Sfoglia per Autore
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi
Conformational requirements for interaction of L-glutamate with the metabotropic EAA receptor
1993 Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto
SULFATE ESTERS OF HYDROXY AMINO-ACIDS AS STEREOSPECIFIC GLUTAMATE-RECEPTOR AGONISTS
1994 G., Mannaioni; M., Alesiani; V., Carla'; Natalini, Benedetto; Marinozzi, Maura; Pellicciari, Roberto; F., Moroni
MODULATION OF THE KYNURENINE PATHWAY IN SEARCH FOR NEW NEUROPROTECTIVE AGENTS - SYNTHESIS AND PRELIMINARY EVALUATION OF (M-NITROBENZOYL)ALANINE, A POTENT INHIBITOR OF KYNURENINE-3-HYDROXYLASE
1994 Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; M. R., Mahmoud; L., Mattoli; B. M., Sadeghpour; F., Moroni; A., Chiarugi; R., Carpenedo
AMINO-ACID DERIVATIVES OF 5-ASA AS NOVEL PRODRUGS FOR INTESTINAL DRUG-DELIVERY
1994 C., Clerici; G., Gentili; M. A., Pelli; E., Boschetti; C., Santucci; A., Garzon Aburbeh; Natalini, Benedetto; Pellicciari, Roberto; A., Morelli
Amino acid derivateves of 5-ASA as novel prodrugs for intestinal drug delivery
1994 Clerici, C.; Gentili, G.; Boschetti, Enrico; Santucci, G.; Aburbeh, A. G.; Natalini, Benedetto; Pellicciari, R.; Morelli, A.
SYNTHESIS OF 2-AZABICYCLO[3.1.0]HEXANE TRICARBOXYLATE AND ITS TRANSFORMATION INTO A NEW PROLINE-GAMMA-ACETIC ACID EQUIVALENT
1994 L., Arenare; P., De Caprariis; Marinozzi, Maura; Natalini, Benedetto; Pellicciari, Roberto
SYNTHESIS AND ACTIVITY OF ENANTIOPURE (S)(M-NITROBENZOYL) ALANINE, POTENT KYNURENINE-3-HYDROXYLASE INHIBITOR
1995 Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto; R., Carpenedo; A., Chiarugi; F., Moroni
SYNTHESIS AND BIOLOGICAL EVALUATION OF 6-CARBOXY-3,4-METHANOPROLINES, NEW RIGID GLUTAMATE ANALOGS
1995 Marinozzi, Maura; Natalini, Benedetto; M. H., Ni; Costantino, Gabriele; Pellicciari, Roberto; C., Thomsen
Synthesis of All Four Diastereomers of 4-Carboxymethyl-proline, a Conformationally Constrained Analog of 2-Amino Adipic Acid
1995 Pellicciari, Roberto; L., Arenare; P., De Caprariis; Natalini, Benedetto; Marinozzi, Maura; A., Galli
METABOLISM, PHARMACOKINETICS, AND ACTIVITY OF A NEW 6-FLUORO ANALOG OF URSODEOXYCHOLIC ACID IN RATS AND HAMSTERS
1995 A., Roda; Pellicciari, Roberto; C., Polimeni; C., Cerré; G., Cantelli Forti; B., Sadeghpour; E., Sapigni; A. M., Gioacchini; Natalini, Benedetto
1-AMINOINDAN-1,5-DICARBOXYLIC ACID - A NOVEL ANTAGONIST AT PHOSPHOLIPASE C-LINKED METABOTROPIC GLUTAMATE RECEPTORS
1995 Pellicciari, Roberto; R., Luneia; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; P., Jakobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen
The Pseudoactive Site as a Tool for Indirect Drug Design. Application to Inhibitors of Kynurenine-3-hydroxylase
1995 Costantino, Gabriele; Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto
S-(+)-2-(3'carboxy-bicyclo[1.1.1]pentyl)glycine, a structurally new group I metabotropic glutamate receptor antagonist
1996 Pellicciari, Roberto; Raimondo, M. R.; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Thomsen, C.
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-Phenylcarboxycyclopropylglycine (PCCG-4): a Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors
1996 Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; P., Tijskens; C., Thomsen; Pellicciari, Roberto
Conformationally constrained tryptophan analogs. Synthesis of (+/-)-(Z)- and (+/-)-(E)-2-amino-2,3-methano-3-(indol-3-yl)-propanoic acids
1996 D., Donati; A., Garzon Aburbeh; Natalini, Benedetto; C., Marchioro; Pellicciari, Roberto
The reaction of alpha-diazo-beta-hydroxy esters with boron trifluoride etherate: Generation and rearrangement of destabilized vinyl cations. A detailed experimental and theoretical study
1996 Pellicciari, Roberto; Natalini, Benedetto; B. M., Sadeghpour; Marinozzi, Maura; J. P., Snyder; B. L., Williamson; J. T., Kuethe; A., Padwa
Synthesis and receptor binding affinity of cholecystokinin receptor ligands: 2- and 1-indolyl derivatives of PD134308
1996 G., Araldi; D., Donati; B., Oliosi; A., Ursini; F., Vanamsterdam; Natalini, Benedetto; Pellicciari, Roberto; G., Tarzia
Synthesis of 6,6-dicarboxy-3,4-methano-L-proline, a new constrained glutamate analog endowed with neuroprotective properties
1996 Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Pellicciari, Roberto; V., Bruno; F., Nicoletti
Kynurenine-3-hydroxylase and its selective inhibitors. Molecular modeling studies.
1996 Costantino, Gabriele; L., Mattoli; F., Moroni; Natalini, Benedetto; Pellicciari, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Definition of a pharmacophore for the metabotropic glutamate receptors negatively linked to adenylyl cyclase | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto; F., Moroni; G., Lombardi | |
Conformational requirements for interaction of L-glutamate with the metabotropic EAA receptor | 1993 | Costantino, Gabriele; Natalini, Benedetto; Pellicciari, Roberto | |
SULFATE ESTERS OF HYDROXY AMINO-ACIDS AS STEREOSPECIFIC GLUTAMATE-RECEPTOR AGONISTS | 1994 | G., Mannaioni; M., Alesiani; V., Carla'; Natalini, Benedetto; Marinozzi, Maura; Pellicciari, Roberto; F., Moroni | |
MODULATION OF THE KYNURENINE PATHWAY IN SEARCH FOR NEW NEUROPROTECTIVE AGENTS - SYNTHESIS AND PRELIMINARY EVALUATION OF (M-NITROBENZOYL)ALANINE, A POTENT INHIBITOR OF KYNURENINE-3-HYDROXYLASE | 1994 | Pellicciari, Roberto; Natalini, Benedetto; Costantino, Gabriele; M. R., Mahmoud; L., Mattoli; B. M., Sadeghpour; F., Moroni; A., Chiarugi; R., Carpenedo | |
AMINO-ACID DERIVATIVES OF 5-ASA AS NOVEL PRODRUGS FOR INTESTINAL DRUG-DELIVERY | 1994 | C., Clerici; G., Gentili; M. A., Pelli; E., Boschetti; C., Santucci; A., Garzon Aburbeh; Natalini, Benedetto; Pellicciari, Roberto; A., Morelli | |
Amino acid derivateves of 5-ASA as novel prodrugs for intestinal drug delivery | 1994 | Clerici, C.; Gentili, G.; Boschetti, Enrico; Santucci, G.; Aburbeh, A. G.; Natalini, Benedetto; Pellicciari, R.; Morelli, A. | |
SYNTHESIS OF 2-AZABICYCLO[3.1.0]HEXANE TRICARBOXYLATE AND ITS TRANSFORMATION INTO A NEW PROLINE-GAMMA-ACETIC ACID EQUIVALENT | 1994 | L., Arenare; P., De Caprariis; Marinozzi, Maura; Natalini, Benedetto; Pellicciari, Roberto | |
