FELICETTI, TOMMASO
FELICETTI, TOMMASO
DIPARTIMENTO DI SCIENZE FARMACEUTICHE
1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors
2021 Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S.
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
2018 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
An overview on small molecules acting as broad-spectrum agents for yellow fever infection
2022 Desantis, J.; Felicetti, T.; Cannalire, R.
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors
2020 Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O.
Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation
2021 Pica, M.; Messere, N.; Felicetti, T.; Sabatini, S.; Pietrella, D.; Nocchetti, M.
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions
2019 Cannalire, R.; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G.
Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View
2020 Felicetti, T.; Manfroni, G.; Cecchetti, V.; Cannalire, R.
Building up efflux-mediated antimicrobial resistance in Staphylococcus pseudintermedius
2022 Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors
2020 Felicetti, T.; Mangiaterra, G.; Cannalire, R.; Cedraro, N.; Pietrella, D.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Biavasco, F.; Sabatini, S.
Deciphering the molecular recognition mechanism of multidrug resistance staphylococcus aureus nora efflux pump using a supervised molecular dynamics approach
2019 Palazzotti, D.; Bissaro, M.; Bolcato, G.; Astolfi, A.; Felicetti, T.; Sabatini, S.; Sturlese, M.; Cecchetti, V.; Barreca, M. L.; Moro, S.
Design and synthesis of WM5 analogues as HIV-1 TAR RNA binders.
2019 Desantis, J.; Massari, S.; Sosic, A.; Manfroni, G.; Cannalire, R.; Felicetti, T.; Pannecouque, P.; Gatto, B.; Tabarrini, O.
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity
2022 Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana
Discovery of 2‐phenylquinazolines as potent Mycobacterium avium efflux pump inhibitors able to synergize with clarithromycin against clinical isolate
2024 Cernicchi, Giada; Rampacci, Elisa; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Cecchetti, Violetta; Felicetti, Tommaso; Di Luca, Mariagrazia; Poma, Noemi Violeta; Tavanti, Arianna; Passamonti, Fabrizio; Rindi, Laura; Sabatini, Stefano
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation
2019 Astolfi, A.; Kudolo, M.; Brea, J.; Manni, G.; Manfroni, G.; Palazzotti, D.; Sabatini, S.; Cecchetti, F.; Felicetti, T.; Cannalire, R.; Massari, S.; Tabarrini, O.; Loza, M. I.; Fallarino, F.; Cecchetti, V.; Laufer, S. A.; Barreca, M. L.
Drug efflux transporters in Staphylococcus pseudintermedius: in silico prediction and characterization of resistance
2022 Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio
Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi
2021 Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio
EVALUATION OF DRUG EFFLUX ACTIVITY IN ANTIMICROBIAL RESISTANT STAPHYLOCOCCUS PSEUDINTERMEDIUS CLINICAL ISOLATES
2023 Rampacci, Elisa; Felicetti, Tommaso; Birettoni, Francesco; Arcelli, Rolando; Zelli, Riccardo; Sabatini, Stefano; Passamonti, Fabrizio
Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations
2023 Palazzotti, Deborah; Felicetti, Tommaso; Sabatini, Stefano; Moro, Stefano; Barreca, Maria Letizia; Sturlese, Mattia; Astolfi, Andrea
From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors
2019 Massari, Serena; Corona, Angela; Distinto, Simona; Desantis, Jenny; Caredda, Alessia; Sabatini, Stefano; Manfroni, Giuseppe; Felicetti, Tommaso; Cecchetti, Violetta; Pannecouque, Christophe; Maccioni, Elias; Tramontano, Enzo; Tabarrini, Oriana
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
2021 Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors | 2021 | Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S. | |
| 2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction | 2018 | Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano | |
| An overview on small molecules acting as broad-spectrum agents for yellow fever infection | 2022 | Desantis, J.; Felicetti, T.; Cannalire, R. | |
| Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors | 2020 | Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O. | |
| Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation | 2021 | Pica, M.; Messere, N.; Felicetti, T.; Sabatini, S.; Pietrella, D.; Nocchetti, M. | |
| Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions | 2019 | Cannalire, R.; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G. | |
| Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View | 2020 | Felicetti, T.; Manfroni, G.; Cecchetti, V.; Cannalire, R. | |
| Building up efflux-mediated antimicrobial resistance in Staphylococcus pseudintermedius | 2022 | Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio | |
| C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors | 2020 | Felicetti, T.; Mangiaterra, G.; Cannalire, R.; Cedraro, N.; Pietrella, D.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Biavasco, F.; Sabatini, S. | |
| Deciphering the molecular recognition mechanism of multidrug resistance staphylococcus aureus nora efflux pump using a supervised molecular dynamics approach | 2019 | Palazzotti, D.; Bissaro, M.; Bolcato, G.; Astolfi, A.; Felicetti, T.; Sabatini, S.; Sturlese, M.; Cecchetti, V.; Barreca, M. L.; Moro, S. | |
| Design and synthesis of WM5 analogues as HIV-1 TAR RNA binders. | 2019 | Desantis, J.; Massari, S.; Sosic, A.; Manfroni, G.; Cannalire, R.; Felicetti, T.; Pannecouque, P.; Gatto, B.; Tabarrini, O. | |
| Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus Activity | 2022 | Nizi, Maria Giulia; Persoons, Leentje; Corona, Angela; Felicetti, Tommaso; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Vangeel, Laura; Barreca, Maria Letizia; Esposito, Francesca; Jochmans, Dirk; Milia, Jessica; Cecchetti, Violetta; Schols, Dominique; Neyts, Johan; Tramontano, Enzo; Sabatini, Stefano; De Jonghe, Steven; Tabarrini, Oriana | |
| Discovery of 2‐phenylquinazolines as potent Mycobacterium avium efflux pump inhibitors able to synergize with clarithromycin against clinical isolate | 2024 | Cernicchi, Giada; Rampacci, Elisa; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Cecchetti, Violetta; Felicetti, Tommaso; Di Luca, Mariagrazia; Poma, Noemi Violeta; Tavanti, Arianna; Passamonti, Fabrizio; Rindi, Laura; Sabatini, Stefano | |
| Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation | 2019 | Astolfi, A.; Kudolo, M.; Brea, J.; Manni, G.; Manfroni, G.; Palazzotti, D.; Sabatini, S.; Cecchetti, F.; Felicetti, T.; Cannalire, R.; Massari, S.; Tabarrini, O.; Loza, M. I.; Fallarino, F.; Cecchetti, V.; Laufer, S. A.; Barreca, M. L. | |
| Drug efflux transporters in Staphylococcus pseudintermedius: in silico prediction and characterization of resistance | 2022 | Rampacci, Elisa; Felicetti, Tommaso; Pietrella, Donatella; Sabatini, Stefano; Passamonti, Fabrizio | |
| Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi | 2021 | Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio | |
| EVALUATION OF DRUG EFFLUX ACTIVITY IN ANTIMICROBIAL RESISTANT STAPHYLOCOCCUS PSEUDINTERMEDIUS CLINICAL ISOLATES | 2023 | Rampacci, Elisa; Felicetti, Tommaso; Birettoni, Francesco; Arcelli, Rolando; Zelli, Riccardo; Sabatini, Stefano; Passamonti, Fabrizio | |
| Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations | 2023 | Palazzotti, Deborah; Felicetti, Tommaso; Sabatini, Stefano; Moro, Stefano; Barreca, Maria Letizia; Sturlese, Mattia; Astolfi, Andrea | |
| From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors | 2019 | Massari, Serena; Corona, Angela; Distinto, Simona; Desantis, Jenny; Caredda, Alessia; Sabatini, Stefano; Manfroni, Giuseppe; Felicetti, Tommaso; Cecchetti, Violetta; Pannecouque, Christophe; Maccioni, Elias; Tramontano, Enzo; Tabarrini, Oriana | |
| From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | 2021 | Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano |