COSTANTINO, Gabriele

COSTANTINO, Gabriele  

DIPARTIMENTO DI SCIENZE FARMACEUTICHE  

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Titolo Data di pubblicazione Autore(i) File
"*-Diazocarbonyl Chemistry - Target Driven Applications" 1998 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Mattoli, L.; Natalini, Benedetto
(2R,1’S,2’R,3’S)-2-(2’-Carboxy-3’-phenylcyclopropyl)glycine (PCCG-13), the First Potent and Selective Competitive Antagonist of Phospholipase D-Coupled Metabotropic Glutamate Receptors: Asymmetric Synthesis and Preliminary Biological Properties 2001 Pellicciari, Roberto; Marinozzi, Maura; Costantino, Gabriele; Natalini, Benedetto; Moroni, F.; Pellegrini Giampietro, D.
1,4 Benzothiazine and 1,4 benzoxazine imidazole derivatives with antifungal activity: a docking study 2002 Macchiarulo, Antonio; Costantino, Gabriele; Fringuelli, D.; Vecchiarelli, Anna; Schiaffella, Fausto; Fringuelli, Renata
1-AMINOINDAN-1,5-DICARBOXYLIC ACID - A NOVEL ANTAGONIST AT PHOSPHOLIPASE C-LINKED METABOTROPIC GLUTAMATE RECEPTORS 1995 Pellicciari, Roberto; R., Luneia; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; P., Jakobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen
Asymmetric synthesis of (2R, 1’S, 2’R, 3’S)-2-(2’- Carboxy-3’-phenylcyclopropyl)glicine (PCCG 13), the first selective antagonist of metabotropic glutamate receptors coupled phospholipase D 1998 Marinozzi, Maura; Costantino, Gabriele; D. E., Pellegrini Giampietro; Pellicciari, Roberto
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-Phenylcarboxycyclopropylglycine (PCCG-4): a Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors 1996 Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; P., Tijskens; C., Thomsen; Pellicciari, Roberto
Autocorrelation as a tool for a congruent description of molecu¬les in 3D-QSAR studies 1993 Clementi, Sergio; Cruciani, Gabriele; D., Riganelli; Valigi, Roberta; Costantino, Gabriele; Baroni, Massimo; S., Wold
Bile Acid Derivatives as Ligands of the Farnesoid X Receptor. Synthesis, Evaluation, and Structure Activity Relationship of a Series of Body and Side Chain Modified Analogs of Chenodeoxycholic Acid 2004 Pellicciari, Roberto; Costantino, Gabriele; Camaioni, Emidio; Sadeghpour, B. M.; Entrena Guadix, A.; Willson, T.; Fiorucci, Stefano; Clerici, C.; Gioiello, Antimo
Binding Mode of 6ECDCA, a Potent Bile Acid Agonist of the Farnesoid X Receptor (FXR) 2003 Costantino, Gabriele; Macchiarulo, Antonio; Entrena Guadix, A.; Camaioni, Emidio; Pellicciari, Roberto
Binding modes of noncompetitive AMPA Antagonists: A computational approach 2003 De Luca, L.; Macchiarulo, Antonio; Costantino, Gabriele; Barreca, MARIA LETIZIA; Gitto, R.; Chimirri, A.; Pellicciari, Roberto
Bulky 1,4-benzoxazine derivatives with antifungal activity 2009 Fringuelli, Renata; Giacche', Nicola; Milanese, Lara; Cenci, Elio; Macchiarulo, Antonio; Vecchiarelli, Anna; Costantino, Gabriele; Schiaffella, Fausto
Chromatographic separation and evaluation of the lipophilicity by reversed-phase high-performance liquid chromatography of fullerene-C60 derivatives 2001 Natalini, Benedetto; Marinozzi, Maura; Costantino, Gabriele; Pellicciari, Roberto; Capodiferro, V.; Mattoli, L.
Conformational requirements for interaction of L-glutamate with the metabotropic EAA receptor 1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase 1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi
Design and synthesis of 4H-thieno[2,3-c]isoquinolin-5-one derivatives as potent PARP-1 inhibitors, on route of new antiischemic agents 2003 Camaioni, Emidio; Costantino, Gabriele; Macchiarulo, Antonio; Marinozzi, Maura; F., Moroni; Pellicciari, Roberto
Design, Molecular Modeling Studies, Synthesis and Preliminary Evaluation of Novel PARP-1 Inhibitors on the Road of Antiischemic Agents 2006 Camaioni, Emidio; P., Sabbatini; Costantino, Gabriele; D., Bellocchi; A., Chiarugi; F., Moroni; A., Wood; Pellicciari, Roberto
Design, Synthesis and Preliminay Evaluation of Novel 3’-Substituted Carboxycyclopropylglycines as Antagonists at Group 2 Metabotropic Glutamate Receptors 2001 Pellicciari, Roberto; Costantino, Gabriele; Marinozzi, Maura; Macchiarulo, Antonio; Amori, L.; Flor, P.; Gasparini, F.; Kuhn, R.; Urwyler, S.
Design, Synthesis, and Microbiolgical Evaluation of New Candida albicans CYP51 Inhibitors 2005 Schiaffella, Fausto; Macchiarulo, Antonio; Milanese, Lara; Vecchiarelli, Anna; Costantino, Gabriele; Pietrella, Donatella; Fringuelli, Renata
Dirhodium(II)-tetraacetate-Mediated Decomposition of Ethyldiazo- acetate and Ethyldiazomalonate in the Presence of Fullerene. A New Procedure for the Selective Synthesis of [6-6]-Closed Methanofullerenes 1997 Pellicciari, Roberto; Annibali, D; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto
Discovery of a AHR pelargonidin agonist that counter-regulates Ace2 expression and attenuates ACE2-SARS-CoV-2 interaction 2021 Biagioli, Michele; Marchianò, Silvia; Roselli, Rosalinda; Di Giorgio, Cristina; Bellini, Rachele; Bordoni, Martina; Gidari, Anna; Sabbatini, Samuele; Francisci, Daniela; Fiorillo, Bianca; Catalanotti, Bruno; Distrutti, Eleonora; Carino, Adriana; Zampella, Angela; Costantino, Gabriele; Fiorucci, Stefano