FRAVOLINI, Arnaldo
 Distribuzione geografica
Continente #
NA - Nord America 2.987
AS - Asia 2.319
EU - Europa 2.178
SA - Sud America 303
AF - Africa 52
OC - Oceania 1
Totale 7.840
Nazione #
US - Stati Uniti d'America 2.926
SG - Singapore 952
UA - Ucraina 521
CN - Cina 358
IE - Irlanda 346
VN - Vietnam 322
SE - Svezia 316
HK - Hong Kong 289
RU - Federazione Russa 274
BR - Brasile 244
IT - Italia 152
DE - Germania 149
FI - Finlandia 103
KR - Corea 98
FR - Francia 86
GB - Regno Unito 77
TR - Turchia 54
IN - India 50
BE - Belgio 42
JP - Giappone 39
BD - Bangladesh 31
PL - Polonia 30
CA - Canada 27
IQ - Iraq 23
AR - Argentina 22
MX - Messico 22
ZA - Sudafrica 18
CH - Svizzera 13
UZ - Uzbekistan 13
NL - Olanda 12
PK - Pakistan 12
CZ - Repubblica Ceca 11
SA - Arabia Saudita 11
AT - Austria 10
EC - Ecuador 10
ID - Indonesia 9
PH - Filippine 9
ES - Italia 8
MY - Malesia 8
IL - Israele 7
RO - Romania 7
AE - Emirati Arabi Uniti 6
CO - Colombia 6
EG - Egitto 6
KG - Kirghizistan 6
KE - Kenya 5
LT - Lituania 5
VE - Venezuela 5
CI - Costa d'Avorio 4
CL - Cile 4
LB - Libano 4
MA - Marocco 4
PE - Perù 4
PY - Paraguay 4
AL - Albania 3
NP - Nepal 3
PA - Panama 3
PT - Portogallo 3
TN - Tunisia 3
BO - Bolivia 2
BW - Botswana 2
DK - Danimarca 2
DZ - Algeria 2
HN - Honduras 2
JM - Giamaica 2
JO - Giordania 2
LY - Libia 2
NI - Nicaragua 2
QA - Qatar 2
SN - Senegal 2
SV - El Salvador 2
TM - Turkmenistan 2
AM - Armenia 1
AO - Angola 1
AU - Australia 1
BA - Bosnia-Erzegovina 1
BG - Bulgaria 1
BH - Bahrain 1
CY - Cipro 1
EE - Estonia 1
ET - Etiopia 1
GA - Gabon 1
GR - Grecia 1
KZ - Kazakistan 1
LA - Repubblica Popolare Democratica del Laos 1
LK - Sri Lanka 1
LV - Lettonia 1
MM - Myanmar 1
NE - Niger 1
NO - Norvegia 1
OM - Oman 1
RS - Serbia 1
SK - Slovacchia (Repubblica Slovacca) 1
SR - Suriname 1
SY - Repubblica araba siriana 1
TT - Trinidad e Tobago 1
UY - Uruguay 1
Totale 7.840
Città #
Singapore 692
Chandler 386
Dublin 346
Jacksonville 289
Hong Kong 284
San Jose 253
Dong Ket 217
San Mateo 195
Ashburn 177
Boardman 114
Ann Arbor 101
Santa Clara 99
Seoul 97
Beijing 81
Medford 80
Princeton 79
Moscow 78
Lauterbourg 67
Wilmington 62
Andover 61
The Dalles 57
Altamura 52
Los Angeles 50
Lawrence 48
Munich 45
Brussels 42
Piscataway 39
Ho Chi Minh City 38
Tokyo 38
Nanjing 37
New York 32
Izmir 28
Des Moines 26
Hanoi 25
Perugia 24
Woodbridge 24
Saint Petersburg 22
São Paulo 22
Dallas 21
West Jordan 20
Warsaw 19
Brooklyn 17
Orem 15
San Paolo di Civitate 15
Fremont 14
Turku 14
Chongqing 12
London 12
San Diego 12
Atlanta 11
Baghdad 11
Chennai 11
Auburn Hills 10
Dhaka 10
Helsinki 10
Norwalk 10
Rio de Janeiro 10
Denver 9
Chicago 8
Columbus 8
Johannesburg 8
Montreal 8
Mumbai 8
Philadelphia 8
Poplar 8
Stockholm 8
Barnet 7
Boston 7
Brno 7
Charlotte 7
Guadalupe 7
Porto Alegre 7
Salvador 7
Seattle 7
Shanghai 7
Guayaquil 6
Hefei 6
Houston 6
Mexico City 6
Tashkent 6
Timisoara 6
Belo Horizonte 5
Bishkek 5
Da Nang 5
Haiphong 5
Hanover 5
Ottawa 5
Secaucus 5
Toronto 5
Abidjan 4
Aracaju 4
Cape Town 4
Curitiba 4
Istanbul 4
Mcallen 4
Medellín 4
Querétaro 4
Rome 4
San Francisco 4
Amsterdam 3
Totale 4.916
Nome #
1,4-Benzothiazine-2-carboxylic Acids 1-Oxide as Analogue of Antibacterial Quinolones 339
(1,4-Benzothiazinyloxy)alkylpiperazine Derivatives as Potential Antihypertensive Agents 315
6-Aminoquinolones, their Synthesis and their Use as Antibacterial Agents. 251
4H-1,4-Benzothiopyran-4-one-3-carboxylic Acids and 3,4-Dihydro-2H-isothiazolo[5,4-b][1]benzothiopyran-3,4-diones as Quinolone Antibacterial Analogs 162
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction. 143
6-Aminoquinolones: a New Class of Quinolone Antibacterials? 143
