MASSARI, SERENA
MASSARI, SERENA
DIPARTIMENTO DI SCIENZE FARMACEUTICHE
1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors
2021 Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S.
1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity
2020 Desantis, J.; Massari, S.; Corona, A.; Astolfi, A.; Sabatini, S.; Manfroni, G.; Palazzotti, D.; Cecchetti, V.; Pannecouque, C.; Tramontano, E.; Tabarrini, O.
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions
2013 Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities
2013 Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana
2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors
2018 Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
2018 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction.
2009 Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta
4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10
2018 Murthy, S; Desantis, J; Verheugd, P; Maksimainen, Mm; Venkannagari, H; Massari, S; Ashok, Y; Obaji, E; Nkizinkinko, Y; Lüscher, B; Tabarrini, O; Lehtiö, L
6-Aminoquinolones targeting HCV NS5B polymerase.
2012 Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta
6-Desfluoroquinolones as HIV-1 Tat-mediated Transcription Inhibitors
2010 Tabarrini, Oriana; Massari, Serena; Cecchetti, Violetta
6-Desfluoroquinolones as promising HIV transcription inhibitors
2007 Tabarrini, Oriana; Cecchetti, Violetta; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Stevens, M.; Daelemans, D.; Pannecouque, C.
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis
2012 Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Scott G., Franzblau; Cecchetti, Violetta
[1,2,4]Triazolo[3,4-b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes
2023 Murthy, Sudarshan; Nizi, Maria Giulia; Maksimainen, Mirko M; Massari, Serena; Alaviuhkola, Juho; Lippok, Barbara E; Vagaggini, Chiara; Sowa, Sven T; Galera-Prat, Albert; Ashok, Yashwanth; Venkannagari, Harikanth; Prunskaite-Hyyryläinen, Renata; Dreassi, Elena; Lüscher, Bernhard; Korn, Patricia; Tabarrini, Oriana; Lehtiö, Lari
A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication.
2010 Massari, Serena; D., Daelemans; Barreca, MARIA LETIZIA; A., Knezevich; Sabatini, Stefano; Cecchetti, Violetta; A., Marcello; C., Pannecouque; Tabarrini, Oriana
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction
2015 Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana
A New Derivative with Ultra-Potent Anti-HIV Activity
2008 Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta; Daelemans, D; Pannecouque, C.
A new quinolone derivative with ultra-potent anti-HIV activity.
2008 Massari, Serena; Tabarrini, O; Manfroni, Giuseppe; V., Cecchetti; D., Daelemans; C., Pannecouque
Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency
2017 Tabarrini, O.; Massari, S.
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors
2020 Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O.
Biotinylated Tryptophan Catabolites for Target Fishing.
2012 Tabarrini, Oriana; Massari, Serena; Sabatini, Stefano; Fallarino, Francesca; Vacca, Carmine; Grohmann, Ursula
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,2,4-Triazolo[1,5-a]pyrimidines: Efficient One-step Synthesis and Functionalization as Influenza Polymerase PA-PB1 Interaction Disruptors | 2021 | Pismataro, M. C.; Felicetti, T.; Bertagnin, C.; Nizi, M. G.; Bonomini, A.; Barreca, M. L.; Cecchetti, V.; Jochmans, D.; De Jonghe, S.; Neyts, J.; Loregian, A.; Tabarrini, O.; Massari, S. | |
| 1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity | 2020 | Desantis, J.; Massari, S.; Corona, A.; Astolfi, A.; Sabatini, S.; Manfroni, G.; Palazzotti, D.; Cecchetti, V.; Pannecouque, C.; Tramontano, E.; Tabarrini, O. | |
| 1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions | 2013 | Alma, Martelli; Manfroni, Giuseppe; Sabbatini, Paola; Barreca, MARIA LETIZIA; Lara, Testai; Michela, Novelli; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Pellegrino, Masiello; Vincenzo, Calderone; Cecchetti, Violetta | |