SYNTHESIS AND ACTIVITY OF ENANTIOPURE (S)(M-NITROBENZOYL) ALANINE, POTENT KYNURENINE-3-HYDROXYLASE INHIBITOR | 1995 | Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto; R., Carpenedo; A., Chiarugi; F., Moroni | |
SYNTHESIS AND BIOLOGICAL EVALUATION OF 6-CARBOXY-3,4-METHANOPROLINES, NEW RIGID GLUTAMATE ANALOGS | 1995 | Marinozzi, Maura; Natalini, Benedetto; M. H., Ni; Costantino, Gabriele; Pellicciari, Roberto; C., Thomsen | |
Synthesis of All Four Diastereomers of 4-Carboxymethyl-proline, a Conformationally Constrained Analog of 2-Amino Adipic Acid | 1995 | Pellicciari, Roberto; L., Arenare; P., De Caprariis; Natalini, Benedetto; Marinozzi, Maura; A., Galli | |
METABOLISM, PHARMACOKINETICS, AND ACTIVITY OF A NEW 6-FLUORO ANALOG OF URSODEOXYCHOLIC ACID IN RATS AND HAMSTERS | 1995 | A., Roda; Pellicciari, Roberto; C., Polimeni; C., Cerré; G., Cantelli Forti; B., Sadeghpour; E., Sapigni; A. M., Gioacchini; Natalini, Benedetto | |
1-AMINOINDAN-1,5-DICARBOXYLIC ACID - A NOVEL ANTAGONIST AT PHOSPHOLIPASE C-LINKED METABOTROPIC GLUTAMATE RECEPTORS | 1995 | Pellicciari, Roberto; R., Luneia; Costantino, Gabriele; Marinozzi, Maura; Natalini, Benedetto; P., Jakobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen | |
The Pseudoactive Site as a Tool for Indirect Drug Design. Application to Inhibitors of Kynurenine-3-hydroxylase | 1995 | Costantino, Gabriele; Natalini, Benedetto; L., Mattoli; Pellicciari, Roberto | |
S-(+)-2-(3'carboxy-bicyclo[1.1.1]pentyl)glycine, a structurally new group I metabotropic glutamate receptor antagonist | 1996 | Pellicciari, Roberto; Raimondo, M. R.; Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Thomsen, C. | |
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-Phenylcarboxycyclopropylglycine (PCCG-4): a Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors | 1996 | Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; P., Tijskens; C., Thomsen; Pellicciari, Roberto | |
Conformationally constrained tryptophan analogs. Synthesis of (+/-)-(Z)- and (+/-)-(E)-2-amino-2,3-methano-3-(indol-3-yl)-propanoic acids | 1996 | D., Donati; A., Garzon Aburbeh; Natalini, Benedetto; C., Marchioro; Pellicciari, Roberto | |
The reaction of alpha-diazo-beta-hydroxy esters with boron trifluoride etherate: Generation and rearrangement of destabilized vinyl cations. A detailed experimental and theoretical study | 1996 | Pellicciari, Roberto; Natalini, Benedetto; B. M., Sadeghpour; Marinozzi, Maura; J. P., Snyder; B. L., Williamson; J. T., Kuethe; A., Padwa | |
Synthesis and receptor binding affinity of cholecystokinin receptor ligands: 2- and 1-indolyl derivatives of PD134308 | 1996 | G., Araldi; D., Donati; B., Oliosi; A., Ursini; F., Vanamsterdam; Natalini, Benedetto; Pellicciari, Roberto; G., Tarzia | |
Synthesis of 6,6-dicarboxy-3,4-methano-L-proline, a new constrained glutamate analog endowed with neuroprotective properties | 1996 | Marinozzi, Maura; Natalini, Benedetto; Costantino, Gabriele; Pellicciari, Roberto; V., Bruno; F., Nicoletti | |
Kynurenine-3-hydroxylase and its selective inhibitors. Molecular modeling studies. | 1996 | Costantino, Gabriele; L., Mattoli; F., Moroni; Natalini, Benedetto; Pellicciari, Roberto |
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