ELEUTERI, MICHELA

ELEUTERI, MICHELA  

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Titolo Data di pubblicazione Autore(i) File
Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity 2024 Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura
Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization 2022 Mercorelli, Beatrice; Desantis, Jenny; Celegato, Marta; Bazzacco, Alessandro; Siragusa, Lydia; Benedetti, Paolo; Eleuteri, Michela; Croci, Federico; Cruciani, Gabriele; Goracci, Laura; Loregian, Arianna
PROTACs bearing piperazine-containing linkers: what effect on their protonation state? 2022 Desantis, Jenny; Mammoli, Andrea; Eleuteri, Michela; Coletti, Alice; Croci, Federico; Macchiarulo, Antonio; Goracci, Laura
Understanding the Metabolism of Proteolysis Targeting Chimeras (PROTACs): The Next Step toward Pharmaceutical Applications 2020 Goracci, L.; Desantis, J.; Valeri, A.; Castellani, B.; Eleuteri, M.; Cruciani, G.
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications 2023 Castellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura