Sfoglia per Autore
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor.
2009 Manfroni, Giuseppe; Paeshuyse, J; Massari, Serena; Gatto, B; Zanoli, S; Maga, G; Tabarrini, Oriana; Cecchetti, Violetta; Fravolini, Arnaldo; Neyts, J.
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position
2009 Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta
Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid catalyzed Aminolysis of 2,2-Dimethylthiirane as Precursors of the 1,4-Benzothiazine Nucleus
2009 Spogli, Roberto; Sabatini, Stefano; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta
Sintesi di nuovi inibitori della pompa di efflusso NorA dello S. aureus: dalle 3-fenil-1,4-benzotiazine alle 2-fenilchinossaline
2010 Capone, C.; Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta
Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives
2010 Tabarrini, Oriana; Massari, Serena; Daelemans, D; Meschini, Francesco; Manfroni, Giuseppe; Bottega, L; Gatto, B; Palumbo, M; Pannecouque, C; Cecchetti, Violetta
DERIVATI 2-FENIL-4-IDROSSI-CHINOLINICI COME POTENTI INBITORI DELLA POMPA D’EFFLUSSO NorA DELLO S. aureus
2011 Sabatini, Stefano; Gosetto, Francesca; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta
N-Benzoyl-N-methylsulfonyl anthranilates: unexpected cyclization reaction to 4-alkoxy-2,1-benzothiazines
2011 Manfroni, Giuseppe; Meschini, Francesco; Costantino, Ferdinando; Tabarrini, Oriana; Cecchetti, Violetta
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus.
2011 Brincat, JEAN PIERRE; Carosati, Emanuele; Sabatini, Stefano; Manfroni, Giuseppe; Fravolini, Arnaldo; Raygada, Jl; Patel, D; Kaatz, Gw; Cruciani, Gabriele
Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump.
2011 Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Kaatz, G. W.; Patel, D.; Cecchetti, Violetta
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development
2011 Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Cecchetti, Violetta
Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity.
2011 Tabarrini, Oriana; Massari, Serena; Sancineto, Luca; Daelemans, D.; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Pannecouque, C.
6-Aminoquinolones targeting HCV NS5B polymerase.
2012 Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta
Structural optimization of the 2-Phenyl-4-hydroxyquinoline Class of S. aureus NorA Efflux Pump Inhibitors
2012 Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; A. M., Schito; G. W., Kaatz; Cecchetti, Violetta
Targeting the HIV Tat-mediated transcriptional machinery: P-TEFb complex inhibitors
2012 Tabarrini, Oriana; Sancineto, Luca; Iraci, Nunzio; Massari, Serena; V., Attanasio; Sabatini, Stefano; Manfroni, Giuseppe; A., Marcello; Cecchetti, Violetta
New chemotypes to fight HCV infection: discovery of selective inhibitors of HCV replication with pyrazolobenzothiazine scaffold
2012 Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Iraci, Nunzio; Cannalire, R.; Tabarrini, Oriana; Cecchetti, Violetta
A New Promising Class of pyrazolobenzothiazine inhibitors of S. aureus NorA Efflux Pump
2012 Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Carosati, Emanuele; Cecchetti, Violetta
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors
2012 Sabatini, Stefano; Gosetto, F; Serritella, S; Manfroni, Giuseppe; Tabarrini, Oriana; Iraci, Nunzio; Brincat, Jp; Carosati, Emanuele; Villarini, Milena; Kaatz, Gw; Cecchetti, Violetta
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase
2012 Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors
2013 Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor. | 2009 | Manfroni, Giuseppe; Paeshuyse, J; Massari, Serena; Gatto, B; Zanoli, S; Maga, G; Tabarrini, Oriana; Cecchetti, Violetta; Fravolini, Arnaldo; Neyts, J. | |
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position | 2009 | Massari, Serena; Daelemans, D; Manfroni, Giuseppe; Sabatini, Stefano; Tabarrini, Oriana; Pannecouque, C; Cecchetti, Violetta | |
Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid catalyzed Aminolysis of 2,2-Dimethylthiirane as Precursors of the 1,4-Benzothiazine Nucleus | 2009 | Spogli, Roberto; Sabatini, Stefano; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta | |
Sintesi di nuovi inibitori della pompa di efflusso NorA dello S. aureus: dalle 3-fenil-1,4-benzotiazine alle 2-fenilchinossaline | 2010 | Capone, C.; Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Cecchetti, Violetta | |
Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives | 2010 | Tabarrini, Oriana; Massari, Serena; Daelemans, D; Meschini, Francesco; Manfroni, Giuseppe; Bottega, L; Gatto, B; Palumbo, M; Pannecouque, C; Cecchetti, Violetta | |
DERIVATI 2-FENIL-4-IDROSSI-CHINOLINICI COME POTENTI INBITORI DELLA POMPA D’EFFLUSSO NorA DELLO S. aureus | 2011 | Sabatini, Stefano; Gosetto, Francesca; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta | |
N-Benzoyl-N-methylsulfonyl anthranilates: unexpected cyclization reaction to 4-alkoxy-2,1-benzothiazines | 2011 | Manfroni, Giuseppe; Meschini, Francesco; Costantino, Ferdinando; Tabarrini, Oriana; Cecchetti, Violetta | |
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus. | 2011 | Brincat, JEAN PIERRE; Carosati, Emanuele; Sabatini, Stefano; Manfroni, Giuseppe; Fravolini, Arnaldo; Raygada, Jl; Patel, D; Kaatz, Gw; Cruciani, Gabriele | |
Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump. | 2011 | Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Kaatz, G. W.; Patel, D.; Cecchetti, Violetta | |
Allosteric inhibition of the hepatitis C virus NS5B polymerase: in silico strategies for drug discovery and development | 2011 | Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Cecchetti, Violetta | |
Structural investigation of the naphthyridone scaffold: identification of a 1,6-naphthyridone derivative with potent and selective anti-HIV activity. | 2011 | Tabarrini, Oriana; Massari, Serena; Sancineto, Luca; Daelemans, D.; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Pannecouque, C. | |
6-Aminoquinolones targeting HCV NS5B polymerase. | 2012 | Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta | |
Structural optimization of the 2-Phenyl-4-hydroxyquinoline Class of S. aureus NorA Efflux Pump Inhibitors | 2012 | Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; A. M., Schito; G. W., Kaatz; Cecchetti, Violetta | |
Targeting the HIV Tat-mediated transcriptional machinery: P-TEFb complex inhibitors | 2012 | Tabarrini, Oriana; Sancineto, Luca; Iraci, Nunzio; Massari, Serena; V., Attanasio; Sabatini, Stefano; Manfroni, Giuseppe; A., Marcello; Cecchetti, Violetta | |
New chemotypes to fight HCV infection: discovery of selective inhibitors of HCV replication with pyrazolobenzothiazine scaffold | 2012 | Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Iraci, Nunzio; Cannalire, R.; Tabarrini, Oriana; Cecchetti, Violetta | |
A New Promising Class of pyrazolobenzothiazine inhibitors of S. aureus NorA Efflux Pump | 2012 | Sabatini, Stefano; Gosetto, Francesca; Manfroni, Giuseppe; Tabarrini, Oriana; Carosati, Emanuele; Cecchetti, Violetta | |
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors | 2012 | Sabatini, Stefano; Gosetto, F; Serritella, S; Manfroni, Giuseppe; Tabarrini, Oriana; Iraci, Nunzio; Brincat, Jp; Carosati, Emanuele; Villarini, Milena; Kaatz, Gw; Cecchetti, Violetta | |
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase | 2012 | Manfroni, Giuseppe; Meschini, Francesco; Barreca, MARIA LETIZIA; P., Leyssen; A., Samuele; Iraci, Nunzio; Sabatini, Stefano; Massari, Serena; G., Maga; J., Neyts; Cecchetti, Violetta | |
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors | 2013 | Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana |
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