Attivatori dei canali K-ATP a struttura 1,4-benzotiazinica: modificazioni in C-2 e C-6 141
Chemometric Methodologies in a Quantitative Structure-Activity Relationship Study: the Antibacterial Activity of 6-Aminoquinolones 138
Derivati 2-fenilchinolonici come inibitori della pompa di efflusso NorA dello Staphylococcus aureus ciprofloxacin resistente 136
Chemometric Rationalization of the Structural and Physicochemical Basis for Selective Cyclooxygenase-2 Inhibition: Toward More Specific Ligands 134
8-Methyl-7-substituted-1,6-naphthyridine-3-carboxylic Acids as New 6-Desfluoroquinolone Antibacterials 134
2-phenylquinolones as HIV-1 Tat/TAR interaction inhibitors 133
Syhtesis and Biological Evaluation of 2-Phenylquinolones Targeted at Tat/TAR Recognition 128
6-Aminoquinolones as New Potential Anti-HIV Agents 126
7-(Disubstituted thiazolyl)-3,5-dihydroxy-6-heptenoic/heptanoic acid derivatives as HMG-COa reductase inhibitors 124
Structure-activity relationship study on anti-HIV 6-desfluoroquinolones. 123
Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones 123
6-Aminoquinolones: photostability, cellular distribution and phototoxicity. 120
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus. 120
Process for the Preparation of 9-Fluoro-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic Acid Hydrochloride 118
Chemometric rationalization of the structural features affecting the antibacterial activity of quinolones 116
Cell-dependent Interference with viral transactivation by 6-aminoquinolone derivatives. 115
Inhibition of Subgenomic Hepatitis C Virus RNA Replication by Acridone Derivatives: Identification of an NS3 Helicase Inhibitor. 113
Enantiomers of 8-(3-tert-Butylamino-2-hydroxypropoxy)-3,4-dihydro-3-oxo-2H-(1,4)benzothiazine: Racemic Resolution, Chiral Synthesis and Biological Activity. 113
From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps. 110
6-Hydroxy Derivative as New Desfluoroquinolone (DFQ): Synthesis and DNA-binding Study 109
New Heterocyclic Ring Systems. XIII.7,11-Dithiaazasteroid Analogues 107
Highly Potent 1,4-Benzothiazine Derivatives as KATP-Channel Openers 106
Synthesis and Antibacterial Evaluation of [1,3]Benzothiazino[3,2-a]quinoline and [3,1]Benzothiazino[1,2-a]quinoline-6-carboxylic Acid Derivatives 105
The antibacterial activity of quinolones against E.coli: a chemometric study 105
Chemometric Rationalization of the Structural Features Affecting the Antibacterial Activity of Quinolones Against Staphylococcus aureus 100
Pyrazolobenzothiazines as potent TNF-alpha production inhibitors. 98
Antiviral 6-aminoquinolones: Molecolar basis for potency and selectivity. 96
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition 94
One-Pot Synthesis of Rufloxacin 94
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump 92
New Heterocyclic Ring Systems. XIV. 7,11-Dithiaoxasteroids analogues 88
Structure modifications of 6-aminoquinolones with potent anti-HIV activity 87
Predictive models for hERG potassium channel blockers 87
A pharmacophore hypothesis for P-glycoprotein substrate recognition using GRIND-based 3D-QSAR. 87
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump 86
Symbiotic approach to drug design: N-[(4-chloro-3-sulfamoylbenzamido)-ethyl]propanolamine derivatives as β-adrenergic blocking agents with diuretic activity 86
New 1,8-peri-Annelated Tricyclic Quinolone Antibacterials 85
Novel 1,4-Benzothiazine Derivatives as large conductance Ca2+-activated potassium channel activators 84
Quinoline Carboxylic Acids. 3. Synthesis and Antibacterial Evaluation of 2- Subsituted-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic Acids Related to Rufloxacin 82
