IRIS - Res&Arch Institutional Research Information System - Research & Archive

SABATINI, Stefano
 Distribuzione geografica
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Continente #
NA - Nord America 3.067
AS - Asia 2.857
EU - Europa 2.675
AF - Africa 9
OC - Oceania 8
SA - Sud America 6
Continente sconosciuto - Info sul continente non disponibili 2
Totale 8.624
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Nazione #
US - Stati Uniti d'America 3.066
CN - Cina 2.167
IT - Italia 618
IE - Irlanda 601
UA - Ucraina 482
SE - Svezia 356
HK - Hong Kong 331
VN - Vietnam 280
DE - Germania 151
FI - Finlandia 122
RU - Federazione Russa 110
BE - Belgio 67
GB - Regno Unito 52
FR - Francia 27
CH - Svizzera 22
TR - Turchia 21
RO - Romania 19
JP - Giappone 17
NL - Olanda 12
UZ - Uzbekistan 11
AT - Austria 10
PL - Polonia 9
AU - Australia 7
SG - Singapore 7
CZ - Repubblica Ceca 6
EG - Egitto 5
KR - Corea 5
LB - Libano 5
IR - Iran 4
PK - Pakistan 4
BG - Bulgaria 3
BR - Brasile 3
CI - Costa d'Avorio 3
CL - Cile 3
GR - Grecia 3
IN - India 3
DK - Danimarca 2
EU - Europa 2
PT - Portogallo 2
CA - Canada 1
HU - Ungheria 1
ID - Indonesia 1
IQ - Iraq 1
NZ - Nuova Zelanda 1
ZA - Sudafrica 1
Totale 8.624
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Città #
Guangzhou 2.072
Chandler 774
Dublin 601
Hong Kong 325
San Mateo 293
Dong Ket 276
Jacksonville 271
Perugia 259
Medford 133
Princeton 133
Ann Arbor 101
Wilmington 99
Altamura 91
Andover 79
Lawrence 70
Brussels 67
Beijing 64
Fremont 47
Redmond 46
Des Moines 38
Saint Petersburg 36
Dearborn 30
Boardman 29
Norwalk 24
Izmir 21
Falls Church 20
West Jordan 20
Spoleto 19
Ashburn 18
Los Angeles 18
Woodbridge 18
Rome 17
Helsinki 14
Moscow 14
Redwood City 14
San Diego 12
Tokyo 12
Den Haag 10
New York 10
San Paolo di Civitate 10
San Giustino 9
Bologna 7
Bucharest 7
Hanover 7
Houston 7
Melbourne 7
Seattle 6
Singapore 6
Frankfurt Am Main 5
Napoli 5
Shanghai 5
Arak 4
Auburn Hills 4
Fairfield 4
Hanoi 4
Lausanne 4
Philadelphia 4
Tappahannock 4
Timisoara 4
Urbino 4
Vienna 4
Abidjan 3
Cerro Maggiore 3
Chicago 3
Ferrara 3
Foligno 3
Kunming 3
Mit Ghamr 3
Parma 3
Seoul 3
Siena 3
Silver Spring 3
Simi Valley 3
Terni 3
Albinea 2
Anguillara Sabazia 2
Bastia 2
Boydton 2
Cairo 2
Cambridge 2
Campegine 2
Carrara 2
Chongqing 2
Dallas 2
Edinburgh 2
Gujranwala 2
Hangzhou 2
Jinan 2
Kagoya 2
Licata 2
London 2
Marano Ticino 2
Mazzano Romano 2
Mcallen 2
Milan 2
Nanjing 2
Pitesti 2
San Jose 2
Serra 2
Torino 2
Totale 6.407
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Nome #
Structural investigation of Small Molecules Targeting Influenza A Virus Polymerase 2.090
1,4-Benzothiazine ATP-Sensitive Potassium Channel Openers: Modifications at the C-2 and C-6 Positions 215
1,2,4-triazolo[1,5-α]pyrimidines as a novel class of inhibitors of the HIV-1 reverse transcriptase-αssociated ribonuclease h activity 178
Derivati benzotiazinici come inibitori della pompa estrudente MDR NorA dello Staphylococcus aureus 114
Sintesi di nuovi inibitori della pompa di efflusso NorA dello S. aureus: dalle 3-fenil-1,4-benzotiazine alle 2-fenilchinossaline 100
Efficient microwave assisted synthesis of metal-organic framework UiO-66: optimization and scale up 94
Attivatori dei canali K-ATP a struttura 1,4-benzotiazinica: modificazioni in C-2 e C-6 85
SINTESI DI NUOVI INIBITORI DELLA POMPA DI EFFLUSSO NorA DELLO S. aureus: DALLE 3-FENIL-1,4-BENZOTIAZINE ALLE 2-FENILCHINOLINE 85
Structure-activity relationship study on anti-HIV 6-desfluoroquinolones. 84
Syhtesis and Biological Evaluation of 2-Phenylquinolones Targeted at Tat/TAR Recognition 83
Targeting CDKs to inhibit the HIV-1 TAT-mediated transcription 74
A 1,8-Naphthyridone Derivative Targets the HIV-1 Tat-Mediated Transcription and Potently Inhibits the HIV-1 Replication. 72
Functionalized 2,1-benzothiazine 2,2-dioxides as new inhibitors of Dengue NS5 RNA-dependent RNA polymerase 71
CYCLOHEPTATHIOPHENE-3-CARBOXAMIDE DERIVATIVES AS INFLUENZA A VIRUS POLYMERASE INHIBITORS 69
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction 69
Studies on 6-Aminoquinolones: Synthesis and Antibacterial Evaluation of 6-Amino-8-ethyl- and 6-Amino-8-methoxyquinolones 68