| 2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities | 2013 | Sancineto, Luca; Iraci, Nunzio; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Cecchetti, Violetta; Tabarrini, Oriana | |
| 2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors | 2018 | Nkizinkiko, Yves; Desantis, Jenny; Koivunen, Jarkko; Teemu, Haikarainen; Murthy, Sudarshan; Sancineto, Luca; Massari, Serena; Ianni, Federica; Obaji, Ezeogo; Loza Maria, I; Pihlajaniemi, Taina; Brea, Jose; Tabarrini, Oriana; Lehtiö, Lari | |
| 2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction | 2018 | Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano | |
| 2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction. | 2009 | Gatto, B; Tabarrini, Oriana; Massari, Serena; Giaretta, G; Sabatini, Stefano; DEL VECCHIO, C; Parolin, C; Fravolini, Arnaldo; Palumbo, M; Cecchetti, Violetta | |
| 4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10 | 2018 | Murthy, S; Desantis, J; Verheugd, P; Maksimainen, Mm; Venkannagari, H; Massari, S; Ashok, Y; Obaji, E; Nkizinkinko, Y; Lüscher, B; Tabarrini, O; Lehtiö, L | |
| 6-Aminoquinolones targeting HCV NS5B polymerase. | 2012 | Cannaliere, R.; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Cecchetti, Violetta | |
| 6-Desfluoroquinolones as HIV-1 Tat-mediated Transcription Inhibitors | 2010 | Tabarrini, Oriana; Massari, Serena; Cecchetti, Violetta | |
| 6-Desfluoroquinolones as promising HIV transcription inhibitors | 2007 | Tabarrini, Oriana; Cecchetti, Violetta; Massari, Serena; Sabatini, Stefano; Manfroni, Giuseppe; Stevens, M.; Daelemans, D.; Pannecouque, C. | |
| 6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis | 2012 | Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Scott G., Franzblau; Cecchetti, Violetta | |
| [1,2,4]Triazolo[3,4-b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes | 2023 | Murthy, Sudarshan; Nizi, Maria Giulia; Maksimainen, Mirko M; Massari, Serena; Alaviuhkola, Juho; Lippok, Barbara E; Vagaggini, Chiara; Sowa, Sven T; Galera-Prat, Albert; Ashok, Yashwanth; Venkannagari, Harikanth; Prunskaite-Hyyryläinen, Renata; Dreassi, Elena; Lüscher, Bernhard; Korn, Patricia; Tabarrini, Oriana; Lehtiö, Lari | |
| A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication. | 2010 | Massari, Serena; D., Daelemans; Barreca, MARIA LETIZIA; A., Knezevich; Sabatini, Stefano; Cecchetti, Violetta; A., Marcello; C., Pannecouque; Tabarrini, Oriana | |
| A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction | 2015 | Massari, Serena; Nannetti, Giulio; Desantis, Jenny; Muratore, Giulia; Sabatini, Stefano; Manfroni, Giuseppe; Mercorelli, Beatrice; Cecchetti, Violetta; Palù, Giorgio; Cruciani, Gabriele; Loregian, Arianna; Goracci, Laura; Tabarrini, Oriana | |
| A New Derivative with Ultra-Potent Anti-HIV Activity | 2008 | Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Cecchetti, Violetta; Daelemans, D; Pannecouque, C. | |
| A new quinolone derivative with ultra-potent anti-HIV activity. | 2008 | Massari, Serena; Tabarrini, O; Manfroni, Giuseppe; V., Cecchetti; D., Daelemans; C., Pannecouque | |
| Acting on Tat-Mediated Transcription to Achieve a Long Term Control of HIV-1 Latency | 2017 | Tabarrini, O.; Massari, S. | |
| Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors | 2020 | Nizi, M. G.; Desantis, J.; Nakatani, Y.; Massari, S.; Mazzarella, M. A.; Shetye, G.; Sabatini, S.; Barreca, M. L.; Manfroni, G.; Felicetti, T.; Rushton-Green, R.; Hards, K.; Latacz, G.; Satala, G.; Bojarski, A. J.; Cecchetti, V.; Kolar, M. H.; Handzlik, J.; Cook, G. M.; Franzblau, S. G.; Tabarrini, O. | |
| Biotinylated Tryptophan Catabolites for Target Fishing. | 2012 | Tabarrini, Oriana; Massari, Serena; Sabatini, Stefano; Fallarino, Francesca; Vacca, Carmine; Grohmann, Ursula |