MASSARI, SERENA
MASSARI, SERENA
DIPARTIMENTO DI SCIENZE FARMACEUTICHE
1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors
2021-01-01 Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S.
1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity
2020-01-01 Desantis, J.; Massari, S.; Corona, A.; Astolfi, A.; Sabatini, S.; Manfroni, G.; Palazzotti, D.; Cecchetti, V.; Pannecouque, C.; Tramontano, E.; Tabarrini, O.
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions
2013-01-01 Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities
2013-01-01 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors
2018-01-01 Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
2018-01-01 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction.
2009-01-01 Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta
4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10
2018-01-01 Murthy, S; Desantis, J; Verheugd, P; Maksimainen, Mm; Venkannagari, H; Massari, S; Ashok, Y; Obaji, E; Nkizinkinko, Y; Lüscher, B; Tabarrini, O; Lehtiö, L
6-Aminoquinolones targeting HCV NS5B polymerase.
2012-01-01 Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta
6-Desfluoroquinolones as HIV-1 Tat-mediated Transcription Inhibitors
2010-01-01 Tabarrini, Oriana; Massari, Serena; Cecchetti, Violetta
6-Desfluoroquinolones as promising HIV transcription inhibitors
2007-01-01 Tabarrini, Oriana; Cecchetti, Violetta; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Stevens, M.; Daelemans, D.; Pannecouque, C.
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis
2012-01-01 Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Scott G., Franzblau; Cecchetti, Violetta
A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication.
2010-01-01 Massari, Serena; D., Daelemans; Barreca, MARIA LETIZIA; A., Knezevich; Sabatini, Stefano; Cecchetti, Violetta; A., Marcello; C., Pannecouque; Tabarrini, Oriana
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction
2015-01-01 Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana
A New Derivative with Ultra-Potent Anti-HIV Activity
2008-01-01 Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta; Daelemans, D; Pannecouque, C.
A new quinolone derivative with ultra-potent anti-HIV activity.
2008-01-01 Massari, Serena; Tabarrini, O; Manfroni, Giuseppe; V., Cecchetti; D., Daelemans; C., Pannecouque
Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency
2017-01-01 Tabarrini, O.; Massari, S.
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors
2020-01-01 Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O.
Biotinylated Tryptophan Catabolites for Target Fishing.
2012-01-01 Tabarrini, Oriana; Massari, Serena; Sabatini, Stefano; Fallarino, Francesca; Vacca, Carmine; Grohmann, Ursula
Blocking HIV-1 Replication by Targeting the TAT-Hijacked Transcriptional Machinery
2013-01-01 Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors | 1-gen-2021 | Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S. | |
1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity | 1-gen-2020 | Desantis, J.; Massari, S.; Corona, A.; Astolfi, A.; Sabatini, S.; Manfroni, G.; Palazzotti, D.; Cecchetti, V.; Pannecouque, C.; Tramontano, E.; Tabarrini, O. | |
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions | 1-gen-2013 | Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta | |
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities | 1-gen-2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors | 1-gen-2018 | Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari | |
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction | 1-gen-2018 | Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano | |
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction. | 1-gen-2009 | Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta | |
4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10 | 1-gen-2018 | Murthy, S; Desantis, J; Verheugd, P; Maksimainen, Mm; Venkannagari, H; Massari, S; Ashok, Y; Obaji, E; Nkizinkinko, Y; Lüscher, B; Tabarrini, O; Lehtiö, L | |
6-Aminoquinolones targeting HCV NS5B polymerase. | 1-gen-2012 | Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta | |
6-Desfluoroquinolones as HIV-1 Tat-mediated Transcription Inhibitors | 1-gen-2010 | Tabarrini, Oriana; Massari, Serena; Cecchetti, Violetta | |
6-Desfluoroquinolones as promising HIV transcription inhibitors | 1-gen-2007 | Tabarrini, Oriana; Cecchetti, Violetta; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Stevens, M.; Daelemans, D.; Pannecouque, C. | |
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis | 1-gen-2012 | Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Scott G., Franzblau; Cecchetti, Violetta | |
A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication. | 1-gen-2010 | Massari, Serena; D., Daelemans; Barreca, MARIA LETIZIA; A., Knezevich; Sabatini, Stefano; Cecchetti, Violetta; A., Marcello; C., Pannecouque; Tabarrini, Oriana | |
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction | 1-gen-2015 | Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana | |
A New Derivative with Ultra-Potent Anti-HIV Activity | 1-gen-2008 | Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta; Daelemans, D; Pannecouque, C. | |
A new quinolone derivative with ultra-potent anti-HIV activity. | 1-gen-2008 | Massari, Serena; Tabarrini, O; Manfroni, Giuseppe; V., Cecchetti; D., Daelemans; C., Pannecouque | |
Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency | 1-gen-2017 | Tabarrini, O.; Massari, S. | |
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors | 1-gen-2020 | Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O. | |
Biotinylated Tryptophan Catabolites for Target Fishing. | 1-gen-2012 | Tabarrini, Oriana; Massari, Serena; Sabatini, Stefano; Fallarino, Francesca; Vacca, Carmine; Grohmann, Ursula | |
Blocking HIV-1 Replication by Targeting the TAT-Hijacked Transcriptional Machinery | 1-gen-2013 | Massari, Serena; Sabatini, Stefano; Tabarrini, Oriana |