Design and Synthesis of Modified Quinolones as Antitumoral Acridones 82
Cell-dependent interference of a series of new 6-aminoquinolone derivatives with viral (HIV/CMV) transactivation. 80
Derivati Chinolonici non Fluorurati e Loro Impiego come Agenti Antibatterici. 80
New 6-Aminoquinolones as Antiviral Agents. 79
Effects of Novel 6-Desfluoroquinolones and Classic Quinolones on Pentylentetrazole-Induced Seizures in Mice 78
Synthesis and Antibacterial Evaluation of 1,4-Thiazinoquinoline Carboxylic Acids 77
Composto antiipertensivo ad attivita' beta-bloccante e diuretica. 77
Synthesis and Evaluation of Benzothiazine Derivatives as Inhibitors of NorA Efflux Pump of Staphylococcus aureus 76
Quinolones as potential anti HIV-1 agents targeted at Tat/TAR recognition. Abstr. P62 76
Mg2+ - Mediate Binding of 6-Substituted Quinolones to DNA: Relevance to Biological Activity. 76
Highly potent KATP channel activators. 76
From phenothiazine to 3-phenyl-1,4-benzothiazine derivatives as inhibitors of the Staphylococcus aureus NorA multidrug efflux pump. 75
New Heterocyclic Ring Systems.XI. Azadithiasteroid Analogues 72
Effetto inibitorio di derivati acridonici sulla replicazione del virus dell'epatite C (HCV) 72
STUDIES ON 6-AMINOQUINOLONES: SYNTHESIS AND ANTIBACTERIAL EVALUATION OF 6-AMINO-8-METHYLQUINOLONES. 70
o-Chlorobenzenesulfonamidic derivatives of (aryloxy)propanolamines as .beta.-blocking/diuretic agents 70
Selective anti-BVDV acridones as new potential anti-HCV agents 70
Cell-dependent interference with viral transactivation by 6-aminoquinolone derivatives 70
Synthesis and β-adrenergic blocking activity of 1,4-benzothiazine oxime ethers 68
In Vitro Activity of MF 5137, a New Potent 6-aminoquinolone 66
In Vitro Phototoxic Properties of new 6-Desfluoro and 6-Fluoro-8-methylquinolones 66
Dibenzo[1,6]naphthyridindiones as Modified Quinolone Antibacterials 65
Novel In Vivo Model for the Study of Human Immunodeficiency Virus Type 1 Transcription Inhibitors: Evaluation of New 6-Desfluoroquinolone Derivatives 64
Quinolonecarboxylic Acids. 2. Synthesis and Antibacterial Evaluation of 7-Oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic Acids 63
Sintesi ed Attivita’ Farmacologica di Carbossiamidi di Pirazolo-1,2-benzotiazine e di Isossazolo-1,2-benzotiazine 62
Inhibition of cell growth and induction of apoptosis in human prostatecancer cell lines by 6-aminoquinolone WM13 62
Synthesis and Beta-Adrenergic Blocking Activity of Oxypropanolamines of 3,4-Dihydro-3-oxo-2H-1,4-benzothiazine 61
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents 61
SYNTHESIS AND ANTIINFLAMMATORY ANALGESIC ACTIVITIES OF N-HETEROCYCLIC CARBOXAMIDES OF THIOPYRANO-1,2-BENZOTHIAZINE 60
Studies on anti-HIV Quinolones 57
Synthesis and Activity of New Modified 1,4-Benzothiazine Derivatives as Inhibitors of the NorA Efflux Pump of Staphylococcus aureus 57
Structural modifications on anti-HIV quinolones 57
Potent 6-Desfluoro-8-methylquinolones as New Lead Compounds in Antibacterial Chemotherapy 57
New Anti-Human Immunodeficency Virus Type 1 6-Aminoquinolones: Mechanism of Action 54
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Totale 7.978
Categoria #
all - tutte 32.776
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 32.776


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021234 0 0 0 0 0 0 0 0 0 0 0 234
2021/2022785 24 149 23 59 55 3 11 236 5 14 101 105
2022/20231.189 93 193 19 103 99 130 2 56 440 7 36 11
2023/2024486 27 65 26 9 6 12 80 2 108 29 59 63
2024/20251.308 25 110 59 142 181 64 32 70 222 68 216 119
2025/20262.396 195 185 127 337 293 237 384 122 257 185 66 8
Totale 7.978