Sfoglia per Autore
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana
Blocking HIV-1 Replication by Targeting the TAT-Hijacked Transcriptional Machinery
2013 Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana
Structural Investigation of Cycloheptathiophene-3-carboxamide Derivatives Targeting Influenza Virus Polymerase Assembly
2013 Massari, Serena; Nannetti, Giulio; Goracci, Laura; Sancineto, Luca; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Facchini, Marzia; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Tabarrini, Oriana
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions
2013 Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance
2013 Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta
Design, Synthesis, and Evaluation of WC5 Analogues as Inhibitors of Human Cytomegalovirus Immediate-Early 2 Protein, a Promising Target for Anti-HCMV Treatment
2013 Massari, Serena; Mercorelli, Beatrice; Sancineto, Luca; Sabatini, Stefano; Cecchetti, Violetta; Gribaudo, Giorgio; Palù, Giorgio; Pannecouque, Arianna; Loregian, Christophe; Tabarrini, Oriana
From Small to Powerful: The Fragments Universe and its "Chem-Appeal"
2013 Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Tabarrini, Oriana
The 6-Aminoquinolone WC5 inhibits different functions of the immediate-early 2 (IE2) protein of human cytomegalovirus that are essential for viral replication
2014 Mercorelli, Beatrice; Luganini, Anna; Muratore, Giulia; Massari, Serena; Terlizzi, Maria Elena; Tabarrini, Oriana; Gribaudo, Giorgio; Palù, Giorgio; Loregian, Arianna
Modulation of HIV-1-Induced Activation of Plasmacytoid Dendritic Cells by 6-Desfluoroquinolones
2014 Caroline M., Royle; Ming Han, Tsai; Tabarrini, Oriana; Massari, Serena; David R., Graham; Veronica N., Aquino; Adriano, Boasso
Ethyl 1,8-Naphthyridone-3-carboxylates Downregulate Human Papillomavirus-16 (HPV-16) E6 and E7 Oncogenes Expression
2014 Donalisio, Manuela; Massari, Serena; Argenziano, Monica; Manfroni, Giuseppe; Cagno, Valeria; Civra, Andrea; Sabatini, Stefano; Cecchetti, Violetta; Loregian, Arianna; Cavalli, Roberta; Lembo, David; Tabarrini, Oriana
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands
2014 Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction
2015 Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana
The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors
2015 Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Bauer, Silke M; Gargaro, Marco; Cannalire, Rolando; Astolfi, Andrea; Brea, Jose; Vacca, Carmine; Pirro, Matteo; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Laufer, Stefan A; Cecchetti, Violetta
Phospholipidosis effect of drugs by adsorption into lipid monolayers
2015 Ceccarelli, Martina; Germani, Raimondo; Massari, Serena; Petit, Charlotte; Nurisso, Alessandra; Wolfender, Jean Luc; Goracci, Laura
Recent advances in the identification of Tat-mediated transactivation inhibitors: progressing toward a functional cure of HIV
2016 Tabarrini, Oriana; Desantis, Jenny; Massari, Serena
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors
2016 Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J.; Tramontano, Enzo; Tabarrini, Oriana
Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Protein-protein Interaction as a Target for Next-generation Anti-influenza Therapeutics.
2016 Massari, Serena; Goracci, Laura; Desantis, Jenny; Tabarrini, Oriana
Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency
2017 Tabarrini, O.; Massari, S.
Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium
2017 Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors
2017 Astolfi, Andrea; Felicetti, Tommaso; Iraci, Nunzio; Manfroni, Giuseppe; Massari, Serena; Pietrella, Donatella; Tabarrini, Oriana; Kaatz, Glenn W.; Barreca, MARIA LETIZIA; Sabatini, Stefano; Cecchetti, Violetta
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana | |
| Blocking HIV-1 Replication by Targeting the TAT-Hijacked Transcriptional Machinery | 2013 | Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana | |
| Structural Investigation of Cycloheptathiophene-3-carboxamide Derivatives Targeting Influenza Virus Polymerase Assembly | 2013 | Massari, Serena; Nannetti, Giulio; Goracci, Laura; Sancineto, Luca; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Facchini, Marzia; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Tabarrini, Oriana | |
| 1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions | 2013 | Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta | |
| Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance | 2013 | Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta | |
| Design, Synthesis, and Evaluation of WC5 Analogues as Inhibitors of Human Cytomegalovirus Immediate-Early 2 Protein, a Promising Target for Anti-HCMV Treatment | 2013 | Massari, Serena; Mercorelli, Beatrice; Sancineto, Luca; Sabatini, Stefano; Cecchetti, Violetta; Gribaudo, Giorgio; Palù, Giorgio; Pannecouque, Arianna; Loregian, Christophe; Tabarrini, Oriana | |
| From Small to Powerful: The Fragments Universe and its "Chem-Appeal" | 2013 | Sancineto, Luca; Massari, Serena; Iraci, Nunzio; Tabarrini, Oriana | |
| The 6-Aminoquinolone WC5 inhibits different functions of the immediate-early 2 (IE2) protein of human cytomegalovirus that are essential for viral replication | 2014 | Mercorelli, Beatrice; Luganini, Anna; Muratore, Giulia; Massari, Serena; Terlizzi, Maria Elena; Tabarrini, Oriana; Gribaudo, Giorgio; Palù, Giorgio; Loregian, Arianna | |
| Modulation of HIV-1-Induced Activation of Plasmacytoid Dendritic Cells by 6-Desfluoroquinolones | 2014 | Caroline M., Royle; Ming Han, Tsai; Tabarrini, Oriana; Massari, Serena; David R., Graham; Veronica N., Aquino; Adriano, Boasso | |
| Ethyl 1,8-Naphthyridone-3-carboxylates Downregulate Human Papillomavirus-16 (HPV-16) E6 and E7 Oncogenes Expression | 2014 | Donalisio, Manuela; Massari, Serena; Argenziano, Monica; Manfroni, Giuseppe; Cagno, Valeria; Civra, Andrea; Sabatini, Stefano; Cecchetti, Violetta; Loregian, Arianna; Cavalli, Roberta; Lembo, David; Tabarrini, Oriana | |
| Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands | 2014 | Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana | |
| A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction | 2015 | Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana | |
| The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors | 2015 | Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Bauer, Silke M; Gargaro, Marco; Cannalire, Rolando; Astolfi, Andrea; Brea, Jose; Vacca, Carmine; Pirro, Matteo; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Laufer, Stefan A; Cecchetti, Violetta | |
| Phospholipidosis effect of drugs by adsorption into lipid monolayers | 2015 | Ceccarelli, Martina; Germani, Raimondo; Massari, Serena; Petit, Charlotte; Nurisso, Alessandra; Wolfender, Jean Luc; Goracci, Laura | |
| Recent advances in the identification of Tat-mediated transactivation inhibitors: progressing toward a functional cure of HIV | 2016 | Tabarrini, Oriana; Desantis, Jenny; Massari, Serena | |
| Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors | 2016 | Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J.; Tramontano, Enzo; Tabarrini, Oriana | |
| Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Protein-protein Interaction as a Target for Next-generation Anti-influenza Therapeutics. | 2016 | Massari, Serena; Goracci, Laura; Desantis, Jenny; Tabarrini, Oriana | |
| Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency | 2017 | Tabarrini, O.; Massari, S. | |
| Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium | 2017 | Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta | |
| Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors | 2017 | Astolfi, Andrea; Felicetti, Tommaso; Iraci, Nunzio; Manfroni, Giuseppe; Massari, Serena; Pietrella, Donatella; Tabarrini, Oriana; Kaatz, Glenn W.; Barreca, MARIA LETIZIA; Sabatini, Stefano; Cecchetti, Violetta |
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