhefnawi, Mahmoud; Sanchez, Massimo; Venturi, Giulietta; Barreca, Maria Letizia; Manfroni, Giuseppe; Bresciani, Alberto; Vasudevan, Subhash G; Sgarbanti, Marco
A Comprehensive Structural Overview of p38 Mitogen-Activated Protein Kinase in Complex with ATP-Site and Non-ATP-Site Binders 2018 Astolfi, Andrea; Manfroni, Giuseppe; Cecchetti, Violetta; Barreca, Maria Letizia
A Comprehensive Structural Overview of p38α MAPK in Complex with Type I Inhibitors 2015 Astolfi, Andrea; Iraci, Nunzio; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Cecchetti, Violetta
A Journey around the Medicinal Chemistry of Hepatitis C Virus Inhibitors Targeting NS4B: From Target to Preclinical Drug Candidates 2016 Cannalire, Rolando; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Cecchetti, Violetta
A New Derivative with Ultra-Potent Anti-HIV Activity 2008 Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta; Daelemans, D; Pannecouque, C.
A New Promising Class of pyrazolobenzothiazine inhibitors of S. aureus NorA Efflux Pump 2012 Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Carosati, Emanuele; Cecchetti, Violetta
A new quinolone derivative with ultra-potent anti-HIV activity. 2008 Massari, Serena; Tabarrini, O; Manfroni, Giuseppe; V., Cecchetti; D., Daelemans; C., Pannecouque
Accounting for target flexibility and water molecules by docking to ensembles of target structures: The HCV NS5B Palm Site I inhibitors case study. 2014 Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Gaetani, Rosy; Guercini, Chiara; Sabatini, Stefano; Tabarrini, Oriana; Cecchetti, Violetta
Advantageous Use of Ionic Liquids for the Synthesis of Pharmaceutically Relevant Quinolones 2018 Cannalire, Rolando; Tiecco, Matteo; Cecchetti, Violetta; Germani, Raimondo; Manfroni, Giuseppe
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development 2011 Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Cecchetti, Violetta
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors 2020 Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O.
Bicyclic octahydrocyclohepta[b]pyrrol-4(1H)one derivatives as novel selective anti-hepatitis C virus agents 2016 Kaushik Basu, Neerja; Ratmanova, Nina K.; Manvar, Dinesh; Belov, Dmitry S.; Cevik, Ozge; Basu, Amartya; Yerukhimovich, Mark M.; Lukyanenko, Evgeny R.; Andreev, Ivan A.; Belov, Grigory M.; Manfroni, Giuseppe; Cecchetti, Violetta; Frick, David N.; Kurkin, Alexander V.; Altieri, Andrea; Barreca, MARIA LETIZIA