Sfoglia per Rivista
1,4 Benzothiazine and 1,4 benzoxazine imidazole derivatives with antifungal activity: a docking study
2002 Macchiarulo, Antonio; Costantino, Gabriele; Fringuelli, D.; Vecchiarelli, Anna; Schiaffella, Fausto; Fringuelli, Renata
1,4-Benzothiazine analogues and apoptosis: structure-activity relationship
2003 Fringuelli, Renata; Schiaffella, Fausto; Utrilla Navarro, M. P.; Milanese, Lara; Santini, C.; Rapucci, M.; Marchetti, Maria Cristina; Riccardi, Carlo
5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel anti-inflammatory agents
2005 Ottanà, R.; Maccari, R.; Barreca, MARIA LETIZIA; Bruno, G.; Rotondo, A.; Rossi, A.; Chiricosta, G.; Di Paola, R.; Sautebin, L.; Cuzzocrea, S.; Vigorita, M. G.
7-(Disubstituted thiazolyl)-3,5-dihydroxy-6-heptenoic/heptanoic acid derivatives as HMG-COa reductase inhibitors
1994 Cecchetti, Violetta; Fravolini, Arnaldo; Pier Giuseppe, Pagella; Tabarrini, Oriana; Temperini, Andrea
Adenosine receptor agonists: Synthesis and biological evaluation of the diastereoisomers of 2-(3-hydroxy-3-phenyl-1-propyn-1-yl)NECA
1997 Camaioni, Emidio; Di Francesco, E; Vittori, S; Volpini, R; Cristalli, G.
Anti-Candida albicans properties of novel benzoxazine analogues
2002 Fringuelli, Renata; Pietrella, Donatella; Schiaffella, Fausto; Guarraci, Alessia; Perito, Stefano; Bistoni, Francesco; Vecchiarelli, Anna
Asymmetric synthesis of the four diastereoisomers of a novel non-steroidal farnesoid X receptor (FXR) agonist: Role of the chirality on the biological activity
2013 Marinozzi, Maura; Carotti, Andrea; Sardella, Roccaldo; Federica, Buonerba; Ianni, Federica; Natalini, Benedetto; Daniela, Passeri; Giovanni, Rizzo; Pellicciari, Roberto
Azole derivatives of 1,4 benzothiazine as antifungal agents.
1998 Fringuelli, Renata; Schiaffella, Fausto; Bistoni, Francesco; Pitzurra, Lucia; Vecchiarelli, Anna
Azole derivatives of 1,4-benzothiazine as antifungal agents.
1998 Fringuelli, Renata; Schiaffella, Fausto; Bistoni, Francesco; Pitzurra, Lucia; Vecchiarelli, Anna
Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K-ATP channel openers
2005 Carosati, Emanuele; Lemoine, H.; Spogli, Roberto; Grittner, D.; Mannhold, R.; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta
Bulky 1,4-benzoxazine derivatives with antifungal activity
2009 Fringuelli, Renata; Giacche', Nicola; Milanese, Lara; Cenci, Elio; Macchiarulo, Antonio; Vecchiarelli, Anna; Costantino, Gabriele; Schiaffella, Fausto
Cyathane diterpenes from Sarcodon cyrneus and evaluation of their activities of neuritegenesis and nerve growth factor production
2007 Marcotullio, Maria Carla; Pagiotti, Rita; Maltese, F.; Oball Mond Mwankie, G. N.; Hoshino, T.; Obara, Y.; Nakahata, N.
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands.
2009 Filosa, R.; Fulco, MARIA CARMELA; Marinozzi, Maura; Giacchè, N.; Macchiarulo, Antonio; Peduto, A.; Massa, A.; De Caprariis, P.; Thomsen, C.; Christoffersen, C.; Pellicciari, Roberto
Design, synthesis and in vitro antitumor activity of new trans 2-[2-(heteroaryl)vinyl]-1,3-dimethylimidazolium iodides
2004 Ballistreri, Francesco P.; Barresi, Vincenza; Benedetti, Paolo; Caltabiano, Gianluigi; Fortuna, COSIMO GIANLUCA; Longo, Maria L.; Musumarra, Giuseppe
Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents.
2009 Monforte, A. M.; Logoteta, P.; Ferro, S.; De Luca, L.; Iraci, Nunzio; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A.
Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole.
