CANNALIRE, ROLANDO
CANNALIRE, ROLANDO
DIPARTIMENTO DI SCIENZE FARMACEUTICHE
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
2018 Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano
A Journey around the Medicinal Chemistry of Hepatitis C Virus Inhibitors Targeting NS4B: From Target to Preclinical Drug Candidates
2016 Cannalire, Rolando; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Cecchetti, Violetta
Advantageous Use of Ionic Liquids for the Synthesis of Pharmaceutically Relevant Quinolones
2018 Cannalire, Rolando; Tiecco, Matteo; Cecchetti, Violetta; Germani, Raimondo; Manfroni, Giuseppe
An overview on small molecules acting as broad-spectrum agents for yellow fever infection
2022 Desantis, J.; Felicetti, T.; Cannalire, R.
Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium
2015 Machado, Diana; Cannalire, Rolando; Santos Costa, Sofia; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions
2019 Cannalire, R.; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G.
Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View
2020 Felicetti, T.; Manfroni, G.; Cecchetti, V.; Cannalire, R.
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors
2020 Felicetti, T.; Mangiaterra, G.; Cannalire, R.; Cedraro, N.; Pietrella, D.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Biavasco, F.; Sabatini, S.
Design and synthesis of WM5 analogues as HIV-1 TAR RNA binders.
2019 Desantis, J.; Massari, S.; Sosic, A.; Manfroni, G.; Cannalire, R.; Felicetti, T.; Pannecouque, P.; Gatto, B.; Tabarrini, O.
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation
2019 Astolfi, A.; Kudolo, M.; Brea, J.; Manni, G.; Manfroni, G.; Palazzotti, D.; Sabatini, S.; Cecchetti, F.; Felicetti, T.; Cannalire, R.; Massari, S.; Tabarrini, O.; Loza, M. I.; Fallarino, F.; Cecchetti, V.; Laufer, S. A.; Barreca, M. L.
Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi
2021 Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio
Evolution of HCV NS4B Inhibitors
2019 Manfroni, G.; Cannalire, R.
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
2021 Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano
Functionalized 2,1-benzothiazine 2,2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase
2018 Cannalire, Rolando; Tarantino, Delia; Astolfi, Andrea; Barreca, MARIA LETIZIA; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Milani, Mario; Querat, Gilles; Mastrangelo, Eloise; Manfroni, Giuseppe; Cecchetti, Violetta
Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli
2017 Machado, Diana; Fernandes, Laura; Costa, Sofia S.; Cannalire, Rolando; Manfroni, Giuseppe; Tabarrini, Oriana; Couto, Isabel; Sabatini, Stefano; Viveiros, Miguel
Modifications on C6 and C7 Positions of 3-Phenylquinolone Efflux Pump Inhibitors Led to Potent and Safe Antimycobacterial Treatment Adjuvants
2019 Felicetti, T.; Machado, D.; Cannalire, R.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Viveiros, M.; Sabatini, S.
Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium
2017 Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta
New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors
2014 Manfroni, Giuseppe; Manvar, Dinesh; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta
Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 Polymerase
2020 Cannalire, R.; Ki Chan, K. W.; Burali, M. S.; Gwee, C. P.; Wang, S.; Astolfi, A.; Massari, S.; Sabatini, S.; Tabarrini, O.; Mastrangelo, E.; Barreca, M. L.; Cecchetti, V.; Vasudevan, S. G.; Manfroni, G.
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues
2017 Felicetti, Tommaso; Cannalire, Rolando; Burali, MARIA SOLE; Massari, Serena; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Tabarrini, Oriana; Schindler, Bryan D; Sabatini, Stefano; Kaatz, Glenn W; Cecchetti, Violetta
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction | 2018 | Felicetti, Tommaso; Cannalire, Rolando; Pietrella, Donatella; Latacz, Gniewomir; Lubelska, Annamaria; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Massari, Serena; Tabarrini, Oriana; Kieć-Kononowicz, Katarzyna; Schindler, Bryan D.; Kaatz, Glenn W.; Cecchetti, Violetta; Sabatini, Stefano | |
| A Journey around the Medicinal Chemistry of Hepatitis C Virus Inhibitors Targeting NS4B: From Target to Preclinical Drug Candidates | 2016 | Cannalire, Rolando; Barreca, MARIA LETIZIA; Manfroni, Giuseppe; Cecchetti, Violetta | |
| Advantageous Use of Ionic Liquids for the Synthesis of Pharmaceutically Relevant Quinolones | 2018 | Cannalire, Rolando; Tiecco, Matteo; Cecchetti, Violetta; Germani, Raimondo; Manfroni, Giuseppe | |
| An overview on small molecules acting as broad-spectrum agents for yellow fever infection | 2022 | Desantis, J.; Felicetti, T.; Cannalire, R. | |
| Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium | 2015 | Machado, Diana; Cannalire, Rolando; Santos Costa, Sofia; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano | |
| Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions | 2019 | Cannalire, R.; Tarantino, D.; Piorkowski, G.; Carletti, T.; Massari, S.; Felicetti, T.; Barreca, M. L.; Sabatini, S.; Tabarrini, O.; Marcello, A.; Milani, M.; Cecchetti, V.; Mastrangelo, E.; Manfroni, G.; Querat, G. | |
| Broad-Spectrum Flavivirus Inhibitors: a Medicinal Chemistry Point of View | 2020 | Felicetti, T.; Manfroni, G.; Cecchetti, V.; Cannalire, R. | |
| C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors | 2020 | Felicetti, T.; Mangiaterra, G.; Cannalire, R.; Cedraro, N.; Pietrella, D.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Biavasco, F.; Sabatini, S. | |
| Design and synthesis of WM5 analogues as HIV-1 TAR RNA binders. | 2019 | Desantis, J.; Massari, S.; Sosic, A.; Manfroni, G.; Cannalire, R.; Felicetti, T.; Pannecouque, P.; Gatto, B.; Tabarrini, O. | |
| Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation | 2019 | Astolfi, A.; Kudolo, M.; Brea, J.; Manni, G.; Manfroni, G.; Palazzotti, D.; Sabatini, S.; Cecchetti, F.; Felicetti, T.; Cannalire, R.; Massari, S.; Tabarrini, O.; Loza, M. I.; Fallarino, F.; Cecchetti, V.; Laufer, S. A.; Barreca, M. L. | |
| Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi | 2021 | Rampacci, Elisa; Marenzoni, Maria Luisa; Cannalire, Rolando; Pietrella, Donatella; Sabatini, Stefano; Giovagnoli, Stefano; Felicetti, Tommaso; Pepe, Marco; Passamonti, Fabrizio | |
| Evolution of HCV NS4B Inhibitors | 2019 | Manfroni, G.; Cannalire, R. | |
| From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search | 2021 | Cedraro, Nicholas; Cannalire, Rolando; Astolfi, Andrea; Mangiaterra, Gianmarco; Felicetti, Tommaso; Vaiasicca, Salvatore; Cernicchi, Giada; Massari, Serena; Manfroni, Giuseppe; Tabarrini, Oriana; Cecchetti, Violetta; Barreca, Maria Letizia; Biavasco, Francesca; Sabatini, Stefano | |
| Functionalized 2,1-benzothiazine 2,2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase | 2018 | Cannalire, Rolando; Tarantino, Delia; Astolfi, Andrea; Barreca, MARIA LETIZIA; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Milani, Mario; Querat, Gilles; Mastrangelo, Eloise; Manfroni, Giuseppe; Cecchetti, Violetta | |
| Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli | 2017 | Machado, Diana; Fernandes, Laura; Costa, Sofia S.; Cannalire, Rolando; Manfroni, Giuseppe; Tabarrini, Oriana; Couto, Isabel; Sabatini, Stefano; Viveiros, Miguel | |
| Modifications on C6 and C7 Positions of 3-Phenylquinolone Efflux Pump Inhibitors Led to Potent and Safe Antimycobacterial Treatment Adjuvants | 2019 | Felicetti, T.; Machado, D.; Cannalire, R.; Astolfi, A.; Massari, S.; Tabarrini, O.; Manfroni, G.; Barreca, M. L.; Cecchetti, V.; Viveiros, M.; Sabatini, S. | |
| Natural isoflavone biochanin A as a template for the design of new and potent 3-phenylquinolone efflux inhibitors against Mycobacterium avium | 2017 | Cannalire, Rolando; Machado, Diana; Felicetti, Tommaso; Santos Costa, Sofia; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Couto, Isabel; Viveiros, Miguel; Sabatini, Stefano; Cecchetti, Violetta | |
| New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors | 2014 | Manfroni, Giuseppe; Manvar, Dinesh; Barreca, MARIA LETIZIA; Kaushik Basu, Neerja; Leyssen, Pieter; Paeshuyse, Jan; Cannalire, Rolando; Iraci, Nunzio; Basu, Amartya; Chudaev, Maxim; Zamperini, Claudio; Dreassi, Elena; Sabatini, Stefano; Tabarrini, Oriana; Neyts, Johan; Cecchetti, Violetta | |
| Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 Polymerase | 2020 | Cannalire, R.; Ki Chan, K. W.; Burali, M. S.; Gwee, C. P.; Wang, S.; Astolfi, A.; Massari, S.; Sabatini, S.; Tabarrini, O.; Mastrangelo, E.; Barreca, M. L.; Cecchetti, V.; Vasudevan, S. G.; Manfroni, G. | |
| Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues | 2017 | Felicetti, Tommaso; Cannalire, Rolando; Burali, MARIA SOLE; Massari, Serena; Manfroni, Giuseppe; Barreca, MARIA LETIZIA; Tabarrini, Oriana; Schindler, Bryan D; Sabatini, Stefano; Kaatz, Glenn W; Cecchetti, Violetta |