Synthesis of 2-(Arylamino)ethanethiols via Lewis Acid catalyzed Aminolysis of 2,2-Dimethylthiirane as Precursors of the 1,4-Benzothiazine Nucleus 65
Investigation of targeted pyrrolizidine alkaloids in traditional Chinese medicines and selected herbal teas sourced in Ireland using LC-ESI-MS/MS 65
Accounting for target flexibility and water molecules by docking to ensembles of target structures: The HCV NS5B Palm Site I inhibitors case study. 65
Small Molecules as HIV-1 Tat-TAR Complex Inhibitors 64
Antitubercular polyhalogenated phenothiazines and phenoselenazine with reduced binding to CNS receptors 63
Studies on Anti-HIV Quinolones: New Insights on the C-6 Position 62
6-Desfluoroquinolones as promising HIV transcription inhibitors 62
2-Phenylquinolones as Inhibitors of the HIV-1 Tat/TAR Interaction. 62
From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors 62
Discovery of potent p38α MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation 62
The Pyrazolobenzothiazine Core as a New Chemotype of p38 Alpha Mitogen-Activated Protein Kinase Inhibitors 61
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors 61
A GRIND based pharmacophoric model for Factor Xa inhibitors 60
Alternate NF-κB-independent signaling reactivation of latent HIV-1 provirus 60
Pyridobenzothiazolones Exert Potent Anti-Dengue Activity by Hampering Multiple Functions of NS5 Polymerase 60
8-Methyl-7-substituted-1,6-naphthyridine-3-carboxylic Acids as New 6-Desfluoroquinolone Antibacterials 59
Structure-based insights into p38α MAPK: from crystal structures analysis to hit optimization 59
Deciphering the molecular recognition mechanism of multidrug resistance staphylococcus aureus nora efflux pump using a supervised molecular dynamics approach 59
Pyridobenzothiazole derivatives as new chemotype targeting the HCV NS5B polymerase 58
2-phenylquinolones as HIV-1 Tat/TAR interaction inhibitors 57
Evolution from a natural flavones nucleus to obtain 2-(4-Propoxyphenyl)quinoline derivatives as potent inhibitors of the S. aureus NorA efflux pump. 57
Disegno di nuovi chinoloni ad attività antitubercolare: dalla 3D-QSAR agli algoritmi evolutivi. 57
A new 6-aminoquinolone compound with anti-HCMV activity 56
S. aureus NorA efflux pump: the discovery of new potent inhibitors 56
A New Promising Class of pyrazolobenzothiazine inhibitors of S. aureus NorA Efflux Pump 56
Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position 56
Antiviral Activity of WC5, a new 6-aminoquinolone compound against Human Herpesviruses 55
Broad spectrum anti-flavivirus pyridobenzothiazolones leading to less infective virions 55
From 6-Aminoquinolone Antibacterials to 6-Amino-7-thiopyranopyridinylquinolone Ethyl Esters as Inhibitors of Staphylococcus aureus Multidrug Efflux Pumps. 54
Synthesis of Novel Inhibitors of the S. aureus Efflux pumps: from the 4-hydroxy-2-phenylquinolines to the 4-hydroxy-2-phenylquinazolines 54
A Broad Anti-influenza Hybrid Small Molecule that Potently Disrupts the Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Subunits Interaction 54
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors 54
Derivati 1,4-benzotiazinici come agenti anticonvulsivanti. 53
2-Phenylquinazolinone fragment imparts anti-CDKs and anti-HIV activities 53
p38 alpha MAPK and Type I Inhibitors: Binding Site Analysis and Use of Target Ensembles in Virtual Screening 53
Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a] pyrimidine derivatives 53
Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues 52
Impact of conventional/non-conventional extraction methods on the untargeted phenolic profile of Moringa oleifera leaves 52
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors 52
Disegno e sintesi di agenti anti-HIV a duplice attività 51
Discovery of Novel Inhibitors of the NorA Multidrug Transporter of Staphylococcus aureus. 51
RE-EVOLUTION OF THE 2-PHENYL-4-HYDROXYQUINOLINES: OPTIMIZATION OF A POTENT NEW CLASS OF S. AUREUS NorA EFFLUX PUMP INHIBITORS 51
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis 51
Structure modifications of 6-aminoquinolones with potent anti-HIV activity 50
Binding studies and GRIND/ALMOND-based 3D QSAR analysis of benzothiazine type K-ATP channel openers 50
Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorA 50
Pyrazolobenzothiazines as potent TNF-alpha production inhibitors. 50
6-desfluorochinoloni (6-DFQ): sintesi assistita da microonde di 6-amino-7-(4-oxopiridinil) e 6-amino-7-(benzo-4-oxopiridinil) chinoloni 49
Computer-Aided Identification of Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity 49
Synthesis and Characterization of 1,2,4-Triazolo[1,5-a]pyrimidine-2-carboxamide-based Compounds Targeting the PA-PB1 Interface of Influenza A Virus Polymerase. 49
New Pyrazolobenzothiazine Derivatives As Hepatitis C Virus NS5B Polymerase Palm Site I Inhibitors 47
Synthesis and Evaluation of Benzothiazine Derivatives as Inhibitors of NorA Efflux Pump of Staphylococcus aureus 46
Derivati 2-fenilchinolonici come inibitori della pompa di efflusso NorA dello Staphylococcus aureus ciprofloxacin resistente 46
Nuovi Tiopiranopiridinil Chinoloni 46
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump 46
Sintesi del 2,2-dimetil-2,3-diidro-4H-1,4-benzotiazine via 2,2-dimetiltiirano catalizzata da acidi di Lewis. 46
Sitesi one-pot di varie 1,4-benzotiazine tramite apertura regioselettiva del 2,2-dimetiltiirano catalizzata da Cu(II)triflato 46
From cromakalim to different structural classes of KATP channel openers 45
Novel 1,4-Benzothiazine Derivatives as Large Conductance Ca2+-Activated Potassium Channel Openers 45
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity 45
Biotinylated Tryptophan Catabolites for Target Fishing. 45
Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation 45
Design and Synthesis of Modified Quinolones as Antitumoral Acridones 44
Designed Multiple Ligands (DLMs) as innovative anti-HIV agents 44
Re-evolution of the 2-phenylquinolines: Ligand-Based Design, Synthesis, and Biological Evaluation of a Potent New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors to Combat Antimicrobial Resistance 44
Highly Potent 1,4-Benzothiazine Derivatives as KATP-Channel Openers 43
Highly potent KATP channel activators. 43
Ethidium bromide exposure unmasks an antibiotic efflux system in Rhodococcus equi 43
Structure-Based Discovery of Pyrazolobenzothiazine Derivatives As Inhibitors of Hepatitis C Virus Replication 43
Searching New HCV NS5B Polymerase Inhibithors 42
Novel N-benzyl-1,4-benzothiazine derivates as large conductance Ca2+-activated potassium channel activators 42
Studi di molecular modeling per il disegno di inibitori COX-2 selettivi. 42
Investigation on the effect of known potent S. aureus NorA efflux pump inhibitors on the staphylococcal biofilm formation 42
Novel 1,4-Benzothiazine Derivatives as large conductance Ca2+-activated potassium channel activators 41
New 6-Aminoquinolones as Antiviral Agents. 41
Cycloheptathiophene-3-carboxamide derivatives as influenza A virus polymerase inhibitors 41
Structural Modifications of 2-phenylquinoline Inhibitors of S. aureus MDR NorA efflux pump 40
Searching for innovative quinolone-like scaffolds: synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivatives 40
Mode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli 40
DERIVATI 2-FENIL-4-IDROSSI-CHINOLINICI COME POTENTI INBITORI DELLA POMPA D’EFFLUSSO NorA DELLO S. aureus 39
Selective anti-BVDV acridones as new potential anti-HCV agents 39
Design, Synthesis, and Evaluation of WC5 Analogues as Inhibitors of Human Cytomegalovirus Immediate-Early 2 Protein, a Promising Target for Anti-HCMV Treatment 39
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors 38
Boosting Effect of 2-Phenylquinoline Efflux Inhibitors in Combination with Macrolides against Mycobacterium smegmatis and Mycobacterium avium 38
Totale 7.816
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Categoria #
all - tutte 26.213
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 26.213
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/201942 0 0 0 0 0 0 0 0 0 0 32 10
2019/2020547 7 5 78 5 80 27 104 15 101 77 14 34
2020/20211.402 15 94 37 100 340 94 127 10 158 44 86 297
2021/20221.250 34 195 17 71 97 12 50 364 54 33 162 161
2022/20232.236 141 340 36 212 193 236 16 130 799 13 80 40
2023/20242.846 73 145 52 20 21 26 2.303 21 133 49 3 0
Totale 8.967