ELEUTERI, MICHELA
ELEUTERI, MICHELA
Between Theory and Practice: Computational/Experimental Integrated Approaches to Understand the Solubility and Lipophilicity of PROTACs
2024 Venturi, Andrea; Di Bona, Stefano; Desantis, Jenny; Eleuteri, Michela; Bartalucci, Matteo; Baroni, Massimo; Benedetti, Paolo; Goracci, Laura; Cruciani, Gabriele
Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity
2024 Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura
Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization
2022 Mercorelli, Beatrice; Desantis, Jenny; Celegato, Marta; Bazzacco, Alessandro; Siragusa, Lydia; Benedetti, Paolo; Eleuteri, Michela; Croci, Federico; Cruciani, Gabriele; Goracci, Laura; Loregian, Arianna
PROTACs bearing piperazine-containing linkers: what effect on their protonation state?
2022 Desantis, Jenny; Mammoli, Andrea; Eleuteri, Michela; Coletti, Alice; Croci, Federico; Macchiarulo, Antonio; Goracci, Laura
Understanding the Metabolism of Proteolysis Targeting Chimeras (PROTACs): The Next Step toward Pharmaceutical Applications
2020 Goracci, L.; Desantis, J.; Valeri, A.; Castellani, B.; Eleuteri, M.; Cruciani, G.
Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis
2024 Eleuteri, Michela; Desantis, Jenny; Cruciani, Gabriele; Germani, Raimondo; Goracci, Laura
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications
2023 Castellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Between Theory and Practice: Computational/Experimental Integrated Approaches to Understand the Solubility and Lipophilicity of PROTACs | 2024 | Venturi, Andrea; Di Bona, Stefano; Desantis, Jenny; Eleuteri, Michela; Bartalucci, Matteo; Baroni, Massimo; Benedetti, Paolo; Goracci, Laura; Cruciani, Gabriele | |
| Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity | 2024 | Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura | |
| Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization | 2022 | Mercorelli, Beatrice; Desantis, Jenny; Celegato, Marta; Bazzacco, Alessandro; Siragusa, Lydia; Benedetti, Paolo; Eleuteri, Michela; Croci, Federico; Cruciani, Gabriele; Goracci, Laura; Loregian, Arianna | |
| PROTACs bearing piperazine-containing linkers: what effect on their protonation state? | 2022 | Desantis, Jenny; Mammoli, Andrea; Eleuteri, Michela; Coletti, Alice; Croci, Federico; Macchiarulo, Antonio; Goracci, Laura | |
| Understanding the Metabolism of Proteolysis Targeting Chimeras (PROTACs): The Next Step toward Pharmaceutical Applications | 2020 | Goracci, L.; Desantis, J.; Valeri, A.; Castellani, B.; Eleuteri, M.; Cruciani, G. | |
| Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis | 2024 | Eleuteri, Michela; Desantis, Jenny; Cruciani, Gabriele; Germani, Raimondo; Goracci, Laura | |
| VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications | 2023 | Castellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura |