Sfoglia per Autore
CYCLOHEPTATHIOPHENE-3-CARBOXAMIDE DERIVATIVES AS INFLUENZA A VIRUS POLYMERASE INHIBITORS
2013 Massari, Serena; Giulio, Nannetti; Giulia, Muratore; Jenny, Desantis; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Beatrice, Mercorelli; Giorgio, Palù; Arianna, Loregian; Tabarrini, Oriana
Targeting CDKs to inhibit the HIV-1 TAT-mediated transcription
2013 Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Structural investigations of the 2-phenyl-4-hydroxyquinoline class of S. aureus NorA EPIs
2013 Sabatini, Stefano; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; Kaatz, G. W.; Cecchetti, Violetta
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors
2013 Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana
Small molecole targeting HPV E6 and E7 oncoproteins expression.
2013 Massari, Serena; Donaliso, M.; Ansideri, F.; Sancineto, Luca; Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Cecchetti, Violetta; Lembo, D.; Tabarrini, Oriana
STRUCTURAL INVESTIGATIONS OF THE 2-PHENYL-4- HYDROXYQUINOLINE CLASS OF S. AUREUS NORA EPIS
2013 Sabatini, Stefano; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; Glenn W., Kaatz; Cecchetti, Violetta
SMALL MOLECULES TARGETING HPV E6 AND E7 ONCOPROTEINS EXPRESSION
2013 Massari, Serena; Manuela, Donaliso; Francesco, Ansideri; Sancineto, Luca; Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Cecchetti, Violetta; David, Lembo; Tabarrini, Oriana
Structural investigation of Small Molecules Targeting Influenza A Virus Polymerase
2013 Desantis, J.; Nannetti, G.; Massari, Serena; Muratore, G.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Palù, G.; Loregian, A.; Tabarrini, Oriana
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions
2013 Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta
Lipid nanoparticles for brain targeting III. Long-term stability and in vivo toxicity
2013 Paolo, Blasi; Schoubben, Aurelie Marie Madeleine; Traina, Giovanna; Manfroni, Giuseppe; Barberini, Lanfranco; Alberti, Paolo Francesco; Cirotto, Carlo; Ricci, Maurizio
Structural Investigation of Cycloheptathiophene-3-carboxamide Derivatives Targeting Influenza Virus Polymerase Assembly
2013 Massari, Serena; Nannetti, Giulio; Goracci, Laura; Sancineto, Luca; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Facchini, Marzia; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Tabarrini, Oriana
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance
2013 Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta
Accounting for target flexibility and water molecules by docking to ensembles of target structures: The HCV NS5B Palm Site I inhibitors case study.
2014 Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Gaetani, Rosy; Guercini, Chiara; Sabatini, Stefano; Tabarrini, Oriana; Cecchetti, Violetta
The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors
2014 Manfroni, Giuseppe; Cannalire, Rolando; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Winquist, Johan; Iraci, Nunzio; Manvar, Dinesh; Paeshuyse, Jan; Guhamazumder, Rupa; Basu, Amartya; Sabatini, Stefano; Tabarrini, Oriana; Danielson U., Helena; Neyts, Johan; Cecchetti, Violetta
New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors
2014 Manfroni, Giuseppe; Manvar, Dinesh; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta
Enantioresolution, stereochemical characterization and biological activity of a chiral large-conductance calcium-activated potassium channel opener.
2014 Sardella, Roccaldo; Carotti, Andrea; Manfroni, Giuseppe; Tedesco, D; Martelli, A; Bertucci, C; Cecchetti, Violetta; Natalini, Benedetto
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands
2014 Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
CYCLOHEPTATHIOPHENE-3-CARBOXAMIDE DERIVATIVES AS INFLUENZA A VIRUS POLYMERASE INHIBITORS | 2013 | Massari, Serena; Giulio, Nannetti; Giulia, Muratore; Jenny, Desantis; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Beatrice, Mercorelli; Giorgio, Palù; Arianna, Loregian; Tabarrini, Oriana | |
Targeting CDKs to inhibit the HIV-1 TAT-mediated transcription | 2013 | Iraci, Nunzio; Barreca, MARIA LETIZIA; Sancineto, Luca; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Iraci, Nunzio; Sancineto, Luca; Barreca, MARIA LETIZIA; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Structural investigations of the 2-phenyl-4-hydroxyquinoline class of S. aureus NorA EPIs | 2013 | Sabatini, Stefano; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; Kaatz, G. W.; Cecchetti, Violetta | |
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors | 2013 | Massari, Serena; Nannetti, G.; Muratore, G.; Desantis, J.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Mercorelli, B.; Palù, G.; Loregian, A.; Tabarrini, Oriana | |
Small molecole targeting HPV E6 and E7 oncoproteins expression. | 2013 | Massari, Serena; Donaliso, M.; Ansideri, F.; Sancineto, Luca; Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Cecchetti, Violetta; Lembo, D.; Tabarrini, Oriana | |
STRUCTURAL INVESTIGATIONS OF THE 2-PHENYL-4- HYDROXYQUINOLINE CLASS OF S. AUREUS NORA EPIS | 2013 | Sabatini, Stefano; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Tabarrini, Oriana; Glenn W., Kaatz; Cecchetti, Violetta | |
SMALL MOLECULES TARGETING HPV E6 AND E7 ONCOPROTEINS EXPRESSION | 2013 | Massari, Serena; Manuela, Donaliso; Francesco, Ansideri; Sancineto, Luca; Sabatini, Stefano; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Cecchetti, Violetta; David, Lembo; Tabarrini, Oriana | |
Structural investigation of Small Molecules Targeting Influenza A Virus Polymerase | 2013 | Desantis, J.; Nannetti, G.; Massari, Serena; Muratore, G.; Sabatini, Stefano; Sancineto, Luca; Manfroni, Giuseppe; Palù, G.; Loregian, A.; Tabarrini, Oriana | |
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions | 2013 | Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta | |
Lipid nanoparticles for brain targeting III. Long-term stability and in vivo toxicity | 2013 | Paolo, Blasi; Schoubben, Aurelie Marie Madeleine; Traina, Giovanna; Manfroni, Giuseppe; Barberini, Lanfranco; Alberti, Paolo Francesco; Cirotto, Carlo; Ricci, Maurizio | |
Structural Investigation of Cycloheptathiophene-3-carboxamide Derivatives Targeting Influenza Virus Polymerase Assembly | 2013 | Massari, Serena; Nannetti, Giulio; Goracci, Laura; Sancineto, Luca; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Facchini, Marzia; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Tabarrini, Oriana | |
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Vanessa, Attanasio; Gianmarco, Corazza; Barreca, MARIA LETIZIA; Sabatini, Stefano; Manfroni, Giuseppe; Nilla Roberta, Avanzi; Cecchetti, Violetta; Christophe, Pannecouque; Alessandro, Marcello; Tabarrini, Oriana | |
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance | 2013 | Sabatini, Stefano; Gosetto, Francesca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Sancineto, Luca; Manfroni, Giuseppe; Tabarrini, Oriana; Mirjana, Dimovska; Glenn W., Kaatz; Cecchetti, Violetta | |
Accounting for target flexibility and water molecules by docking to ensembles of target structures: The HCV NS5B Palm Site I inhibitors case study. | 2014 | Barreca, MARIA LETIZIA; Iraci, Nunzio; Manfroni, Giuseppe; Gaetani, Rosy; Guercini, Chiara; Sabatini, Stefano; Tabarrini, Oriana; Cecchetti, Violetta | |
The versatile nature of the 6-aminoquinolone scaffold: identification of submicromolar hepatitis C virus NS5B inhibitors | 2014 | Manfroni, Giuseppe; Cannalire, Rolando; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Winquist, Johan; Iraci, Nunzio; Manvar, Dinesh; Paeshuyse, Jan; Guhamazumder, Rupa; Basu, Amartya; Sabatini, Stefano; Tabarrini, Oriana; Danielson U., Helena; Neyts, Johan; Cecchetti, Violetta | |
New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors | 2014 | Manfroni, Giuseppe; Manvar, Dinesh; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta | |
Enantioresolution, stereochemical characterization and biological activity of a chiral large-conductance calcium-activated potassium channel opener. | 2014 | Sardella, Roccaldo; Carotti, Andrea; Manfroni, Giuseppe; Tedesco, D; Martelli, A; Bertucci, C; Cecchetti, Violetta; Natalini, Benedetto | |
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands | 2014 | Sancineto, Luca; Iraci, Nunzio; Barreca, MARIA LETIZIA; Massari, Serena; Manfroni, Giuseppe; Gianmarco, Corazza; Cecchetti, Violetta; Alessandro, Marcello; Dirk, Daelemans; Christophe, Pannecouque; Tabarrini, Oriana |
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