SANCINETO, LUCA
SANCINETO, LUCA
DIPARTIMENTO DI SCIENZE FARMACEUTICHE
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities
2013-01-01 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors
2018-01-01 Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari
A domino approach to pyrazino- indoles and pyrroles using vinyl selenones
2018-01-01 Palomba, M; Sancineto, L.; Marini, F.; Santi, C.; Bagnoli, L.
A mild and efficient method for the synthesis of a new optically active diallyl selenide and its catalytic activity in the allylic chlorination of natural terpenes
2016-01-01 Boualy, Brahim; El Houssame, Soufiane; Sancineto, Luca; Santi, Claudio; Ait Ali, Mustapha; Stoeckli Evans, Helen; El Firdoussi, Larbi
A new vinyl selenone-based domino approach to spirocyclopropyl oxindoles endowed with anti-HIV RT activity
2016-01-01 Palomba, Martina; Rossi, L.; Sancineto, Luca; Tramontano, E.; Corona, A.; Bagnoli, Luana; Santi, Claudio; Pannecouque, C.; Tabarrini, Oriana; Marini, Francesca
A Recyclable Biphasic System for Stereoselective and Easily Handled Hydrochalcogenations
2014-01-01 Tidei, Caterina; Sancineto, Luca; Bagnoli, Luana; Battistelli, Benedetta; Marini, Francesca; Santi, Claudio
A Selenone Mediated Domino Strategy for the Construction of Variously Functionalized Spirocyclopropyl Oxindoles
2015-01-01 Palomba, Martina; Rossi, L.; Sancineto, Luca; Bagnoli, Luana; Santi, Claudio; Marini, Francesca
Advances in Electrophilic Organochalcogen Reagents
2016-01-01 Sancineto, Luca; Palomba, Martina; Bagnoli, Luana; Marini, Francesca; Santi, Claudio
An enantiopure diselenide based on a chiral bicyclic backbone-synthesis and configuration assignment
2017-01-01 Kamińska, Karolina; Wojaczyńska, Elżbieta; Santi, Claudio; Sancineto, Luca; Francesca Pensa, Marianna; Kochel, Andrzej; Wieczorek, Robert; Wojaczyński, Jacek; Slupski, Gauthier
An Update on “Selenium Containing Compounds from Poison to Drug Candidates: A Review on the GPx-like Activity”
2016-01-01 Pacuła, Agata J.; Mangiavacchi, Francesca; Sancineto, Luca; Eder, J. Lenardão; Ścianowski, Jacek; Santi, Claudio
Atom Efficient Preparation of Zinc Selenates for the Synthesis of Selenol Esters under "On Water" Conditions
2017-01-01 Sancineto, Luca; Pinto Vargas, Jaqueline; Monti, Bonifacio; Arca, Massimiliano; Lippolis, Vito; Perin, Gelson; Lenardao, Eder Joao; Santi, Claudio
CHALCOGENS IN NEW CATALYTIC REACTIONS
2014-01-01 Santi, Claudio; Bagnoli, Luana; Marini, Francesca; Tidei, Caterina; Sancineto, L.
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013-01-01 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013-01-01 Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Continuous Bioinspired Oxidation of Sulfides
2020-01-01 Mangiavacchi, F.; Crociani, L.; Sancineto, L.; Marini, F.; Santi, C.
Continuous flow synthesis of 2,2′-diselenobis(benzoic acid) and derivatives
2020-01-01 Begini, F.; Krasowska, D.; Jasiak, A.; Drabowicz, J.; Santi, C.; Sancineto, L.