2005 Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto
Ester derivatives of annulated tetrahydroazocines: a new class of selective acetylcholinesterase inhibitors
2006 Carotti, Andrea; M., de Candia; M., Catto; T. N., Borisova; A. V., Varlamov; E., Mendez Alvarez; R., Soto Otero; L. G., Voskressensky; C., Altomare
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands
2014 Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana
Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3a,7a-dihydroxy-6a-ethyl-24-nor-5b-cholan-23-amine
2011 Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; P., Filipponi; G., Costantino; G., Rizzo; L., Adorini; Pellicciari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,4 Benzothiazine and 1,4 benzoxazine imidazole derivatives with antifungal activity: a docking study | 2002 | Macchiarulo, Antonio; Costantino, Gabriele; Fringuelli, D.; Vecchiarelli, Anna; Schiaffella, Fausto; Fringuelli, Renata | |
1,4-Benzothiazine analogues and apoptosis: structure-activity relationship | 2003 | Fringuelli, Renata; Schiaffella, Fausto; Utrilla Navarro, M. P.; Milanese, Lara; Santini, C.; Rapucci, M.; Marchetti, Maria Cristina; Riccardi, Carlo | |
5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel anti-inflammatory agents | 2005 | Ottanà, R.; Maccari, R.; Barreca, MARIA LETIZIA; Bruno, G.; Rotondo, A.; Rossi, A.; Chiricosta, G.; Di Paola, R.; Sautebin, L.; Cuzzocrea, S.; Vigorita, M. G. | |
7-(Disubstituted thiazolyl)-3,5-dihydroxy-6-heptenoic/heptanoic acid derivatives as HMG-COa reductase inhibitors | 1994 | Cecchetti, Violetta; Fravolini, Arnaldo; Pier Giuseppe, Pagella; Tabarrini, Oriana; Temperini, Andrea | |
Adenosine receptor agonists: Synthesis and biological evaluation of the diastereoisomers of 2-(3-hydroxy-3-phenyl-1-propyn-1-yl)NECA | 1997 | Camaioni, Emidio; Di Francesco, E; Vittori, S; Volpini, R; Cristalli, G. | |
Anti-Candida albicans properties of novel benzoxazine analogues | 2002 | Fringuelli, Renata; Pietrella, Donatella; Schiaffella, Fausto; Guarraci, Alessia; Perito, Stefano; Bistoni, Francesco; Vecchiarelli, Anna | |
Asymmetric synthesis of the four diastereoisomers of a novel non-steroidal farnesoid X receptor (FXR) agonist: Role of the chirality on the biological activity | 2013 | Marinozzi, Maura; Carotti, Andrea; Sardella, Roccaldo; Federica, Buonerba; Ianni, Federica; Natalini, Benedetto; Daniela, Passeri; Giovanni, Rizzo; Pellicciari, Roberto | |
Azole derivatives of 1,4 benzothiazine as antifungal agents. | 1998 | Fringuelli, Renata; Schiaffella, Fausto; Bistoni, Francesco; Pitzurra, Lucia; Vecchiarelli, Anna | |
Azole derivatives of 1,4-benzothiazine as antifungal agents. | 1998 | Fringuelli, Renata; Schiaffella, Fausto; Bistoni, Francesco; Pitzurra, Lucia; Vecchiarelli, Anna | |
Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K-ATP channel openers | 2005 | Carosati, Emanuele; Lemoine, H.; Spogli, Roberto; Grittner, D.; Mannhold, R.; Tabarrini, Oriana; Sabatini, Stefano; Cecchetti, Violetta | |
Bulky 1,4-benzoxazine derivatives with antifungal activity | 2009 | Fringuelli, Renata; Giacche', Nicola; Milanese, Lara; Cenci, Elio; Macchiarulo, Antonio; Vecchiarelli, Anna; Costantino, Gabriele; Schiaffella, Fausto | |
Cyathane diterpenes from Sarcodon cyrneus and evaluation of their activities of neuritegenesis and nerve growth factor production | 2007 | Marcotullio, Maria Carla; Pagiotti, Rita; Maltese, F.; Oball Mond Mwankie, G. N.; Hoshino, T.; Obara, Y.; Nakahata, N. | |
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi | |
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands. | 2009 | Filosa, R.; Fulco, MARIA CARMELA; Marinozzi, Maura; Giacchè, N.; Macchiarulo, Antonio; Peduto, A.; Massa, A.; De Caprariis, P.; Thomsen, C.; Christoffersen, C.; Pellicciari, Roberto | |
Design, synthesis and in vitro antitumor activity of new trans 2-[2-(heteroaryl)vinyl]-1,3-dimethylimidazolium iodides | 2004 | Ballistreri, Francesco P.; Barresi, Vincenza; Benedetti, Paolo; Caltabiano, Gianluigi; Fortuna, COSIMO GIANLUCA; Longo, Maria L.; Musumarra, Giuseppe | |
Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents. | 2009 | Monforte, A. M.; Logoteta, P.; Ferro, S.; De Luca, L.; Iraci, Nunzio; Maga, G.; De Clercq, E.; Pannecouque, C.; Chimirri, A. | |
Docking studies on PARP-1 inhibitors: insights into the role of a binding pocket water molecole. | 2005 | Bellocchi, Daniele; Macchiarulo, Antonio; Costantino, Gabriele; Pellicciari, Roberto | |
Ester derivatives of annulated tetrahydroazocines: a new class of selective acetylcholinesterase inhibitors | 2006 | Carotti, Andrea; M., de Candia; M., Catto; T. N., Borisova; A. V., Varlamov; E., Mendez Alvarez; R., Soto Otero; L. G., Voskressensky; C., Altomare | |
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands | 2014 | Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana | |
Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3a,7a-dihydroxy-6a-ethyl-24-nor-5b-cholan-23-amine | 2011 | Gioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; P., Filipponi; G., Costantino; G., Rizzo; L., Adorini; Pellicciari, Roberto |
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