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors
2013-01-01 Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana
CYCLOHEPTATHIOPHENE-3-CARBOXAMIDE DERIVATIVES AS INFLUENZA A VIRUS POLYMERASE INHIBITORS
2013-01-01 Massari, Serena; Giulio, Nannetti; Giulia, Muratore; Jenny, Desantis; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Beatrice, Mercorelli; Giorgio, Palù; Arianna, Loregian; Tabarrini, Oriana
Design and Synthesis of DiselenoBisBenzamides (DISeBAs) as Nucleocapsid Protein 7 (NCp7) Inhibitors with anti-HIV Activity
2015-01-01 Sancineto, Luca; Mariotti, Alice; Bagnoli, Luana; Marini, Francesca; Desantis, Jenny; Iraci, Nunzio; Santi, Claudio; Pannecouque, Christophe; Tabarrini, Oriana
Design and synthesis of new biologically active diselenides
2013-01-01 Sancineto, Luca; A., Mariotti; Tidei, Caterina; Bagnoli, Luana; Marini, Francesca; Tabarrini, Oriana; Santi, Claudio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities | 1-gen-2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors | 1-gen-2018 | Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari | |
A domino approach to pyrazino- indoles and pyrroles using vinyl selenones | 1-gen-2018 | Palomba, M; Sancineto, L.; Marini, F.; Santi, C.; Bagnoli, L. | |
A mild and efficient method for the synthesis of a new optically active diallyl selenide and its catalytic activity in the allylic chlorination of natural terpenes | 1-gen-2016 | Boualy, Brahim; El Houssame, Soufiane; Sancineto, Luca; Santi, Claudio; Ait Ali, Mustapha; Stoeckli Evans, Helen; El Firdoussi, Larbi | |
A new vinyl selenone-based domino approach to spirocyclopropyl oxindoles endowed with anti-HIV RT activity | 1-gen-2016 | Palomba, Martina; Rossi, L.; Sancineto, Luca; Tramontano, E.; Corona, A.; Bagnoli, Luana; Santi, Claudio; Pannecouque, C.; Tabarrini, Oriana; Marini, Francesca | |
A Recyclable Biphasic System for Stereoselective and Easily Handled Hydrochalcogenations | 1-gen-2014 | Tidei, Caterina; Sancineto, Luca; Bagnoli, Luana; Battistelli, Benedetta; Marini, Francesca; Santi, Claudio | |
A Selenone Mediated Domino Strategy for the Construction of Variously Functionalized Spirocyclopropyl Oxindoles | 1-gen-2015 | Palomba, Martina; Rossi, L.; Sancineto, Luca; Bagnoli, Luana; Santi, Claudio; Marini, Francesca | |
Advances in Electrophilic Organochalcogen Reagents | 1-gen-2016 | Sancineto, Luca; Palomba, Martina; Bagnoli, Luana; Marini, Francesca; Santi, Claudio | |
An enantiopure diselenide based on a chiral bicyclic backbone-synthesis and configuration assignment | 1-gen-2017 | Kamińska, Karolina; Wojaczyńska, Elżbieta; Santi, Claudio; Sancineto, Luca; Francesca Pensa, Marianna; Kochel, Andrzej; Wieczorek, Robert; Wojaczyński, Jacek; Slupski, Gauthier | |
An Update on “Selenium Containing Compounds from Poison to Drug Candidates: A Review on the GPx-like Activity” | 1-gen-2016 | Pacuła, Agata J.; Mangiavacchi, Francesca; Sancineto, Luca; Eder, J. Lenardão; Ścianowski, Jacek; Santi, Claudio | |
Atom Efficient Preparation of Zinc Selenates for the Synthesis of Selenol Esters under "On Water" Conditions | 1-gen-2017 | Sancineto, Luca; Pinto Vargas, Jaqueline; Monti, Bonifacio; Arca, Massimiliano; Lippolis, Vito; Perin, Gelson; Lenardao, Eder Joao; Santi, Claudio | |
CHALCOGENS IN NEW CATALYTIC REACTIONS | 1-gen-2014 | Santi, Claudio; Bagnoli, Luana; Marini, Francesca; Tidei, Caterina; Sancineto, L. | |
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 1-gen-2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana | |
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 1-gen-2013 | Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Continuous Bioinspired Oxidation of Sulfides | 1-gen-2020 | Mangiavacchi, F.; Crociani, L.; Sancineto, L.; Marini, F.; Santi, C. | |
Continuous flow synthesis of 2,2′-diselenobis(benzoic acid) and derivatives | 1-gen-2020 | Begini, F.; Krasowska, D.; Jasiak, A.; Drabowicz, J.; Santi, C.; Sancineto, L. | |
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors | 1-gen-2013 | Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana | |
CYCLOHEPTATHIOPHENE-3-CARBOXAMIDE DERIVATIVES AS INFLUENZA A VIRUS POLYMERASE INHIBITORS | 1-gen-2013 | Massari, Serena; Giulio, Nannetti; Giulia, Muratore; Jenny, Desantis; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Beatrice, Mercorelli; Giorgio, Palù; Arianna, Loregian; Tabarrini, Oriana | |
Design and Synthesis of DiselenoBisBenzamides (DISeBAs) as Nucleocapsid Protein 7 (NCp7) Inhibitors with anti-HIV Activity | 1-gen-2015 | Sancineto, Luca; Mariotti, Alice; Bagnoli, Luana; Marini, Francesca; Desantis, Jenny; Iraci, Nunzio; Santi, Claudio; Pannecouque, Christophe; Tabarrini, Oriana | |
Design and synthesis of new biologically active diselenides | 1-gen-2013 | Sancineto, Luca; A., Mariotti; Tidei, Caterina; Bagnoli, Luana; Marini, Francesca; Tabarrini, Oriana; Santi, Claudio |